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Volume 11; Issue 2

Bioorganic & Medicinal Chemistry

Volume 11; Issue 2

1

A ribozyme with michaelase activity: Synthesis of the substrate precursors

Alexander Eisenführ, Paramjit S Arora, Gerhard Sengle, Leo R Takaoka, James S Nowick, Michael Famulok

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 489 KB

english, 2003

2

Anti-MRSA cephems. Part 2: C-7 cinnamic acid derivatives

Dane M. Springer, Bing-Yu Luh, Jason Goodrich, Joanne J. Bronson

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 345 KB

english, 2003

3

Synthesis of Solution-Phase Combinatorial Library of 4,6-Diamino-1,2-dihydro-1,3,5-triazine and Identification of New Leads Against A16V+S108T Mutant Dihydrofolate Reductase of Plasmodium falciparum

Tirayut Vilaivan, Neungruthai Saesaengseerung, Deanpen Jarprung, Sumalee Kamchonwongpaisan, Worachart Sirawaraporn, Yongyuth Yuthavong

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 234 KB

english, 2003

4

N-Thiolated β-Lactam Antibacterials: Defining the Role of Unsaturation in the C4 Side Chain

Cristina Coates, Timothy E Long, Edward Turos, Sonja Dickey, Daniel V Lim

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 125 KB

english, 2003

5

Inhibition of dipeptidyl peptidase IV (DPP IV) by 2-(2-amino-1-fluoro-propylidene)-cyclopentanecarbonitrile, a fluoroolefin containing peptidomimetic

Kake Zhao, Dong Sung Lim, Takashi Funaki, John T. Welch

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 233 KB

english, 2003

6

Synthesis and Structure–Activity Relationship Studies of Novel 2-Diarylethyl Substituted (2-Carboxycycloprop-1-yl)glycines as High-Affinity Group II Metabotropic Glutamate Receptor Ligands

Ulrik S Sørensen, Thomas J Bleisch, Anne E Kingston, Rebecca A Wright, Bryan G Johnson, Darryle D Schoepp, Paul L Ornstein

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 250 KB

english, 2003

7

2,3-Diaryl-5-anilino[1,2,4]thiadiazoles as melanocortin MC4 receptor agonists and their effects on feeding behavior in rats

Kevin Pan, Malcolm K Scott, Daniel H.S Lee, Louis J Fitzpatrick, Jeffery J Crooke, Ralph A Rivero, Daniel I Rosenthal, Anil H Vaidya, Boyu Zhao, Allen B Reitz

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 353 KB

english, 2003

8

Inside Front Cover

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 54 KB

english, 2003

9

Tricyclic Pyrazoles. Part 1: Synthesis and Biological Evaluation of Novel 1,4-Dihydroindeno[1,2-c]pyrazol-based Ligands for CB1and CB2 Cannabinoid Receptors

Jean-Mario Mussinu, Stefania Ruiu, Antonio C Mulè, Amedeo Pau, Mauro A.M Carai, Giovanni Loriga, Gabriele Murineddu, Gérard A Pinna

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 265 KB

english, 2003

10

Anti-MRSA cephems. Part 3: Additional C-7 acid derivatives

Dane M Springer, Bing-Yu Luh, Jason T Goodrich, Joanne J Bronson

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 266 KB

english, 2003

11

Synthesis of 2-(5-Bromo-2,3-dimethoxyphenyl)-5-(aminomethyl)-1H-pyrrole analogues and their binding affinities for dopamine D2, D3, and D4 receptors

Robert H Mach, Yunsheng Huang, Rebekah A Freeman, Li Wu, Suwanna Blair, Robert R Luedtke

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 221 KB

english, 2003

12

New minor taxanes analogues from the needles of Taxus canadensis

Qing Wen Shi, Françoise Sauriol, Orval Mamer, Lolita O Zamir

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 203 KB

english, 2003

13

Synthesis and pharmacological characterisation of 2,4-Dicarboxy-pyrroles as selective non-Competitive mGluR1 antagonists

Fabrizio Micheli, Romano Di Fabio, Paolo Cavanni, Joseph M Rimland, Anna Maria Capelli, Cristiano Chiamulera, Mauro Corsi, Corrado Corti, Daniele Donati, Aldo Feriani, Francesco Ferraguti, Micaela Maf

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 394 KB

english, 2003

14

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 188 KB

english, 2003