Volume 85; Issue 9

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Biochemical Pharmacology
Volume 85; Issue 9

Biochemical Pharmacology

Volume 85; Issue 9

1

Catalytic-site conformational equilibrium in nerve-agent adducts of acetylcholinesterase: Possible implications for the HI-6 antidote substrate specificity

Artursson, Elisabet, Andersson, Per Ola, Akfur, Christine, Linusson, Anna, Börjegren, Susanne, Ekström, Fredrik

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 408 KB

english, 2013

2

Parguerenes: Marine red alga bromoditerpenes as inhibitors of P-glycoprotein (ABCB1) in multidrug resistant human cancer cells

Huang, Xiao-cong, Sun, Yue-Li, Salim, Angela A., Chen, Zhe-Sheng, Capon, Robert J.

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 857 KB

english, 2013

3

Discovery of a new small-molecule inhibitor of p53–MDM2 interaction using a yeast-based approach

Leão, Mariana, Pereira, Clara, Bisio, Alessandra, Ciribilli, Yari, Paiva, Ana M., Machado, Neuza, Palmeira, Andreia, Fernandes, Miguel X., Sousa, Emília, Pinto, Madalena, Inga, Alberto, Saraiva, Lucíl

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 1.16 MB

english, 2013

4

Sulforaphane enhances Nrf2 expression in prostate cancer TRAMP C1 cells through epigenetic regulation

Zhang, Chengyue, Su, Zheng-Yuan, Khor, Tin Oo, Shu, Limin, Kong, Ah-Ng Tony

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 736 KB

english, 2013

5

Betulinic acid alleviates non-alcoholic fatty liver by inhibiting SREBP1 activity via the AMPK–mTOR–SREBP signaling pathway

Quan, Hai Yan, Kim, Do Yeon, Kim, Soo Jung, Jo, Hee Kyung, Kim, Go Woon, Chung, Sung Hyun

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 1.64 MB

english, 2013

6

Modulation of A-type K+ channels by the short-chain cobrotoxin through the protein kinase C-delta isoform decreases membrane excitability in dorsal root ganglion neurons

Guo, Qiang, Jiang, You-Jing, Jin, Hong, Jiang, Xing-Hong, Gu, Bo, Zhang, Yi-Ming, Wang, Jian-Gong, Qin, Zheng-Hong, Tao, Jin

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 1.19 MB

english, 2013

7

SIRT1 inhibits NADPH oxidase activation and protects endothelial function in the rat aorta: Implications for vascular aging

Zarzuelo, María José, López-Sepúlveda, Rocío, Sánchez, Manuel, Romero, Miguel, Gómez-Guzmán, Manuel, Ungvary, Zoltan, Pérez-Vizcaíno, Francisco, Jiménez, Rosario, Duarte, Juan

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 1.25 MB

english, 2013

8

Magnolol suppresses hypoxia-induced angiogenesis via inhibition of HIF-1α/VEGF signaling pathway in human bladder cancer cells

Chen, Meng-Chuan, Lee, Chi-Feng, Huang, Wen-Hsin, Chou, Tz-Chong

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 1.76 MB

english, 2013

9

Anti-diabetic and anti-lipidemic effects of chlorogenic acid are mediated by ampk activation

Ong, Khang Wei, Hsu, Annie, Tan, Benny Kwong Huat

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 2.37 MB

english, 2013

10

Chemical informatics uncovers a new role for moexipril as a novel inhibitor of cAMP phosphodiesterase-4 (PDE4)

Cameron, Ryan T., Coleman, Ryan G., Day, Jon P., Yalla, Krishna C., Houslay, Miles D., Adams, David R., Shoichet, Brian K., Baillie, George S.

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 1.23 MB

english, 2013

11

Tryptophan hydroxylase-2: An emerging therapeutic target for stress disorders

Chen, Guo-Lin, Miller, Gregory M.

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 325 KB

english, 2013

12

Beneficial effect of the non-psychotropic plant cannabinoid cannabigerol on experimental inflammatory bowel disease

Borrelli, Francesca, Fasolino, Ines, Romano, Barbara, Capasso, Raffaele, Maiello, Francesco, Coppola, Diana, Orlando, Pierangelo, Battista, Giovanni, Pagano, Ester, Di Marzo, Vincenzo, Izzo, Angelo A.

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 2.07 MB

english, 2013

13

Editorial Board

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 34 KB

english, 2013

14

Modulation of mitochondrial glutathione status and cellular energetics in primary cultures of proximal tubular cells from remnant kidney of uninephrectomized rats

Benipal, Bavneet, Lash, Lawrence H.

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 1.54 MB

english, 2013

15

A high-throughput-compatible, fluorescence anisotropy-based assay for ATP-dependent supercoiled DNA relaxation by human topoisomerase IIα

Shapiro, Adam B.

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 615 KB

english, 2013

16

Inhibition of gastric tumor growth by a novel Hsp90 inhibitor

Lu, Chunwan, Liu, Di, Jin, Jing, Deokar, Hemantkumar, Zhang, Yi, Buolamwini, John K., Yu, Xiaoming, Yan, Chunhong, Chen, Xiaoguang

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 2.03 MB

english, 2013

17

Pro-inflammatory and pathogenic properties of Annexin-A1: The whole is greater than the sum of its parts

D’Acquisto, Fulvio, Piras, Giuseppa, Rattazzi, Lorenza

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 377 KB

english, 2013

18

Carbonyl reduction of triadimefon by human and rodent 11β-hydroxysteroid dehydrogenase 1

Meyer, Arne, Vuorinen, Anna, Zielinska, Agnieszka E., Da Cunha, Thierry, Strajhar, Petra, Lavery, Gareth G., Schuster, Daniela, Odermatt, Alex

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 868 KB

english, 2013

19

The second extracellular loop of GPCRs determines subtype-selectivity and controls efficacy as evidenced by loop exchange study at A2 adenosine receptors

Seibt, Benjamin F., Schiedel, Anke C., Thimm, Dominik, Hinz, Sonja, Sherbiny, Farag F., Müller, Christa E.

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 2.27 MB

english, 2013

20

RO4938581, a GABAAα5 modulator, displays strong CYP1A2 autoinduction properties in rats

Bundgaard, Christoffer, Badolo, Lassina, Redrobe, John P.

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 413 KB

english, 2013

21

Molecular aspects of cancer cell resistance to chemotherapy

Rebucci, Magali, Michiels, Carine

Journal:

Biochemical Pharmacology

Year:

2013

Language:

english

File:

PDF, 858 KB

english, 2013