Volume 11; Issue 19

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Bioorganic & Medicinal Chemistry Letters
Volume 11; Issue 19

Bioorganic & Medicinal Chemistry Letters

Volume 11; Issue 19

1

Novel 3-dodecanoylindole-2-carboxylic acid inhibitors of cytosolic phospholipase A2

Matthias Lehr, Monika Klimt, Alwine Schulze Elfringhoff

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 143 KB

english, 2001

2

EDTA bis-(ethyl phenylalaninate): A novel transition metal-Ion chelating hydroxyl radical scavenger with a potential anti-inflammatory role

Declan P. Naughton, Martin Grootveld

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 114 KB

english, 2001

3

Inhibition of hiv-1 infection by synthetic peptide analogues derived from the nh2-Terminal extracellular region of gpr1

Kiyoshi Ikeda, Koji Konishi, Masayuki Sato, Hiroo Hoshino, Kiyoshi Tanaka

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 107 KB

english, 2001

4

A new reactive nucleoside analogue for highly reactive and selective cross-linking reaction to cytidine under neutral conditions

Fumi Nagatsugi, Natsuko Tokuda, Minoru Maeda, Shigeki Sasaki

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 131 KB

english, 2001

5

Combinatorial synthesis of SSAO inhibitors using sonogashira coupling: SAR of aryl propargylic amines

Costa Conn, Ronald Shimmon, Frank Cordaro, Tracey-Lea Hargraves, Peter Ibrahim

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 133 KB

english, 2001

6

Solid-Phase synthesis of a library constructed of aromatic phosphate, long alkyl chains and tryptophane components, and identification of potent dipeptide telomerase inhibitors

Shigeki Sasaki, Takeru Ehara, Md Rowshon Alam, Yasuhiro Fujino, Naozumi Harada, Junko Kimura, Hideo Nakamura, Minoru Maeda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 188 KB

english, 2001

7

Synthesis and in vitro evaluation of a series of diketopiperazine inhibitors of plasminogen activator inhibitor-1

Adrian Folkes, Michael B Roe, Sukhjit Sohal, Julian Golec, Richard Faint, Teresa Brooks, Peter Charlton

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 120 KB

english, 2001

8

Asymmetric synthesis of bb-3497—A potent peptide deformylase inhibitor

Lisa M Pratt, R.Paul Beckett, Stephen J Davies, Steven B Launchbury, Andrew Miller, Zoe M Spavold, Richard S Todd, Mark Whittaker

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 115 KB

english, 2001

9

Isoxazolyl, oxazolyl, and thiazolylpropionic acid derivatives as potent α4β1 integrin antagonists

Allen J Duplantier, Gretchen E Beckius, Robert J Chambers, Louis S Chupak, Teresa H Jenkinson, Anne S Klein, Kenneth G Kraus, Elizabeth M Kudlacz, Michael W McKechney, Martin Pettersson, Carrie A Whit

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 132 KB

english, 2001

10

Orally bioavailable, indole-based nonpeptide GnRH receptor antagonists with high potency and functional activity

Wallace T. Ashton, Rosemary M. Sisco, Gerard R. Kieczykowski, Yi Tien Yang, Joel B. Yudkovitz, Jisong Cui, George R. Mount, Rena Ning Ren, Tsuei-Ju Wu, Xiaolan Shen, Kathryn A. Lyons, An-Hua Mao, Jose

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 168 KB

english, 2001

11

Robinlin: A novel bioactive homo-monoterpene from Robinia pseudoacacia L. (Fabaceae)

Feifei Tian, Ching-Jer Chang, John B Grutzner, David E Nichols, Jerry L McLaughlin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 111 KB

english, 2001

12

Novel lipophilic chloroquine analogues for a highly efficient gene transfer into gynecological tumors

Oliver Keil, Hans Bojar, Hans-Bernd Prisack, Peter Dall

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 163 KB

english, 2001

13

Synthesis and acetylcholinesterase inhibition of 5-desamino huperzine A derivatives

Klemens Högenauer, Karl Baumann, Albert Enz, Johann Mulzer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 130 KB

english, 2001

14

Design, synthesis and characterisation of a peptide with oxaloacetate decarboxylase activity

Susan E Taylor, Trevor J Rutherford, Rudolf K Allemann

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 254 KB

english, 2001

15

Synthesis, biological activity and comparative analysis of DNA binding affinities and human DNA topoisomerase I inhibitory activities of novel 12-alkoxy-benzo[c]phenanthridinium salts

Michael A Lynch, Olivier Duval, Alyona Sukhanova, Jerome Devy, Simon P MacKay, Roger D Waigh, Igor Nabiev

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 175 KB

english, 2001

16

Selective heterocyclic amidine inhibitors of human inducible nitric oxide synthase

Alan E Moormann, Sue Metz, Mihaly V Toth, William M Moore, Gina Jerome, Christine Kornmeier, Pamela Manning, Donald W Hansen Jr., Barnett S Pitzele, R.K Webber

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 89 KB

english, 2001

17

Synthesis of a reported calpain inhibitor isolated from Streptomyces griseus

I.O Donkor, M.Lee Sanders

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 118 KB

english, 2001

18

New inhibitors of the thioredoxin–thioredoxin reductase system based on a naphthoquinone spiroketal natural product lead

Peter Wipf, Tamara D. Hopkins, Jae-Kyu Jung, Sonia Rodriguez, Anne Birmingham, Eileen C. Southwick, John S. Lazo, Garth Powis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 173 KB

english, 2001

19

Potent peptide α-Ketohydroxamate inhibitors of recombinant human calpain I

Kurt A Josef, Frederick W Kauer, Ron Bihovsky

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 102 KB

english, 2001

20

RNA–DNA Hybrids Containing Damaged DNA are Substrates for RNase H

Jerome C Shiels, Bozidar Jerkovic, Anne M Baranger, Philip H Bolton

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 124 KB

english, 2001

21

Antiprotozoal and cytotoxicity evaluation of sulfonamide and urea analogues of quinacrine

Kelly Chibale, Hayley Haupt, Howard Kendrick, Vanessa Yardley, Ahilan Saravanamuthu, Alan H Fairlamb, Simon L Croft

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 91 KB

english, 2001

22

1,2,4-Triazolo[3,4-a]pyridine as a novel, constrained template for fibrinogen receptor (GPIIb/IIIa) antagonists

Edward C Lawson, William J Hoekstra, Michael F Addo, Patricia Andrade-Gordon, Bruce P Damiano, Jack A Kauffman, John A Mitchell, Bruce E Maryanoff

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 125 KB

english, 2001

23

Synthesis of diaminobutane derivatives as potent Ca2+-Permeable AMPA receptor antagonists

Yoshiyuki Yoneda, Shinichi Kawajiri, Masunobu Sugimura, Ken Osanai, Fusako Kito, Emi Ota, Tetuya Mimura

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 140 KB

english, 2001

24

Synthesis, topoisomerase I inhibition and antitumor cytotoxicity of 2,2′:6′,2″-, 2,2′:6′,3″- and 2,2′:6′,4″-Terpyridine derivatives

Long-Xuan Zhao, Tae Sung Kim, Soo-Hyun Ahn, Tae-Hyung Kim, Eun-kyung Kim, Won-Jea Cho, Heesung Choi, Chong-Soon Lee, Jung-Ae Kim, Tae Cheon Jeong, Ching-jer Chang, Eung-Seok Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 134 KB

english, 2001

25

Contributors to this Issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 37 KB

english, 2001

26

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 183 KB

english, 2001

27

Instructions to Contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 96 KB

english, 2001

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