Volume 11; Issue 20

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Bioorganic & Medicinal Chemistry Letters
Volume 11; Issue 20

Bioorganic & Medicinal Chemistry Letters

Volume 11; Issue 20

1

Synthesis, characterisation and antiamoebic activity of new thiophene-2-carboxaldehyde thiosemicarbazone derivatives and Their cyclooctadiene Ru(II) complexes

N.S. Shailendra, Neelam Bharti, M.T Gonzalez Garza, Delia E Cruz-Vega, J Castro Garza, Kishwar Saleem, Fehmida Naqvi, Amir Azam

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 106 KB

english, 2001

2

Naphthalene derivatives: A new series of selective cyclooxygenase-2 inhibitors

Joan Feixas, Juan-Miguel Jiménez, Núria Godessart, Carles Puig, Lı́dia Soca, Marı́a I Crespo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 121 KB

english, 2001

3

Synthesis and biological evaluation of novel bisindolylmaleimides that inhibit vascular endothelial cell proliferation

Miguel F Braña, Loreto Añorbe, Gema Tarrasón, Francesc Mitjans, Jaume Piulats

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 118 KB

english, 2001

4

Regiospecific phosphohydrolases from Dictyostelium as tools for the chemoenzymatic synthesis of the enantiomers d-myo-inositol 1,2,4-trisphosphate and d-myo-inositol 2,3,6-trisphosphate: non-physiological, potential analogues of biologically active d-myo-inositol 1,3,4-trisphosphate

Stephan Adelt, Oliver Plettenburg, Guido Dallmann, Frank P Ritter, Stephen B Shears, Hans-Josef Altenbach, Günter Vogel

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 176 KB

english, 2001

5

Discovery and initial structure–Activity relationships of trisubstituted ureas as thrombin receptor (PAR-1) antagonists

James C Barrow, Philippe G Nantermet, Harold G Selnick, Kristen L Glass, Phung L Ngo, Mary Beth Young, Janetta M Pellicore, Michael J Breslin, John H Hutchinson, Roger M Freidinger, Cindra Condra, Jer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 180 KB

english, 2001

6

The synthesis and properties of new 2-pyrrolylthiones as chelating agents for transition metals and technetium

Svetlana V Selivanova, David Dolphin, Christian Brückner, Johan E. van Lier, Svetlana Kudrevich

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 96 KB

english, 2001

7

Microwave assisted synthesis of N-Arylphthalamic acids with hyperlipidemic activity

Vera L.M Sena, Rajendra M Srivastava, Shalom P Oliveira, Vera L.M Lima

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 103 KB

english, 2001

8

N,N′-Bis[4-(N-alkylamidino)phenyl]homopiperazines as anti-Pneumocystis carinii agents

Tien L Huang, Bin Tao, Yvonne Quarshie, Sherry F Queener, Isaac O Donkor

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 95 KB

english, 2001

9

Design and synthesis of irreversible depsipeptidyl human rhinovirus 3C protease inhibitors

Stephen E. Webber, Joseph T. Marakovits, Peter S. Dragovich, Thomas J. Prins, Ru Zhou, Shella A. Fuhrman, Amy K. Patick, David A. Matthews, Caroline A. Lee, Babu Srinivasan, Terry Moran, Clifford E. F

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 132 KB

english, 2001

10

Mixed κ agonists and μ agonists/Antagonists as potential pharmacotherapeutics for cocaine abuse: synthesis and opioid receptor binding affinity of N-substituted derivatives of morphinan

John L Neumeyer, Xiao-Hui Gu, L.Alexander van Vliet, Nicholas J DeNunzio, Daniela E Rusovici, Dana J Cohen, S.Stevens Negus, Nancy K Mello, Jean M Bidlack

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 136 KB

english, 2001

11

The discovery of sulfonylated dipeptides as Potent VLA-4 antagonists

William K Hagmann, Philippe L Durette, Thomas Lanza, Nancy Jo Kevin, Stephen E de Laszlo, Ihor E Kopka, David Young, Plato A Magriotis, Bing Li, Linus S Lin, Ginger Yang, Theodore Kamenecka, Linda L C

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 142 KB

english, 2001

12

1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 2: lead optimization affording selective, orally bioavailable compounds with potent Anti-HIV activity

Jeffrey J. Hale, Richard J. Budhu, Edward B. Holson, Paul E. Finke, Bryan Oates, Sander G. Mills, Malcolm MacCoss, Sandra L. Gould, Julie A. DeMartino, Martin S. Springer, Salvatore Siciliano, Lorrain

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 123 KB

english, 2001

13

Synthesis of N-propargylphenelzine and analogues as neuroprotective agents

Lei Ling, Liana J. Urichuk, B.Duff Sloley, Ronald T. Coutts, Glen B. Baker, Jacqueline J. Shan, Peter K.T. Pang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 106 KB

english, 2001

14

Efficient synthesis of lactosaminylated core-2 O-glycans

Anup Kumar Misra, Minoru Fukuda, Ole Hindsgaul

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 116 KB

english, 2001

15

Small molecule/Nucleic acid affinity chromatography: application for the identification of telomerase inhibitors which target its key RNA/DNA heteroduplex

