Volume 11; Issue 14

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Bioorganic & Medicinal Chemistry Letters
Volume 11; Issue 14

Bioorganic & Medicinal Chemistry Letters

Volume 11; Issue 14

1

Inhibition of fucosyltransferase V by a GDP–Azasugar

Matthias Schuster, Siegfried Blechert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 114 KB

english, 2001

2

Novel piperidinyloxy oxazolidinone antimicrobial agents

Michele A Weidner-Wells, Christine M Boggs, Barbara D Foleno, Ellyn Wira, Karen Bush, Raul M Goldschmidt, Dennis J Hlasta

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 156 KB

english, 2001

3

Nitrobenzene Compounds Inhibit Expression of VCAM-1

Charles Q. Meng, X.Sharon Zheng, Lisa A. Holt, Lee K. Hoong, Patricia K. Somers, Russell R. Hill, Uday Saxena

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 184 KB

english, 2001

4

Preparation of oligonucleotides without aldehyde abasic sites

Achim H. Krotz, Hans Gaus, Vasulinga T. Ravikumar, Douglas L. Cole

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 168 KB

english, 2001

5

Design, synthesis, and biological evaluation of a series of simple and novel potential antimalarial compounds

Hongyu Ren, Shannon Grady, Daniela Gamenara, Horacio Heinzen, Patrick Moyna, Simon L. Croft, Howard Kendrick, Vanessa Yardley, Guillermo Moyna

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 137 KB

english, 2001

6

Synthesis of oxorhenium(V) and oxotechnetium(V) [SN(R)S/S] mixed ligand complexes containing a phenothiazine moiety on the tridentate SN(R)S ligand

Ioannis Pirmettis, Georgios Patsis, Maria Pelecanou, Charalampos Tsoukalas, Apostolos Papadopoulos, Catherine P. Raptopoulou, Aris Terzis, Minas Papadopoulos, Efstratios Chiotellis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 149 KB

english, 2001

7

Diaminopurine-acridine heterodimers for specific recognition of abasic site containing DNA. Influence on the biological activity of the position of the linker on the purine ring

Karine Alarcon, Martine Demeunynck, Jean Lhomme, Danièle Carrez, Alain Croisy

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 203 KB

english, 2001

8

Development of potent and selective factor Xa inhibitors

Roopa Rai, Aleksandr Kolesnikov, Yong Li, Wendy B Young, Ellen Leahy, Paul A Sprengeler, Erik Verner, William D Shrader, Jana Burgess-Henry, Joan C Sangalang, Darin Allen, Xi Chen, Bradley A Katz, Chr

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 562 KB

english, 2001

9

Neutral inhibitors of the serine protease factor Xa

William D. Shrader, Wendy B. Young, Paul A. Sprengeler, Joan C. Sangalang, Kyle Elrod, Grant Carr

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 369 KB

english, 2001

10

Novel Tricyclic Benzothiazolo[2,3-c]thiadiazine Antagonists of the Platelet ADP Receptor (P2Y12)

Robert M. Scarborough, Alan M. Laibelman, Lane A. Clizbe, Larry J. Fretto, Pamela B. Conley, Elwood E. Reynolds, David M. Sedlock, Hans-Michael Jantzen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 136 KB

english, 2001

11

Macrocyclization in the design of a conformationally constrained Grb2 SH2 domain inhibitor

Yang Gao, Johannes Voigt, Jane X Wu, Dajun Yang, Terrence R Burke, Jr

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 659 KB

english, 2001

12

Synthesis and biological activity of novel macrocyclic antifungals: modification of the tyrosine moiety of the lipopeptidolactone FR901469

David Barrett, Akira Tanaka, Keiko Harada, Etsuko Watabe, Katsuyuki Maki, Fumiaki Ikeda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 291 KB

english, 2001

13

Phytoestrogens from the roots of Polygonum cuspidatum (polygonaceae): structure-Requirement of hydroxyanthraquinones for estrogenic activity

Hisashi Matsuda, Hiroshi Shimoda, Toshio Morikawa, Masayuki Yoshikawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 177 KB

english, 2001

14

Design and synthesis of novel benzofurans as a new class of antifungal agents targeting fungal N-myristoyltransferase. Part 1

