Volume 18; Issue 24

Bioorganic & Medicinal Chemistry

Volume 18; Issue 24

1

Design, synthesis, and characterization of BK channel openers based on oximation of abietane diterpene derivatives

Yong-Mei Cui, Eriko Yasutomi, Yuko Otani, Katsutoshi Ido, Takashi Yoshinaga, Kohei Sawada, Tomohiko Ohwada

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.86 MB

english, 2010

2

ApoA-I mimetic peptides promote pre-β HDL formation in vivo causing remodeling of HDL and triglyceride accumulation at higher dose

Ester Carballo-Jane, Zhu Chen, Edward O’Neill, Jun Wang, Charlotte Burton, Ching H. Chang, Xun Chen, Suzanne Eveland, Betsy Frantz-Wattley, Karen Gagen, Brian Hubbard, Marina Ichetovkin, Silvi Luell,

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1014 KB

english, 2010

3

Convergent synthesis of fluorescence-labeled probes of Annonaceous acetogenins and visualization of their cell distribution

Naoto Kojima, Takekuni Morioka, Daisuke Urabe, Masahiro Yano, Yuki Suga, Naoyoshi Maezaki, Ayako Ohashi-Kobayashi, Yasuyuki Fujimoto, Masatomo Maeda, Takao Yamori, Takehiko Yoshimitsu, Tetsuaki Tanaka

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.39 MB

english, 2010

4

Structure based optimization of chromen-based TNF-α converting enzyme (TACE) inhibitors on S1′ pocket and their quantitative structure–activity relationship (QSAR) study

Jee Sun Yang, Kwangwoo Chun, Jung Eun Park, Misun Cho, Jeongjea Seo, Doona Song, Hongchul Yoon, Chun-Ho Park, Bo-Young Joe, Jong-Hee Choi, Myung-Hwa Kim, Gyoonhee Han

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 852 KB

english, 2010

5

The ODN probes conjugating the Cu(II) complex enhance the luminol chemiluminescence by assembling on the DNA template

Yosuke Taniguchi, Akiko Nitta, Sun Min Park, Akiko Kohara, Takahiro Uzu, Shigeki Sasaki

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 577 KB

english, 2010

6

Effect of Reishi polysaccharides on human stem/progenitor cells

Wan-Yu Chen, Wen-Bin Yang, Chi-Huey Wong, Daniel Tzu-Bi Shih

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.07 MB

english, 2010

7

A novel PET marker for in vivo quantification of myelination

Chunying Wu, Changning Wang, Daniela C. Popescu, Wenxia Zhu, Eduardo A. Somoza, Junqing Zhu, Allison G. Condie, Christopher A. Flask, Robert H. Miller, Wendy Macklin, Yanming Wang

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.10 MB

english, 2010

8

Investigating the activity of 2-substituted alkyl-6-(2,5-dioxopyrrolidin-1-yl)hexanoates as skin penetration enhancers

Katerina Brychtova, Radka Opatrilova, Ivan Raich, Danuta S. Kalinowski, Lenka Dvorakova, Lukas Placek, Jozef Csollei, Des R. Richardson, Josef Jampilek

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 870 KB

english, 2010

9

2-Aminohydroxamic acid derivatives as inhibitors of Bacillus cereus phosphatidylcholine preferred phospholipase C PC-PLCBc

Patricia González-Bulnes, Albert González-Roura, Daniel Canals, Antonio Delgado, Josefina Casas, Amadeu Llebaria

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 679 KB

english, 2010

10

High-throughput identification of antibacterials against methicillin-resistant Staphylococcus aureus (MRSA) and the transglycosylase

Ting-Jen Rachel Cheng, Ying-Ta Wu, Shih-Ting Yang, Kien-Hock Lo, Shao-Kang Chen, Yin-Hsuan Chen, Wen-I Huang, Chih-Hung Yuan, Chih-Wei Guo, Lin-Ya Huang, Kuo-Ting Chen, Hao-Wei Shih, Yih-Shyun E. Chen

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 8.65 MB

english, 2010

11

Novel lipophilic 7H-pyrido[1,2,3-de]-1,4-benzoxazine-6-carboxylic acid derivatives as potential antitumor agents: Improved synthesis and in vitro evaluation

Alexander Korolyov, Sandra Dorbes, Joëlle Azéma, Brigitte Guidetti, Mathieu Danel, Delphine Lamoral-Theys, Thierry Gras, Jacques Dubois, Robert Kiss, Robert Martino, Myriam Malet-Martino

