Volume 13; Issue 10

Bioorganic & Medicinal Chemistry

Volume 13; Issue 10

1

Synthesis and biological evaluation of N-{4-[5-(2,4-diamino-6-oxo-1,6-dihydropyrimidin-5-yl)-2-(2,2,2-trifluoroacetyl)pentyl]benzoyl}-l-glutamic acid as a potential inhibitor of GAR Tfase and the de novo purine biosynthetic pathway

Heng Cheng, Inkyu Hwang, Youhoon Chong, Ali Tavassoli, Michael E. Webb, Yan Zhang, Ian A. Wilson, Stephen J. Benkovic, Dale L. Boger

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 168 KB

english, 2005

2

Synthesis and biological evaluation of α- and γ-carboxamide derivatives of 10-CF3CO-DDACTHF

Youhoon Chong, Inkyu Hwang, Ali Tavassoli, Yan Zhang, Ian A. Wilson, Stephen J. Benkovic, Dale L. Boger

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 151 KB

english, 2005

3

Design, synthesis, and biological evaluation of 10-methanesulfonyl-DDACTHF, 10-methanesulfonyl-5-DACTHF, and 10-methylthio-DDACTHF as potent inhibitors of GAR Tfase and the de novo purine biosynthetic pathway

Heng Cheng, Youhoon Chong, Inkyu Hwang, Ali Tavassoli, Yan Zhang, Ian A. Wilson, Stephen J. Benkovic, Dale L. Boger

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 208 KB

english, 2005

4

Synthesis and antibody-binding studies of a series of parasite fuco-oligosaccharides

Anne-Marie M. van Roon, Begoña Aguilera, Francisco Cuenca, Alexandra van Remoortere, Gijsbert A. van der Marel, André M. Deelder, Herman S. Overkleeft, Cornelis H. Hokke

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 357 KB

english, 2005

5

Horseradish peroxidase-mediated aerobic and anaerobic oxidations of 3-alkylindoles

Ke-Qing Ling, Lawrence M. Sayre

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 229 KB

english, 2005

6

Novel anellated pyrazoloquinolin-3-ones: synthesis and in vitro BZR activity

Maria Grazia Ferlin, Gianfranco Chiarelotto, Stefano Dall’Acqua, Elisabetta Maciocco, Maria Paola Mascia, Maria Giuseppina Pisu, Giovanni Biggio

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 229 KB

english, 2005

7

Corrigendum to “Synthesis and activity of 1H-benzimidazole and 1H-benzotriazole derivatives as inhibitors of Acanthamoeba castellanii” [Bioorg. Med. Chem. 12 (2004) 2617]

Katarzyna Kopańska (née Zastąpiło), Andzelika Najda, Justyna Żebrowska, Lidia Chomicz, Janusz Piekarczyk, Przemysław Myjak, Maria Bretner

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 65 KB

english, 2005

8

Synthesis and evaluation of sphingoid analogs as inhibitors of sphingosine kinases

Jin-Wook Kim, Yong-Woo Kim, Yuichi Inagaki, You-A Hwang, Susumu Mitsutake, Yeon-Woo Ryu, Won Koo Lee, Hyun-Joon Ha, Chang-Seo Park, Yasuyuki Igarashi

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 449 KB

english, 2005

9

Syntheses of novel heterocycles as anticancer agents

Prem M.S. Chauhan, Cristina J.A. Martins, David C. Horwell

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 139 KB

english, 2005

10

An efficient preparation of polyanionic affinity agent and its evaluation for the measurement of glycated hemoglobin

Rajarathnam E. Reddy, You Pan, Donald D. Johnson, Yon-Yih Chen, Saul A. Datwyler, Michelle S. Hauptman, John K. Thottathil

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 148 KB

english, 2005

11

Two novel series of allocolchicinoids with modified seven membered B-rings: design, synthesis, inhibition of tubulin assembly and cytotoxicity

Frank Büttner, Silke Bergemann, Daniel Guénard, Ronald Gust, Gunther Seitz, Sylviane Thoret

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 296 KB

english, 2005

12

Biphenylquinuclidines as inhibitors of squalene synthase and growth of parasitic protozoa

Silvia Orenes Lorente, Rosario Gómez, Carmen Jiménez, Simon Cammerer, Vanessa Yardley, Kate de Luca-Fradley, Simon L. Croft, Luis M. Ruiz Perez, Julio Urbina, Dolores Gonzalez Pacanowska, Ian H. Gilbe

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 324 KB

english, 2005

13

Mutation of surface cysteine 374 to alanine in monoamine oxidase A alters substrate turnover and inactivation by cyclopropylamines

Ana Paula B. Vintém, Nigel T. Price, Richard B. Silverman, Rona R. Ramsay

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 304 KB

english, 2005

14

Cytotoxicities, cell cycle and caspase evaluations of 1,6-diaryl-3(Z)-hexen-1,5-diynes, 2-(6-aryl-3(Z)-hexen-1,5-diynyl)anilines and their derivatives

Chi-Fong Lin, Yu-Hsiang Lo, Ming-Chu Hsieh, Yi-Hua Chen, Jeh-Jeng Wang, Ming-Jung Wu

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 355 KB

english, 2005

15

Design, synthesis and cytotoxic effect of hydroxy- and 3-alkylaminopropoxy-9,10-anthraquinone derivatives

Chi-Huang Teng, Shen-Jeu Won, Chun-Nan Lin

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 225 KB

english, 2005

16

Synthesis and vasodilatory activity of new N-acylhydrazone derivatives, designed as LASSBio-294 analogues