Miyako Masubuchi, Ken-ichi Kawasaki, Hirosato Ebiike, Yoshihiko Ikeda, Shinji Tsujii, Satoshi Sogabe, Toshihiko Fujii, Kiyoaki Sakata, Yasuhiko Shiratori, Yuko Aoki, Tatsuo Ohtsuka, Nobuo Shimma

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 439 KB

english, 2001

15

Cyclic imides as potent and selective α-1A adrenergic receptor antagonists

Robert M DiPardo, Michael A Patane, Randall C Newton, RoseAnn Price, Theodore P Broten, Raymond S.L Chang, Richard W Ransom, Jerry Di Salvo, Roger M Freidinger, Mark G Bock

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 156 KB

english, 2001

16

2-Amino-4,6-diarylpyridines as novel ligands for the estrogen receptor

Brad R Henke, David H Drewry, Stacey A Jones, Eugene L Stewart, Susan L Weaver, Robert W Wiethe

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 199 KB

english, 2001

17

Carbohydrate recognition of gramicidin S analogues in aqueous medium

Takuro Niidome, Hiroto Murakami, Masahito Kawazoe, Tomomitsu Hatakeyama, Yoshihiro Kobashigawa, Minako Matsushita, Yasuhiro Kumaki, Makoto Demura, Katsutoshi Nitta, Haruhiko Aoyagi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 198 KB

english, 2001

18

Development of specific CXCR4 inhibitors possessing high selectivity indexes as well as complete stability in serum based on an anti-HIV peptide T140

Hirokazu Tamamura, Akane Omagari, Kenichi Hiramatsu, Kazuyo Gotoh, Taisei Kanamoto, Younong Xu, Eiichi Kodama, Masao Matsuoka, Toshio Hattori, Naoki Yamamoto, Hideki Nakashima, Akira Otaka, Nobutaka F

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 218 KB

english, 2001

19

Spiro(indoline-3,4′-piperidine) growth hormone secretagogues as ghrelin mimetics

Brenda L. Palucki, Scott D. Feighner, Sheng-Shung Pong, Karen Kulju McKee, Donna L. Hreniuk, Carina Tan, Andrew D. Howard, Lex H.Y. Van der Ploeg, Arthur A. Patchett, Ravi P. Nargund

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 121 KB

english, 2001

20

α-Ketocarboxylic acid-based inhibitors of protein tyrosine phosphatases

Yen Ting Chen, M.Burak Onaran, Christopher J. Doss, Christopher T. Seto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 152 KB

english, 2001

21

Nicotinamide N-Oxides as CXCR2 antagonists

Neil S Cutshall, Rocky Ursino, Kristin A Kucera, John Latham, Nathan C Ihle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 141 KB

english, 2001

22

Selectivity enhancement induced by substitution of non-natural analogues of arginine and lysine in arginine-based thrombin inhibitors

Kyle P Kokko, Christine E Arrigoni, Thomas A Dix

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 144 KB

english, 2001

23

Synthesis of N1-substituted analogues of (2R,4R)-4-amino-pyrrolidine-2,4-dicarboxylic acid as agonists, partial agonists, and antagonists of group II metabotropic glutamate receptors

Jayanta Kumar Mukhopadhyaya, Alan P. Kozikowski, Ewa Grajkowska, Sergey Pshenichkin, Jarda T. Wroblewski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 257 KB

english, 2001

24

3-Arylpiperidines as potentiators of existing antibacterial agents

Atli Thorarensen, Alice L Presley-Bodnar, Keith R Marotti, Timothy P Boyle, Charlotte L Heckaman, Michael J Bohanon, Paul K Tomich, Gary E Zurenko, Michael T Sweeney, Betty H Yagi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 283 KB

english, 2001

25

Synthesis and evaluation of novel quinolinones as HIV-1 reverse transcriptase inhibitors

Mona Patel, Robert J McHugh Jr., Beverly C Cordova, Ronald M Klabe, Lee T Bacheler, Susan Erickson-Viitanen, James D Rodgers

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 121 KB

english, 2001

26

In vitro and In vivo inhibition of LPS-stimulated tumor necrosis factor-α secretion by the gallotannin β-d-pentagalloylglucose

Ken S. Feldman, Kiran Sahasrabudhe, Michael D. Lawlor, Sarah L. Wilson, Charles H. Lang, William J. Scheuchenzuber

