Volume 11; Issue 13

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Bioorganic & Medicinal Chemistry Letters
Volume 11; Issue 13

Bioorganic & Medicinal Chemistry Letters

Volume 11; Issue 13

1

Enantioselective Synthesis and Complement Inhibitory Assay of A/B-Ring Partial Analogues of Oleanolic Acid

Haregewein Assefa, Alison Nimrod, Larry Walker, Robert Sindelar

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 211 KB

english, 2001

2

Quinoline-4-acetamides as sPLA2 inhibitors

Ying Liu, Yabing Feng, Renxiao Wang, Ying Gao, Luhua Lai

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 214 KB

english, 2001

3

Sequence-Selective Peptide Detection by Small Synthetic Chemosensors Selected from an Encoded Combinatorial Chemosensor Library

Edward James Iorio, Yuefei Shao, Chao-Tsen Chen, Holger Wagner, W.Clark Still

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 405 KB

english, 2001

4

Novel heteroaryl replacements of aromatic 3-tetrafluoroethoxy substituents in trifluoro-3-(tertiaryamino)-2-propanols as potent inhibitors of cholesteryl ester transfer protein

Mark A. Massa, Dale P. Spangler, Richard C. Durley, Brian S. Hickory, Daniel T. Connolly, Bryan J. Witherbee, Mark E. Smith, James A. Sikorski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 275 KB

english, 2001

5

Expedited discovery of second generation NK-1 antagonists: identification of a nonbasic aryloxy substituent

James E. Fritz, Philip A. Hipskind, Karen L. Lobb, James A. Nixon, Penny G. Threlkeld, Bruce D. Gitter, Carl L. McMillian, Stephen W. Kaldor

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 171 KB

english, 2001

6

Dibasic Inhibitors of Human Mast Cell Tryptase. Part 3: Identification of a Series of Potent and Selective Inhibitors Containing the Benzamidine Functionality

Jeffrey M. Dener, Kenneth D. Rice, William S. Newcomb, Vivian R. Wang, Wendy B. Young, Anthony R. Gangloff, Elaine Y.-L. Kuo, Lynne Cregar, Daun Putnam, Martin Wong

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 173 KB

english, 2001

7

Nucleoside Analogues as Highly Potent and Selective Inhibitors of Herpes Simplex Virus Thymidine Kinase

Joseph A Martin, Robert W Lambert, John H Merrett, Kevin E.B Parkes, Gareth J Thomas, Stewart J Baker, David J Bushnell, Julie E Cansfield, Stephen J Dunsdon, Andrew C Freeman, Richard A Hopkins, Ian

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 144 KB

english, 2001

8

Ethambutol analogues as potential antimycobacterial agents

Herwig Häusler, R.Pamela Kawakami, Eva Mlaker, Wayne B. Severn, Arnold E. Stütz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 131 KB

english, 2001

9

Anticonvulsant effects of new morphinan derivatives

Hyoung-Chun Kim, Toshitaka Nabeshima, Wang-Kee Jhoo, Kwang Ho Ko, Won-Ki Kim, Eun-Joo Shin, Minkyoung Cho, Phil Ho Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 109 KB

english, 2001

10

Biological evaluation of hepatitis c virus helicase inhibitors

Chee Wee Phoon, Poh Yong Ng, Anthony E Ting, Su Ling Yeo, Mui Mui Sim

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 157 KB

english, 2001

11

Inhibition of serine proteases: activity of 1,3-diazetidine-2,4-diones

Yasunori Aoyama, Masaaki Uenaka, Toshiro Konoike, Yoko Hayasaki-Kajiwara, Noriyuki Naya, Masatoshi Nakajima

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 133 KB

english, 2001

12

Total synthesis of human chymase inhibitor methyllinderone and structure–activity relationships of its derivatives

Yasunori Aoyama, Toshiro Konoike, Akiko Kanda, Noriyuki Naya, Masatoshi Nakajima

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 182 KB

english, 2001

13

Antimycobacterial activity of 9-sulfonylated/sulfenylated-6-mercaptopurine derivatives

Andrea Scozzafava, Antonio Mastrolorenzo, Claudiu T Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 120 KB

english, 2001

14

Biphenyls as surrogates of the steroidal backbone. Part 1: synthesis and estrogen receptor affinity of an original series of polysubstituted biphenyls

