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Volume 113
Main
Pharmacological Research
Volume 113
Pharmacological Research
Volume 113
1
Pure Δ9-tetrahydrocannabivarin and a Cannabis sativa extract with high content in Δ9-tetrahydrocannabivarin inhibit nitrite production in murine peritoneal macrophages
Romano, Barbara
,
Pagano, Ester
,
Orlando, Pierangelo
,
Capasso, Raffaele
,
Cascio, Maria Grazia
,
Pertwee, Roger
,
Marzo, Vincenzo Di
,
Izzo, Angelo A.
,
Borrelli, Francesca
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 916 KB
Your tags:
english, 2016
2
Timing and crosstalk of glucocorticoid signaling with cytokines, neurotransmitters and growth factors
Arango-Lievano, Margarita
,
Jeanneteau, Freddy
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.71 MB
Your tags:
english, 2016
3
Screening of a composite library of clinically used drugs and well-characterized pharmacological compounds for cystathionine β-synthase inhibition identifies benserazide as a drug potentially suitable for repurposing for the experimental therapy of colon cancer
Druzhyna, Nadiya
,
Szczesny, Bartosz
,
Olah, Gabor
,
Módis, Katalin
,
Asimakopoulou, Antonia
,
Pavlidou, Athanasia
,
Szoleczky, Petra
,
Gerö, Domokos
,
Yanagi, Kazunori
,
Törö, Gabor
,
López-García, Isabel
,
Myr
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 5.07 MB
Your tags:
english, 2016
4
The novel cannabinoid antagonist SM-11 reduces hedonic aspect of food intake through a dopamine-dependent mechanism
Fois, G.R.
,
Fattore, L.
,
Murineddu, G.
,
Salis, A.
,
Pintore, G.
,
Asproni, B.
,
Pinna, G.A.
,
Diana, M.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 720 KB
Your tags:
english, 2016
5
Novel, selective EPO receptor ligands lacking erythropoietic activity reduce infarct size in acute myocardial infarction in rats
Kiss, Krisztina
,
Csonka, Csaba
,
Pálóczi, János
,
Pipis, Judit
,
Görbe, Anikó
,
Kocsis, Gabriella F.
,
Murlasits, Zsolt
,
Sárközy, Márta
,
Szűcs, Gergő
,
Holmes, Christopher P.
,
Pan, Yijun
,
Bhandari, Ashok
,
C
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 730 KB
Your tags:
english, 2016
6
Enzyme-responsive multistage vector for drug delivery to tumor tissue
Mi, Yu
,
Wolfram, Joy
,
Mu, Chaofeng
,
Liu, Xuewu
,
Blanco, Elvin
,
Shen, Haifa
,
Ferrari, Mauro
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 888 KB
Your tags:
english, 2016
7
The hallucinogen d-lysergic diethylamide (LSD) decreases dopamine firing activity through 5-HT1A, D2 and TAAR1 receptors
De Gregorio, Danilo
,
Posa, Luca
,
Ochoa-Sanchez, Rafael
,
McLaughlin, Ryan
,
Maione, Sabatino
,
Comai, Stefano
,
Gobbi, Gabriella
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 1.75 MB
Your tags:
english, 2016
8
Genotype-dependent responsivity to inflammatory pain: A role for TRPV1 in the periaqueductal grey
Madasu, Manish K.
,
Okine, Bright N.
,
Olango, Weredeselam M.