Corinna West, Rawle Francis, Simon H Friedman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 206 KB

english, 2001

16

Synthesis and progesterone receptor antagonist activities of 6-aryl benzimidazolones and benzothiazolones

Puwen Zhang, Eugene A. Terefenko, Jay Wrobel, Zhiming Zhang, Yuan Zhu, Jeffrey Cohen, Keith B. Marschke, Dale Mais

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 132 KB

english, 2001

17

α-Amino-β-sulphone hydroxamates as potent MMP-13 inhibitors that spare MMP-1

Daniel P Becker, Thomas E Barta, Louis Bedell, Gary DeCrescenzo, John Freskos, Daniel P Getman, Susan L Hockerman, Madeleine Li, Pramod Mehta, Brent Mischke, Grace E Munie, Craig Swearingen, Clara I V

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 128 KB

english, 2001

18

α-Alkyl-α-amino-β-sulphone hydroxamates as potent MMP inhibitors that spare MMP-1

Daniel P Becker, Gary DeCrescenzo, John Freskos, Daniel P Getman, Susan L Hockerman, Madeleine Li, Pramod Mehta, Grace E Munie, Craig Swearingen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 119 KB

english, 2001

19

Total synthesis and antifungal activity of 9-methoxystrobilurin L as the originally proposed 1,4-Benzodioxan structure

Yasuyuki Aiba, Daiju Hasegawa, Takahiro Marunouchi, Koh Nagasawa, Hiromi Uchiro, Susumu Kobayashi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 145 KB

english, 2001

20

Anti-Trypanosoma activity of some natural stilbenoids and synthetic related heterocyclic compounds

Esther del Olmo, Marlon Garcı́a Armas, Jose Luis López-Pérez, Grace Ruiz, Fernando Vargas, Alberto Giménez, Eric Deharo, Arturo San Feliciano

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 97 KB

english, 2001

21

NaBH4 in N-methylpyrrolidone: a safe alternative for hydride displacement reaction

Yasuhiro Torisawa, Takao Nishi, Jun-ichi Minamikawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 101 KB

english, 2001

22

Potent second generation vinyl sulfonamide inhibitors of the trypanosomal cysteine protease cruzain

William R. Roush, Jianming Cheng, Beth Knapp-Reed, Alejandro Alvarez-Hernandez, James H. McKerrow, Elizabeth Hansell, Juan C. Engel

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 121 KB

english, 2001

23

Synthesis and structure–activity relationships of thiotetronic acid analogues of thiolactomycin

Subas M Sakya, Melani Suarez-Contreras, John P Dirlam, Thomas N O'Connell, Shigeru F Hayashi, Sheryl L Santoro, Barbara J Kamicker, David M George, Carl B Ziegler

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 119 KB

english, 2001

24

Small molecule somatostatin receptor subtype-2 antagonists

Bruce A. Hay, Bridget M. Cole, Frank DiCapua, Glen W. Kirk, Marianne C. Murray, Rona A. Nardone, Dennis J. Pelletier, Anthony P. Ricketts, Alan S. Robertson, Todd W. Siegel

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 141 KB

english, 2001

25

Discovery of heterocyclic ureas as a new class of raf kinase inhibitors: identification of a second generation lead by a combinatorial chemistry approach

Roger A Smith, James Barbosa, Cheri L Blum, Mark A Bobko, Yolanda V Caringal, Robert Dally, Jeffrey S Johnson, Michael E Katz, Nancy Kennure, Jill Kingery-Wood, Wendy Lee, Timothy B Lowinger, John Lyo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 112 KB

english, 2001

26

Discovery of novel, orally active dual NK1/NK2 antagonists

Peter R. Bernstein, David Aharony, Jeffrey S. Albert, Donald Andisik, Herbert G. Barthlow, Russell Bialecki, Timothy Davenport, Robert F. Dedinas, Bruce T. Dembofsky, Gerard Koether, Benedict J. Kosmi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 150 KB

english, 2001

27

Structure-based design of caspase-1 inhibitor containing a diphenyl ether sulfonamide

Aurash B Shahripour, Mark S Plummer, Elizabeth A Lunney, Tomi K Sawyer, Charles J Stankovic, Michael K Connolly, John R Rubin, Nigel P.C Walker, Kenneth D Brady, Hamish J Allen, Robert V Talanian, Win

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 150 KB

english, 2001

28

Simplified catechin-gallate inhibitors of HIV-1 reverse transcriptase

L.M.V Tillekeratne, A Sherette, P Grossman, L Hupe, D Hupe, R.A Hudson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 143 KB

english, 2001

29

Graphical Abbstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 201 KB

english, 2001

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