Dominique Lesuisse, Eva Albert, Françoise Bouchoux, E Cérède, Jean-Michel Lefrançois, Marc-Olivier Levif, Sophie Tessier, Bernadette Tric, Georges Teutsch

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 220 KB

english, 2001

15

Biphenyls as Surrogates of the Steroidal Backbone. Part 2: Discovery of a Novel Family of Non-steroidal 5-α-Reductase Inhibitors

Dominique Lesuisse, Jean-François Gourvest, Eva Albert, Bernard Doucet, Catherine Hartmann, Jean-Michel Lefrançois, Sophie Tessier, Bernadette Tric, Georges Teutsch

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 156 KB

english, 2001

16

Selective Inhibition of Src SH2 by a Novel Thiol-Targeting Tricarbonyl-Modified Inhibitor and Mechanistic Analysis by 1H/13C NMR Spectroscopy

Raji Sundaramoorthi, Chris Siedem, Chi B Vu, David C Dalgarno, Ellen C Laird, Martyn C Botfield, Amanda B Combs, Susan E Adams, Ruth W Yuan, Manfred Weigele, Surinder S Narula

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 685 KB

english, 2001

17

[3H]MFZ 2-12: A Novel Radioligand for the Dopamine Transporter

Amy Hauck Newman, Mu-Fa Zou, Jasmine V Ferrer, Jonathan A Javitch

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 146 KB

english, 2001

18

Piperazinyl benzamidines: Synthesis and affinity for the delta opioid receptor

Samuel O. Nortey, Ellen W. Baxter, Ellen E. Codd, Sui-Po Zhang, Allen B. Reitz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 118 KB

english, 2001

19

Isoindolines: A new series of potent and selective endothelin-A receptor antagonists

Paivi J. Kukkola, Natalie A. Bilci, Theodore Ikler, Paula Savage, Suraj S. Shetty, Dominick DelGrande, Arco Y. Jeng

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 114 KB

english, 2001

20

Substituted Indole-5-carboxamides and -acetamides as Potent Nonpeptide GnRH Receptor Antagonists

Wallace T. Ashton, Rosemary M. Sisco, Yi Tien Yang, Jane-Ling Lo, Joel B. Yudkovitz, Kang Cheng, Mark T. Goulet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 159 KB

english, 2001

21

Potent nonpeptide GnRH receptor antagonists derived from substituted indole-5-carboxamides and -acetamides bearing a pyridine side-chain terminus

Wallace T. Ashton, Rosemary M. Sisco, Yi Tien Yang, Jane-Ling Lo, Joel B. Yudkovitz, Patrice H. Gibbons, George R. Mount, Rena Ning Ren, Bridget S. Butler, Kang Cheng, Mark T. Goulet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 151 KB

english, 2001

22

A simple method to obtain a covalent immobilized phospholipase A2

R.R. Madoery, G.D. Fidelio

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 81 KB

english, 2001

23

3-Carboxamido analogues of morphine and naltrexone: synthesis and opioid receptor binding properties

Mark P. Wentland, Rongliang Lou, Christoph M. Dehnhardt, Wenhu Duan, Dana J. Cohen, Jean M. Bidlack

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 156 KB

english, 2001

24

Novel sulfonate Derivatives: potent antimitotic agents

Stephen L. Gwaltney II, Hovis M. Imade, Qun Li, Laura Gehrke, R.Bruce Credo, Robert B. Warner, Jang Yun Lee, Peter Kovar, David Frost, Shi-Chung Ng, Hing L. Sham

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 138 KB

english, 2001

25

Synthesis of a novel C-10 spiro-epoxide of paclitaxel

Michael A. Walker, Timothy D. Johnson, Stella Huang, Dolatorai M. Vyas, John F. Kadow

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 143 KB

english, 2001

26

Synthesis of substituted 5[H]phenanthridin-6-ones as potent poly(ADP-ribose)polymerase-1 (PARP1) inhibitors

Jia-He Li, Larisa Serdyuk, Dana V. Ferraris, Ge Xiao, Kevin L. Tays, Paul W. Kletzly, Weixing Li, Susan Lautar, Jie Zhang, Vincent J. Kalish

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 149 KB

english, 2001

27

Some 3-Thioxo/alkylthio-1,2,4-triazoles with a substituted thiourea moiety as possible antimycobacterials