,
Rea, Kieran
,
Lenihan, Róisín
,
Roche, Michelle
,
Finn, David P.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.19 MB
Your tags:
english, 2016
9
Hydrogen sulfide compensates nitric oxide deficiency in murine corpus cavernosum
Yetik-Anacak, Günay
,
Dikmen, Aycan
,
Coletta, Ciro
,
Mitidieri, Emma
,
Dereli, Mehmet
,
Donnarumma, Erminia
,
d'Emmanuele di Villa Bianca, Roberta
,
Sorrentino, Raffaella
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 955 KB
Your tags:
english, 2016
10
Regulation and role of endogenously produced hydrogen sulfide in angiogenesis
Katsouda, Antonia
,
Bibli, Sofia-Iris
,
Pyriochou, Anastasia
,
Szabo, Csaba
,
Papapetropoulos, Andreas
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.68 MB
Your tags:
english, 2016
11
Stimulation of the histamine 4 receptor upregulates thymic stromal lymphopoietin (TSLP) in human and murine keratinocytes
Schaper, Katrin
,
Rossbach, Kristine
,
Köther, Brigitta
,
Stark, Holger
,
Kietzmann, Manfred
,
Werfel, Thomas
,
Gutzmer, Ralf
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 1.11 MB
Your tags:
english, 2016
12
Sex-specific pharmacological modulation of autophagic process in human umbilical artery smooth muscle cells
Campesi, Ilaria
,
Occhioni, Stefano
,
Capobianco, Giampiero
,
Fois, Marco
,
Montella, Andrea
,
Dessole, Salvatore
,
Franconi, Flavia
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.18 MB
Your tags:
english, 2016
13
Pharmacological inhibition of fatty acid amide hydrolase attenuates social behavioural deficits in male rats prenatally exposed to valproic acid
Kerr, Daniel M.
,
Gilmartin, Aoife
,
Roche, Michelle
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 820 KB
Your tags:
english, 2016
14
Celastrol modulates inflammation through inhibition of the catalytic activity of mediators of arachidonic acid pathway: Secretory phospholipase A2 group IIA, 5-lipoxygenase and cyclooxygenase-2
Joshi, Vikram
,
Venkatesha, Shivaprasad H.
,
Ramakrishnan, Chandrasekaran
,
Nanjaraj Urs, Ankanahalli N.
,
Hiremath, Vilas
,
Moudgil, Kamal D.
,
Velmurugan, Devadasan
,
Vishwanath, Bannikuppe Sannanaik
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 3.22 MB
Your tags:
english, 2016
15
Signaling effects of sodium hydrosulfide in healthy donor peripheral blood mononuclear cells
Sulen, André
,
Gullaksen, Stein-Erik
,
Bader, Lucius
,
McClymont, David W.
,
Skavland, Jørn
,
Gavasso, Sonia
,
Gjertsen, Bjørn T.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 3.87 MB
Your tags:
english, 2016
16
The novel H2S-donor 4-carboxyphenyl isothiocyanate promotes cardioprotective effects against ischemia/reperfusion injury through activation of mitoKATP channels and reduction of oxidative stress
Testai, Lara
,
Marino, Alice
,
Piano, Ilaria
,
Brancaleone, Vincenzo
,
Tomita, Kengo
,
Di Cesare Mannelli, Lorenzo
,
Martelli, Alma
,
Citi, Valentina
,
Breschi, Maria C.
,
Levi, Roberto
,
Gargini, Claudia
,
Bucc
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 1.82 MB
Your tags:
english, 2016
17
Palmitoylethanolamide protects mice against 6-OHDA-induced neurotoxicity and endoplasmic reticulum stress: In vivo and in vitro evidence
Avagliano, Carmen
,
Russo, Roberto
,
De Caro, Carmen
,
Cristiano, Claudia
,
La Rana, Giovanna
,
Piegari, Giuseppe
,
Paciello, Orlando
,
Citraro, Rita
,
Russo, Emilio
,
De Sarro, Giovambattista
,
Meli, Rosaria
,
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 3.77 MB
Your tags:
english, 2016
18
Modulation of monocytes by bioactive lipid anandamide in multiple sclerosis involves distinct Toll-like receptors
Chiurchiù, Valerio
,
Leuti, Alessandro
,
Cencioni, Maria Teresa
,
Albanese, Maria
,
De Bardi, Marco
,
Bisogno, Tiziana
,
Centonze, Diego
,
Battistini, Luca
,
Maccarrone, Mauro
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 1.53 MB
Your tags:
english, 2016
19
Histone deacetylase inhibitors: Future therapeutics for insulin resistance and type 2 diabetes
Sharma, Sorabh
,
Taliyan, Rajeev
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 893 KB
Your tags:
english, 2016
20
Graduate Education in Pharmacology: Addressing the need for specialized training for pharmaceutical and biotechnology careers
Barrett, James E.
,
McGonigle, Paul
,
Clark, Janet E.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 253 KB
Your tags:
english, 2016
21
Antinociceptive effects of the 6-O-sulfate ester of morphine in normal and diabetic rats: Comparative role of mu- and delta-opioid receptors
Yadlapalli, Jai Shankar K.
,
Ford, Benjamin M.
