Volume 11; Issue 10

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Bioorganic & Medicinal Chemistry Letters
Volume 11; Issue 10

Bioorganic & Medicinal Chemistry Letters

Volume 11; Issue 10

1

The synthesis of amino-acid functionalized β-Carbolines as topoisomerase II inhibitors

Amy Morin Deveau, Marc A Labroli, Christine M Dieckhaus, Mary T Barthen, Kirsten S Smith, Timothy L Macdonald

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 820 KB

english, 2001

2

Diaryl ether inhibitors of farnesyl-protein transferase

Suzanne C. MacTough, S.Jane deSolms, Anthony W. Shaw, Marc T. Abrams, Terrence M. Ciccarone, Joseph P. Davide, Kelly A. Hamilton, John H. Hutchinson, Kenneth S. Koblan, Nancy E. Kohl, Robert B. Lobell

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 174 KB

english, 2001

3

Synthesis of polyamine derivatives Having non-hypotensive Ca2+-permeable AMPA receptor antagonist activity

Yoshiyuki Yoneda, Shinichi Kawajiri, Atushi Hasegawa, Fusako Kito, Sumie Katano, Emi Takano, Tetuya Mimura

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 143 KB

english, 2001

4

Synthesis and Antifungal Activities of Novel 1,3-β-d-Glucan Synthase Inhibitors. Part 2

Kazunao Masubuchi, Takehiro Okada, Masami Kohchi, Takeshi Murata, Masao Tsukazaki, Osamu Kondoh, Toshikazu Yamazaki, Yasuko Satoh, Yoshinori Ono, Toshiyuki Tsukaguchi, Kazuko Kobayashi, Naomi Ono, Tom

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 191 KB

english, 2001

5

Synthesis and evaluation of a difluoromethylene analogue of sphingomyelin as an inhibitor of sphingomyelinase

Tsutomu Yokomatsu, Hiroaki Takechi, Takeshi Akiyama, Shiroishi Shibuya, Takaaki Kominato, Shinji Soeda, Hiroshi Shimeno

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 243 KB

english, 2001

6

Synthesis and evaluation of hexahydrochrysene and tetrahydrobenzofluorene ligands for the estrogen receptor

Rosanna Tedesco, Michael K Youngman, Scott R Wilson, John A Katzenellenbogen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 225 KB

english, 2001

7

Phospho-azatyrosine, a less effective protein-tyrosine phosphatase substrate than phosphotyrosine

Terrence R Burke Jr., Zhu-Jun Yao, Bin Ye, Kengo Miyoshi, Akira Otaka, Li Wu, Zhong-Yin Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 102 KB

english, 2001

8

Liver cell specific targeting of peptide nucleic acid oligomers

Xiao Zhang, Carla G Simmons, David R Corey

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 567 KB

english, 2001

9

Pharmacological evaluation of a diarylmethylene-piperidine derivative: a new potent atypical antipsychotic?

Patrice Talaga, Alain Matagne, Henrik Klitgaard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 124 KB

english, 2001

10

Identification of a potent and selective oxytocin antagonist, from screening a fully encoded differential release combinatorial chemical library

Brian Evans, Adrian Pipe, Liz Clark, Martyn Banks

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 130 KB

english, 2001

11

Structure–activity relationship investigations of a potent and selective benzodiazepine oxytocin antagonist

Paul G Wyatt, Michael J Allen, Josie Chilcott, Gwen Hickin, Neil D Miller, Patrick M Woollard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 190 KB

english, 2001

12

Synthesis and biological evaluations of condensed pyridine and condensed pyrimidine-based HMG-CoA reductase inhibitors

Mikio Suzuki, Hiroshi Iwasaki, Yoshihiro Fujikawa, Mitsuaki Sakashita, Masaki Kitahara, Ryozo Sakoda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 165 KB

english, 2001

13

Structure–activity study of retinoid agonists bearing substituted dicarba-closo-dodecaborane. Relation between retinoidal activity and conformation of two aromatic nuclei

Yasuyuki Endo, Toru Iijima, Kyoko Yaguchi, Emiko Kawachi, Noriko Inoue, Hiroyuki Kagechika, Asako Kubo, Akiko Itai

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 817 KB

english, 2001

14

Modeling of the Binding Mode of a Non-covalent Inhibitor of the 20S Proteasome. Application to Structure-Based Analogue Design

Pascal Furet, Patricia Imbach, Peter Fürst, Marc Lang, Maria Noorani, Johann Zimmermann, Carlos Garcı́a-Echeverrı́a

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 1.77 MB

english, 2001

15

Design, Synthesis and Enzymatic Activity of Highly Selective Human Mitochondrial Thymidine Kinase Inhibitors

Stefano Manfredini, Pier G Baraldi, Elisa Durini, Luca Porcu, Angela Angusti, Silvia Vertuani, Nicola Solaroli, Erik De Clercq, Anna Karlsson, Jan Balzarini

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 152 KB

english, 2001

16

Powerful probes for glycosidases: novel, fluorescently tagged glycosidase inhibitors

Albin Hermetter, Hubert Scholze, Arnold E. Stütz, Stephen G. Withers, Tanja M. Wrodnigg

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 234 KB

english, 2001

17

Thiazole analogues of the NSAID indomethacin as selective COX-2 Inhibitors

Keith W. Woods, Richard W. McCroskey, Michael R. Michaelides, Carol K. Wada, Keren I. Hulkower, Randy L. Bell

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 145 KB

english, 2001

18

Ring-Constrained (N)-Methanocarba nucleosides as adenosine receptor agonists: independent 5′-Uronamide and 2′-deoxy modifications

Kyeong Lee, Gnana Ravi, Xiao-duo Ji, Victor E Marquez, Kenneth A Jacobson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 146 KB

english, 2001

19

Spirocyclic nonpeptide glycoprotein IIb–IIIa antagonists. Part 1: design of potent and specific 3,9-diazaspiro[5.5]undecanes

M.S Smyth, J Rose, M.M Mehrotra, J Heath, G Ruhter, T Schotten, J Seroogy, D Volkots, A Pandey, R.M Scarborough

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 168 KB

english, 2001

20

Spirocyclic nonpeptide glycoprotein IIb–IIIa antagonists. Part 2: design of potent antagonists containing the 3-azaspiro[5.5]undec-9-yl template

A. Pandey, J. Seroogy, D. Volkots, M.S. Smyth, J. Rose, M.M. Mehrotra, J. Heath, G. Ruhter, T. Schotten, R.M. Scarborough

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 176 KB

english, 2001

21

Anodic Oxidation of Ifosfamide and Cyclophosphamide: A Biomimetic Metabolism Model of the Oxazaphosphorinane Anticancer Drugs

Angelo Paci, Thierry Martens, Jacques Royer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 140 KB

english, 2001

22

A New Method for Chemoselective Conjugation of Unprotected Peptides to Dauno- and Doxorubicin

Paolo Ingallinella, Annalise Di Marco, Marina Taliani, Daniela Fattori, Antonello Pessi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 178 KB

english, 2001

23

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 323 KB

english, 2001

24

Contributors to this Issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 37 KB

english, 2001

25

Bioorganic & Medicinal Chemistry Letters

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 96 KB

english, 2001

26

A New Structural Class of Selective and Non-covalent Inhibitors of the Chymotrypsin-like Activity of the 20S Proteasome

C Garcı́a-Echeverrı́a, P Imbach, D France, P Fürst, M Lang, M Noorani, D Scholz, J Zimmermann, P Furet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 121 KB

english, 2001

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