Australian Journal of Chemistry

1

Fragment-based Drug Discovery: the Shape of Things to Come

Drysdale, Martin J.

Journal:

Year:

2013

Language:

english

File:

PDF, 712 KB

english, 2013

2

A Mild and Convenient Synthesis of 1,2,3-Triiodoarenes via Consecutive Iodination/Diazotization/Iodination Strategy

Al-Zoubi, Raed M., Futouh, Hassan Abul, McDonald, Robert

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 536 KB

english, 2013

3

Fragment Screening on Staphylococcus aureus HPPK – a Folate Pathway Target

Chhabra, Sandeep, Dolezal, Olan, Hattarki, Meghan, Peat, Thomas S., Simpson, Jamie S., Swarbrick, James D.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 838 KB

english, 2013

4

Fragment-Based Drug Discovery

Norton, Raymond S.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 111 KB

english, 2013

5

Construction of the CSIRO Fragment Library

Francis, Craig L., Kenny, Peter W., Dolezal, Olan, Saubern, Simon, Kruger, Megan, Savage, G. Paul, Peat, Thomas S., Ryan, John H.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 1.19 MB

english, 2013

6

Design and Evaluation of the Performance of an NMR Screening Fragment Library

Doak, Bradley C., Morton, Craig J., Simpson, Jamie S., Scanlon, Martin J.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 456 KB

english, 2013

7

Fragment Screening by Native State Mass Spectrometry

Poulsen, Sally-Ann

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 387 KB

english, 2013

8

PAINS: Relevance to Tool Compound Discovery and Fragment-Based Screening

Baell, Jonathan B., Ferrins, Lori, Falk, Hendrik, Nikolakopoulos, George

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 970 KB

english, 2013

9

Synthesis, Characterisation, and X-Ray Crystal Structures of 8-Hydroxyquinoline Complexes of Group IV Metal Alkoxides

Armaghan, Mahsa, Mirzaee, Mahdi, Norouzi, Mahmood, Amini, Mostafa M., Khavasi, Hamid Reza

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 618 KB

english, 2013

10

Interrogating Fragments Using a Protein Thermal Shift Assay

McMahon, Róisín M., Scanlon, Martin J., Martin, Jennifer L.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 255 KB

english, 2013

11

Characterization Methods for Starch-Based Materials: State of the Art and Perspectives

Wu, Alex C., Witt, Torsten, Gilbert, Robert G.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 1.14 MB

english, 2013

12

Development of Inhibitors of Plasmodium falciparum Apical Membrane Antigen 1 Based on Fragment Screening

Lim, San Sui, Debono, Cael O., MacRaild, Christopher A., Chandrashekaran, Indu R., Dolezal, Olan, Anders, Robin F., Simpson, Jamie S., Scanlon, Martin J., Devine, Shane M., Scammells, Peter J., Norton

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 990 KB

english, 2013

13

Al(OTf)3 Catalysed Friedel-Crafts Michael Type Addition of Indoles to α,β-Unsaturated Ketones with PEG-200 as Recyclable Solvent

Gohain, Mukut, Jacobs, Jc, Marais, Charlene, Bezuidenhoudt, Barend C. B.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 441 KB

english, 2013

14

RAFT Polymerization of Monomers with Highly Disparate Reactivities: Use of a Single RAFT Agent and the Synthesis of Poly(styrene-block-vinyl acetate)

Dayter, Lily A., Murphy, Kate A., Shipp, Devon A.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 819 KB

english, 2013

15

Methoxy-Poly(ethylene glycol)-block-Poly(ε-caprolactone) Bearing Pendant Aldehyde Groups as pH-Responsive Drug Delivery Carrier

Ma, Gejun, Li, Deshan, Wang, Ji, Zhang, Xuefei, Tang, Haoyu

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 887 KB

english, 2013

16

A Coumarin Fluorescent Probe for Ca2+ Containing Aza-Crown Ether Unit

Yan, Li-Qiang, Xie, Min-Sui, Peng, Ming-Sheng, Liu, Wei

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 316 KB

english, 2013

17

Detection and Prevention of Aggregation-based False Positives in STD-NMR-based Fragment Screening

Vom, Amelia, Headey, Stephen, Wang, Geqing, Capuano, Ben, Yuriev, Elizabeth, Scanlon, Martin J., Simpson, Jamie S.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 540 KB

english, 2013

19

Blind Man’s Bluff – Elaboration of Fragment Hits in the Absence of Structure for the Development of Antitrypsin Deficiency Inhibitors

Headey, Stephen J., Pearce, Mary C., Scanlon, Martin J., Bottomley, Stephen P.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 723 KB

english, 2013

20

Fragment Screening for the Modelling Community: SPR, ITC, and Crystallography

Dolezal, Olan, Doughty, Larissa, Hattarki, Meghan K., Fazio, Vincent J., Caradoc-Davies, Tom T., Newman, Janet, Peat, Thomas S.

Journal:

Australian Journal of Chemistry

Year:

2013

Language:

english

File:

PDF, 2.36 MB

english, 2013

Volume 66; Issue 12

Fragment-based Drug Discovery: the Shape of Things to Come

A Mild and Convenient Synthesis of 1,2,3-Triiodoarenes via Consecutive Iodination/Diazotization/Iodination Strategy

Fragment Screening on Staphylococcus aureus HPPK – a Folate Pathway Target

Fragment-Based Drug Discovery

Construction of the CSIRO Fragment Library

Design and Evaluation of the Performance of an NMR Screening Fragment Library

Fragment Screening by Native State Mass Spectrometry

PAINS: Relevance to Tool Compound Discovery and Fragment-Based Screening

Synthesis, Characterisation, and X-Ray Crystal Structures of 8-Hydroxyquinoline Complexes of Group IV Metal Alkoxides

Interrogating Fragments Using a Protein Thermal Shift Assay

Characterization Methods for Starch-Based Materials: State of the Art and Perspectives

Development of Inhibitors of Plasmodium falciparum Apical Membrane Antigen 1 Based on Fragment Screening

Al(OTf)3 Catalysed Friedel-Crafts Michael Type Addition of Indoles to α,β-Unsaturated Ketones with PEG-200 as Recyclable Solvent

RAFT Polymerization of Monomers with Highly Disparate Reactivities: Use of a Single RAFT Agent and the Synthesis of Poly(styrene-block-vinyl acetate)

Methoxy-Poly(ethylene glycol)-block-Poly(ε-caprolactone) Bearing Pendant Aldehyde Groups as pH-Responsive Drug Delivery Carrier

A Coumarin Fluorescent Probe for Ca2+ Containing Aza-Crown Ether Unit

Table of Contents

Detection and Prevention of Aggregation-based False Positives in STD-NMR-based Fragment Screening

Blind Man’s Bluff – Elaboration of Fragment Hits in the Absence of Structure for the Development of Antitrypsin Deficiency Inhibitors

Fragment Screening for the Modelling Community: SPR, ITC, and Crystallography