Alexandre G. Silva, Gisele Zapata-Sudo, Arthur E. Kummerle, Carlos A.M. Fraga, Eliezer J. Barreiro, Roberto T. Sudo

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 243 KB

english, 2005

17

Synthesis of DEHP metabolites as biomarkers for GC–MS evaluation of phthalates as endocrine disrupters

Francesca Nuti, Sibylle Hildenbrand, Mario Chelli, Roman Wodarz, Anna Maria Papini

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 158 KB

english, 2005

18

Synthesis of phthalates of betulinic acid and betulin with cytotoxic activity

Miroslav Kvasnica, Jan Sarek, Eva Klinotova, Petr Dzubak, Marian Hajduch

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 168 KB

english, 2005

19

1,4-Dihydropyridine derivatives as calcium channel modulators: the role of 3-methoxy-flavone moiety

Roberta Budriesi, Alessandra Bisi, Pierfranco Ioan, Angela Rampa, Silvia Gobbi, Federica Belluti, Lorna Piazzi, Piero Valenti, Alberto Chiarini

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 202 KB

english, 2005

20

Structure–affinity relationship studies on arylpiperazine derivatives related to quipazine as serotonin transporter ligands. Molecular basis of the selectivity SERT/5HT3 receptor

Andrea Cappelli, Germano Giuliani, Andrea Gallelli, Salvatore Valenti, Maurizio Anzini, Laura Mennuni, Francesco Makovec, Aroldo Cupello, Salvatore Vomero

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 142 KB

english, 2005

21

Synthesis and antiprotozoan evaluation of new alkyl-linked bis(2-thioxo-[1,3,5]thiadiazinan-3-yl) carboxylic acids

Julieta Coro, Rolando Pérez, Hortensia Rodríguez, Margarita Suárez, Celeste Vega, Miriam Rolón, David Montero, Juan José Nogal, Alicia Gómez-Barrio

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 182 KB

english, 2005

22

Linear indices of the ‘macromolecular graph’s nucleotides adjacency matrix’ as a promising approach for bioinformatics studies. Part 1: Prediction of paromomycin’s affinity constant with HIV-1 Ψ-RNA packaging region

Yovani Marrero Ponce, Juan A. Castillo Garit, Delvin Nodarse

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 446 KB

english, 2005

23

Electrophilicity as a possible descriptor for toxicity prediction

D.R. Roy, R. Parthasarathi, B. Maiti, V. Subramanian, P.K. Chattaraj

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 159 KB

english, 2005

24

Structure–activity relationships of tyrosinase inhibitory combinatorial library of 2,5-disubstituted-1,3,4-oxadiazole analogues

Mahmud Tareq Hassan Khan, Muhammad Iqbal Choudhary, Khalid Mohammed Khan, Mubeen Rani, Atta-ur-Rahman

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 237 KB

english, 2005

25

Position-specific incorporation of a highly photodurable and blue-laser excitable fluorescent amino acid into proteins for fluorescence sensing

Hiroyuki Hamada, Naoko Kameshima, Aneta Szymańska, Katarzyna Wegner, Leszek Łankiewicz, Hiroaki Shinohara, Masumi Taki, Masahiko Sisido

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 288 KB

english, 2005

26

Differences between the structural requirements for ABA 8′-hydroxylase inhibition and for ABA activity

Kotomi Ueno, Yoshiharu Araki, Nobuhiro Hirai, Shigeki Saito, Masaharu Mizutani, Kanzo Sakata, Yasushi Todoroki

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 280 KB

english, 2005

27

Biocatalysed synthesis of β-O-glucosides from 9-fluorenon-2-carbohydroxyesters. Part 3: IFN-inducing and anti-HSV-2 properties

Stefano Alcaro, Adriana Arena, Rosaria Di Bella, Simonetta Neri, Rosaria Ottanà, Francesco Ortuso, Bernadette Pavone, Antonio Trincone, Maria Gabriella Vigorita

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 223 KB

english, 2005

28

Biotin-labeled abscisic acid as a probe for investigating abscisic acid binding sites on plasma membranes of barley aleurone protoplasts

Nobutaka Kitahata, Takeshi Nakano, Kazuyuki Kuchitsu, Shigeo Yoshida, Tadao Asami

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 169 KB

english, 2005

29

Volsurf analysis of carbapenem antibiotics

Munikumar Reddy Doddareddy, Joo Hwan Cha, Yong Seo Cho, Hun Yeong Koh, Kyung Ho Yoo, Dong Jin Kim, Ae Nim Pae

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 286 KB

english, 2005

30

Publisher’s note

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 223 KB

english, 2005

31

Editorial board

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 308 KB

english, 2005

32

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

File:

PDF, 187 KB

2005

33

Instructions to contributors

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 73 KB

english, 2005

34

Graphical contents list

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 558 KB

english, 2005

To build up a library is to create a life. It’s never just a random collection of books.

— Carlos María Domínguez

Official channel

Z-Library Desktop Launcher

Tor version

Z-Library

Z-Library Since 2009 support@1delivery.pm

EnglishРусскийEspañolItalianoελληνικάاللغة العربيةBahasa IndonesiaBahasa Malaysiaहिन्दीDeutschFrançaisPortuguêsУкраїнськаPolski中文繁體中文日本語Tiếng ViệtAzərbaycan DiliՀայոց լեզուภาษาไทยTürk Diliქართველიবাংলাپښتوతెలుగుاردو한국어SrpskiБългарски