,
Ketkar, Amit
,
Wan, Anqi
,
Penthala, Narasimha R.
,
Eoff, Robert L.
,
Prather, Paul L.
,
Dobretsov, Maxim
,
Crooks, Peter A.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 1.74 MB
Your tags:
english, 2016
22
Ibrutinib inhibition of Bruton protein-tyrosine kinase (BTK) in the treatment of B cell neoplasms
Roskoski, Robert
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.37 MB
Your tags:
english, 2016
23
Autoimmune therapeutic chloroquine lowers blood pressure and improves endothelial function in spontaneously hypertensive rats
McCarthy, Cameron G.
,
Wenceslau, Camilla F.
,
Goulopoulou, Styliani
,
Ogbi, Safia
,
Matsumoto, Takayuki
,
Webb, R.Clinton
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 850 KB
Your tags:
english, 2016
24
Bisphenol A induces hypothalamic down-regulation of the the cannabinoid receptor 1 and anorexigenic effects in male mice
Suglia, Antonio
,
Chianese, Rosanna
,
Migliaccio, Marina
,
Ambrosino, Concetta
,
Fasano, Silvia
,
Pierantoni, Riccardo
,
Cobellis, Gilda
,
Chioccarelli, Teresa
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 952 KB
Your tags:
english, 2016
25
Both the H2S biosynthesis inhibitor aminooxyacetic acid and the mitochondrially targeted H2S donor AP39 exert protective effects in a mouse model of burn injury
Ahmad, Akbar
,
Szabo, Csaba
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.36 MB
Your tags:
english, 2016
26
Managing epilepsy in the third millenium: Recent achievements and future perspectives
De Sarro, Giovambattista
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 230 KB
Your tags:
english, 2016
27
Chitosan oligosaccharide suppresses synovial inflammation via AMPK activation: An in vitro and in vivo study
Kunanusornchai, Wanlop
,
Witoonpanich, Bhee
,
Pichyangkura, Rath
,
Chatsudthipong, Varanuj
,
Muanprasat, Chatchai
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.65 MB
Your tags:
english, 2016
28
Novel α-substituted tropolones promote potent and selective caspase-dependent leukemia cell apoptosis
Li, Jin
,
Falcone, Eric R.
,
Holstein, Sarah A.
,
Anderson, Amy C.
,
Wright, Dennis L.
,
Wiemer, Andrew J.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 3.06 MB
Your tags:
english, 2016
29
Risk of infections during the first year of life after in utero exposure to drugs acting on immunity: A population-based cohort study
Palosse-Cantaloube, Lucie
,
Hurault-Delarue, Caroline
,
Beau, Anna-Belle
,
Montastruc, Jean-Louis
,
Lacroix, Isabelle
,
Damase-Michel, Christine
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 513 KB
Your tags:
english, 2016
30
Targeting the complex interactions between microbiota, host epithelial and immune cells in inflammatory bowel disease
Hirata, Yoshihiro
,
Ihara, Sozaburo
,
Koike, Kazuhiko
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.31 MB
Your tags:
english, 2016
31
Doxorubicin loaded gold nanoparticles: Implication of passive targeting on anticancer efficacy
Dhamecha, Dinesh
,
Jalalpure, Sunil
,
Jadhav, Kiran
,
Jagwani, Satveer
,
Chavan, Ramesh
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.51 MB
Your tags:
english, 2016
32
Metformin: An anti-diabetic drug to fight cancer
Daugan, Marie
,
Dufaÿ Wojcicki, Amélie
,
d’Hayer, Benoit
,
Boudy, Vincent
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 1.83 MB
Your tags:
english, 2016
33
Hydrogen sulfide donors alleviate itch secondary to the activation of type-2 protease activated receptors (PAR-2) in mice
Coavoy-Sánchez, S.A.
,
Rodrigues, L.
,
Teixeira, S.A.
,
Soares, A.G.
,
Torregrossa, R.
,
Wood, M.E.
,
Whiteman, M.
,
Costa, S.K.P.
,
Muscará, M.N.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.43 MB
Your tags:
english, 2016
34
Berberine and inflammatory bowel disease: A concise review
Habtemariam, Solomon
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.04 MB
Your tags:
english, 2016
35
Forty years later: Mitochondria as therapeutic targets in muscle diseases
Zulian, Alessandra
,
Schiavone, Marco
,
Giorgio, Valentina
,
Bernardi, Paolo
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.72 MB
Your tags:
english, 2016
36
Ligand autoradiographical quantification of histamine H3 receptor in human dementia with Lewy bodies
Lethbridge, Natasha L.