Ilkay Küçükgüzel, S.Güniz Küçükgüzel, Sevim Rollas, Muammer Kiraz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 153 KB

english, 2001

28

Synthesis and nuclease stability of trilysyl dendrimer–oligodeoxyribonucleotide hybrids

David A Sarracino, Clemens Richert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 174 KB

english, 2001

29

Antioxidant activity of water-soluble chitosan derivatives

Wenming Xie, Peixin Xu, Qing Liu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 98 KB

english, 2001

30

Promotion of radiation-induced formation of 8-oxo-7,8-dihydro-2′-deoxyguanosine by nitro 5-Deazaflavin derivatives

Tetsuji Kawamoto, Yoshihiro Ikeuchi, Yuji Mikata, Maki Kishigami, Shigenobu Yano, Chieko Murayama, Tomoyuki Mori, Fumio Yoneda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 126 KB

english, 2001

31

Novel and potent tacrine-related hetero- and homobivalent ligands for acetylcholinesterase and butyrylcholinesterase

Luisa Savini, Giuseppe Campiani, Alessandra Gaeta, Cesare Pellerano, Caterina Fattorusso, Luisa Chiasserini, James M Fedorko, Ashima Saxena

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 156 KB

english, 2001

32

Parallel-stranded hairpins containing 8-aminopurines. novel efficient probes for triple-helix formation

Anna Aviñó, Juan Carlos Morales, Miriam Frieden, Beatriz G. de la Torre, Ramon Güimil Garcı́a, Elena Cubero, F.Javier Luque, Modesto Orozco, Ferran Azorı́n, Ramon Eritja

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 166 KB

english, 2001

33

Biotin labelling of amines by polymer-assisted solution-phase synthesis

Abolfasl Golisade, Claudia Herforth, Karen Wieking, Conrad Kunick, Andreas Link

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 109 KB

english, 2001

34

Phenylcyanoguanidines as inhibitors of glucose-induced insulin secretion from beta cells

Tina M Tagmose, John P Mogensen, Pia C Agerholm, Per O.G Arkhammar, Philip Wahl, Anne Worsaae, J.Bondo Hansen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 127 KB

english, 2001

35

Incorporation of α- and β-LNA (Locked nucleic acid) monomers in oligodeoxynucleotides with polarity reversals

Nanna K Christensen, Britta M Dahl, Poul Nielsen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 145 KB

english, 2001

36

Rational design of a new series of pronucleotide

Thierry Beltran, David Egron, Alain Pompon, Isabelle Lefebvre, Christian Périgaud, Gilles Gosselin, Anne-Marie Aubertin, Jean-Louis Imbach

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 122 KB

english, 2001

37

A mechanism-based affinity-labeling agent for possible use in isolating N-acetylglucosaminidase

Mie Ichikawa, Yoshitaka Ichikawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 454 KB

english, 2001

38

Significance of Hydrogen Bonding at the S1′ Subsite of Calpain I

Isaac O. Donkor, Xiaozhang Zheng, Jie Han, Calvin Lacy, Duane D. Miller

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 137 KB

english, 2001

39

Inactivation of monoamine oxidase B by 1-phenylcyclopropylamine: mass spectral evidence for the flavin adduct

Deanna J. Mitchell, Dejan Nikolic, Richard B. van Breemen, Richard B. Silverman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 164 KB

english, 2001

40

Carbonic anhydrase inhibitors: 4-sulfamoyl-benzenecarboxamides and 4-chloro-3-sulfamoyl-benzenecarboxamides with strong topical antiglaucoma properties

Francesco Mincione, Michele Starnotti, Luca Menabuoni, Andrea Scozzafava, Angela Casini, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 126 KB

english, 2001

41

Discovery of 2,3-diaryl-1,3-thiazolidin-4-ones as potent anti-HIV-1 agents

Maria Letizia Barreca, Alba Chimirri, Laura De Luca, Anna-Maria Monforte, Pietro Monforte, Angela Rao, Maria Zappalà, Jan Balzarini, Erik De Clercq, Christophe Pannecouque, Myriam Witvrouw

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 113 KB

english, 2001

42

Instructions to Contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 96 KB

english, 2001

43

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 42 KB

english, 2001

44

Instructions to Contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 316 KB

english, 2001

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