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 162 KB

english, 2001

27

N-Acyloxymethyl carbamate linked prodrugs of pseudomycins are novel antifungal agents

Xicheng Sun, Douglas J Zeckner, William L Current, Robert Boyer, Carl McMillian, Nathan Yumibe, Shu-Hui Chen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 146 KB

english, 2001

28

Studies towards the next generation of antidepressants. Part 1: indolylcyclohexylamines as potent serotonin reuptake inhibitors

Kristin L Meagher, Richard E Mewshaw, Deborah A Evrard, Ping Zhou, Deborah L Smith, Rosemary Scerni, Taylor Spangler, Susan Abulhawa, Xiaojie Shi, Lee E Schechter, Terrance H Andree

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 191 KB

english, 2001

29

Prodrugs of 3-amido bearing pseudomycin analogues: novel antifungal agents

Xicheng Sun, Douglas J Zeckner, Yan-zhi Zhang, Roberta K Sachs, William L Current, Michael Rodriguez, Shu-Hui Chen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 131 KB

english, 2001

30

Synthesis and biological evaluation of didemnin photoaffinity analogues

Matthew D. Vera, Amy J. Pfizenmayer, Xiaobin Ding, Deepika Ahuja, Peter L. Toogood, Madeleine M. Joullié

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 143 KB

english, 2001

31

Evaluation of amino acid-based linkers in potent macrocyclic inhibitors of farnesyl-protein transferase

Douglas C Beshore, Ian M Bell, Christopher J Dinsmore, Carl F Homnick, J.Christopher Culberson, Ronald G Robinson, Christine Fernandes, Eileen S Walsh, Marc T Abrams, Hema G Bhimnathwala, Joseph P Dav

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 293 KB

english, 2001

32

Corrigendum to “allyl and Propargyl substituted penam sulfones as versatile intermediates toward the syntheses of new β-lactamase inhibitors”: [Bioorg. Med. Chem. Lett. 11 (2001) 997]†

Vincent P. Sandanayaka, Gregg B. Feigelson, Amar S. Prashad, Youjun Yang, Peter J. Petersen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 60 KB

english, 2001

33

1,3-Biarylureas as selective non-peptide antagonists of the orexin-1 receptor

Roderick A Porter, Wai N Chan, Steven Coulton, Amanda Johns, Michael S Hadley, Katherine Widdowson, Jeffrey C Jerman, Stephen J Brough, Martyn Coldwell, Darren Smart, Frances Jewitt, Phillip Jeffrey,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 131 KB

english, 2001

34

Studies leading to the identification of ZD1839 (iressa™): an orally active, selective epidermal growth factor receptor tyrosine kinase inhibitor targeted to the treatment of cancer

Andrew J Barker, Keith H Gibson, Walter Grundy, Andrew A Godfrey, Jeffrey J Barlow, Mark P Healy, James R Woodburn, Susan E Ashton, Brenda J Curry, Lynn Scarlett, Lianne Henthorn, Laura Richards

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 156 KB

english, 2001

35

Highly potent growth hormone secretagogues: Hybrids of NN703 and ipamorelin

Thomas K. Hansen, Michael Ankersen, Kirsten Raun, Birgit S. Hansen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 128 KB

english, 2001

36

1-(Arylpiperazinylamidoalkyl)-pyrimidones: orally active inhibitors of lipoprotein-associated phospholipase A2

Jackie C. Bloomer, Helen F. Boyd, Deirdre M.B. Hickey, Robert J. Ife, Colin A. Leach, Colin H. Macphee, Kevin J. Milliner, Ivan L. Pinto, D.Anthony Rawlings, Stephen A. Smith, Ian G. Stansfield, Steve

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 148 KB

english, 2001

37

Introduction of alkynyl chains on C-8 of adenosine led to very selective antagonists of the A3 adenosine receptor

Rosaria Volpini, Stefano Costanzi, Catia Lambertucci, Sauro Vittori, K.-N Klotz, Anna Lorenzen, Gloria Cristalli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 117 KB

english, 2001

38

Pyrazinone conjugates as potential cephalosporin allergens

Lennart Venemalm

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 97 KB

english, 2001

39

Contributors to this Issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 42 KB

english, 2001

40

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 298 KB

english, 2001

41

Instructions to Contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 96 KB

english, 2001

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