,
Chazot, Paul L.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 944 KB
Your tags:
english, 2016
37
Medication use and survival in diabetic patients with kidney cancer: A population-based cohort study
Nayan, Madhur
,
Macdonald, Erin M.
,
Juurlink, David N.
,
Austin, Peter C.
,
Finelli, Antonio
,
Kulkarni, Girish S.
,
Hamilton, Robert J.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 847 KB
Your tags:
english, 2016
38
The thiirane-based selective MT1-MMP/MMP2 inhibitor ND-322 reduces melanoma tumor growth and delays metastatic dissemination
Marusak, Charles
,
Bayles, Ian
,
Ma, Jun
,
Gooyit, Major
,
Gao, Ming
,
Chang, Mayland
,
Bedogni, Barbara
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 1.15 MB
Your tags:
english, 2016
39
Anti Xa oral anticoagulants inhibit in vivo platelet activation by modulating glycoprotein VI shedding
Pignatelli, Pasquale
,
Pastori, Daniele
,
Bartimoccia, Simona
,
Menichelli, Danilo
,
Vicario, Tommasa
,
Nocella, Cristina
,
Carnevale, Roberto
,
Violi, Francesco
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 1.03 MB
Your tags:
english, 2016
40
The paracrine control of vascular motion. A historical perspective
Nava, Eduardo
,
Llorens, Silvia
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 3.61 MB
Your tags:
english, 2016
41
The endocannabinoid anandamide causes endothelium-dependent vasorelaxation in human mesenteric arteries
Stanley, Christopher P.
,
Hind, William H.
,
Tufarelli, Christina
,
O’Sullivan, Saoirse E.
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 1.52 MB
Your tags:
english, 2016
42
Pharmacogenomic analyzis of the responsiveness of gastrointestinal tumor cell lines to drug therapy: A transportome approach
Grañé-Boladeras, Natàlia
,
Pérez-Torras, Sandra
,
Lozano, Juan José
,
Romero, Marta R.
,
Mazo, Adela
,
Marín, José J.G.
,
Pastor-Anglada, Marçal
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 7.35 MB
Your tags:
english, 2016
43
H2S dependent and independent anti-inflammatory activity of zofenoprilat in cells of the vascular wall
Monti, Martina
,
Terzuoli, Erika
,
Ziche, Marina
,
Morbidelli, Lucia
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 3.63 MB
Your tags:
english, 2016
44
Dibenzo[b,f][1,4]oxazepines and dibenzo[b,e]oxepines: Influence of the chlorine substitution pattern on the pharmacology at the H1R, H4R, 5-HT2AR and other selected GPCRs
Naporra, Franziska
,
Gobleder, Susanne
,
Wittmann, Hans-Joachim
,
Spindler, Julia
,
Bodensteiner, Michael
,
Bernhardt, Günther
,
Hübner, Harald
,
Gmeiner, Peter
,
Elz, Sigurd
,
Strasser, Andrea
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 3.81 MB
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english, 2016
45
A novel slow-releasing hydrogen sulfide donor, FW1256, exerts anti-inflammatory effects in mouse macrophages and in vivo
Huang, Caleb Weihao
,
Feng, Wei
,
Peh, Meng Teng
,
Peh, Kaye
,
Dymock, Brian W.
,
Moore, Philip Keith
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 3.14 MB
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english, 2016
46
Disodium cromoglycate inhibits asthma-like features induced by sphingosine-1-phosphate
Roviezzo, Fiorentina
,
Sorrentino, Rosalinda
,
Iacono, Valentina Mattera
,
Brancaleone, Vincenzo
,
Terlizzi, Michela
,
Riemma, Maria Antonietta
,
Bertolino, Antonio
,
Rossi, Antonietta
,
Matteis, Maria
,
Spazi
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 2.40 MB
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english, 2016
47
Editorial Board
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 53 KB
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english, 2016
48
Editorial Board
Journal:
Pharmacological Research
Year:
2016
Language:
english
File:
PDF, 21 KB
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english, 2016
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