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 474 KB

english, 2010

12

Corrigendum to “Natural and semisynthetic azaphilones as a new scaffold for Hsp90 inhibitors” [Bioorg. Med. Chem. 18 (2010) 6031–6043]

Loana Musso, Sabrina Dallavalle, Lucio Merlini, Adriana Bava, Gianluca Nasini, Sergio Penco, Giuseppe Giannini, Chiara Giommarelli, Andrea De Cesare, Valentina Zuco, Loredana Vesci, Claudio Pisano, Ma

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

File:

PDF, 109 KB

2010

13

Synthesis of 4β-N-polyaromatic substituted podophyllotoxins: DNA topoisomerase inhibition, anticancer and apoptosis-inducing activities

Ahmed Kamal, B. Ashwini Kumar, Paidakula Suresh, Satyam Kumar Agrawal, Gousia Chashoo, Shashank K. Singh, A.K. Saxena

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 484 KB

english, 2010

14

Angiotensin II receptor type 1 (AT1) selective nonpeptidic antagonists—A perspective

Prashant Naik, Prashant Murumkar, Rajani Giridhar, Mange Ram Yadav

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 6.83 MB

english, 2010

15

Design, synthesis, and biological evaluation of novel N-γ-carboline arylsulfonamides as anticancer agents

Jing Chen, Tao Liu, Rui Wu, Jianshu Lou, Ji Cao, Xiaowu Dong, Bo Yang, Qiaojun He, Yongzhou Hu

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 711 KB

english, 2010

16

Thermodynamic and NMR analysis of inhibitor binding to dihydrofolate reductase

Ihor Batruch, Eliott Javasky, Eric D. Brown, Michael G. Organ, Philip E. Johnson

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 906 KB

english, 2010

17

Discovery of 1H-benzo[d][1,2,3]triazol-1-yl 3,4,5-trimethoxybenzoate as a potential antiproliferative agent by inhibiting histone deacetylase

Jie Fu, Ying Yang, Xue-Wei Zhang, Wen-Jun Mao, Zhi-Ming Zhang, Hai-Liang Zhu

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 460 KB

english, 2010

18

Synthesis, binding studies and molecular modeling of novel cannabinoid receptor ligands

Noha A. Osman, Amr H. Mahmoud, Marco Allarà, Raimund Niess, Khaled A. Abouzid, Vincenzo Di Marzo, Ashraf H. Abadi

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.96 MB

english, 2010

19

A protected l-bromophosphonomethylphenylalanine amino acid derivative (BrPmp) for synthesis of irreversible protein tyrosine phosphatase inhibitors

Naresh S. Tulsi, A. Michael Downey, Christopher W. Cairo

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 365 KB

english, 2010

20

Synthesis and biological evaluation of new camptothecin derivatives obtained by modification of position 20

Elena Riva, Daniela Comi, Stella Borrelli, Francesco Colombo, Bruno Danieli, Jurgen Borlak, Lasse Evensen, James B. Lorens, Gabriele Fontana, Ornella Maria Gia, Lisa Dalla Via, Daniele Passarella

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 820 KB

english, 2010

21

Synthesis and pharmacological properties of novel hydrophilic 5-HT4 receptor antagonists

Bjarne Brudeli, Lise Román Moltzau, Kjetil Wessel Andressen, Kurt A. Krobert, Jo Klaveness, Finn Olav Levy

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.10 MB

english, 2010

22

Novel hybrids of 15-membered 8a- and 9a-azahomoerythromycin A ketolides and quinolones as potent antibacterials

Dražen Pavlović, Andrea Fajdetić, Stjepan Mutak

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 879 KB

english, 2010

23

Synthesis and structure–activity relationship of tetrahydropyrazolopyrimidine derivatives—A novel structural class of potent calcium-sensing receptor antagonists

Masato Yoshida, Akira Mori, Atsuhiro Inaba, Masahiro Oka, Haruhiko Makino, Masashi Yamaguchi, Hisashi Fujita, Tomohiro Kawamoto, Mika Goto, Hiroyuki Kimura, Atsuo Baba, Tsuneo Yasuma

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 570 KB

english, 2010

24

abeo-Abietanes from Teucrium polium roots as protective factors against oxidative stress

Antonio Fiorentino, Brigida D’Abrosca, Severina Pacifico, Monica Scognamiglio, Grazia D’Angelo, Pietro Monaco

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 417 KB

english, 2010

25

Editorial board

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 46 KB

english, 2010

26

Graphical contents list

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.24 MB

english, 2010

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