Volume 11; Issue 3

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Bioorganic & Medicinal Chemistry Letters
Volume 11; Issue 3

Bioorganic & Medicinal Chemistry Letters

Volume 11; Issue 3

1

Synthesis and preliminary pharmacological evaluation of coumestans with different patterns of oxygenation

Alcides J.M da Silva, Paulo A Melo, Noelson M.V Silva, Flávia V Brito, Camilla D Buarque, Daniele V de Souza, Verônica P Rodrigues, Elisa S.C Poças, François Noël, Edson X Albuquerque, Paulo R.R Costa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 253 KB

english, 2001

2

Potent and selective bicyclic lactam inhibitors of thrombin. Part 4: transition state inhibitors

Benoit Bachand, Micheline Tarazi, Yves St-Denis, Jeremy J Edmunds, Peter D Winocour, Lorraine Leblond, M.Arshad Siddiqui

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 212 KB

english, 2001

3

General synthesis of α-substituted 3-bisaryloxy propionic acid derivatives as specific mmp inhibitors

Anne-Marie Chollet, Thierry Le Diguarher, Lynne Murray, Marc Bertrand, Gordon C Tucker, Massimo Sabatini, Alain Pierré, Ghanem Atassi, Jacqueline Bonnet, Patrick Casara

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 194 KB

english, 2001

4

Antimycobacterial in vitro activity of cobalt(ii) isonicotinoylhydrazone complexes. Part 10

B. Bottari, R. Maccari, F. Monforte, R. Ottanà, E. Rotondo, M.G. Vigorita

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 109 KB

english, 2001

5

Novel cytotoxic 7-iminomethyl and 7-aminomethyl derivatives of camptothecin

Sabrina Dallavalle, Anna Ferrari, Lucio Merlini, Sergio Penco, Nives Carenini, Michelandrea De Cesare, Paola Perego, Graziella Pratesi, Franco Zunino

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 138 KB

english, 2001

6

Synthesis of 4-alkoxy-2-phenylquinoline derivatives as potent antiplatelet agents

Ting-Chia Ko, Mann-Jen Hour, Jin-Cherng Lien, Che-Ming Teng, Kuo-Hsiung Lee, Sheng-Chu Kuo, Li-Jiau Huang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 146 KB

english, 2001

7

Anthraquinone-peptides as inhibitors of AP-1 transcription factor

Taeeba Ijaz, Phoung Tran, Ketan C. Ruparelia, Paul H. Teesdale-Spittle, Samantha Orr, Laurence H. Patterson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 128 KB

english, 2001

8

The identification of α-ketoamides as potent inhibitors of hepatitis c virus nS3-4a proteinase

J.M. Bennett, A.D. Campbell, A.J. Campbell, M.G. Carr, R.M. Dunsdon, J.R. Greening, D.N. Hurst, N.S. Jennings, P.S. Jones, S. Jordan, P.B. Kay, M.A. O'Brien, J. King-Underwood, T.M. Raynham, C.S. Wilk

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 127 KB

english, 2001

9

Serotonergic and dopaminergic activities of rigidified (R)-aporphine derivatives

Tero Linnanen, Magnus Brisander, Nina Mohell, Anette M Johansson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 193 KB

english, 2001

10

Antifungal activity of octyl gallate: structural criteria and mode of action

Isao Kubo, Ping Xiao, Ken'ichi Fujita

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 149 KB

english, 2001

11

Synthesis and biological activity of novel potent endothelin-converting enzyme-1 inhibitors

Fariborz Firooznia, Candido Gude, Kenneth Chan, Cynthia A. Fink, Ying Qiao, Yoshitaka Satoh, Nicholas Marcopoulos, Paula Savage, Michael E. Beil, Charles W. Bruseo, Angelo J. Trapani, Arco Y. Jeng

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 178 KB

english, 2001

12

Sulfonylated aminothiazoles as new small molecule inhibitors of protein phosphatases

Peter Wipf, Diana C. Aslan, Eileen C. Southwick, John S. Lazo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 143 KB

english, 2001

13

Stereospecific synthesis of (2S)-2-methyl-3-(2′,6′-dimethyl-4′-hydroxyphenyl)-propionic acid (Mdp) and its incorporation into an opioid peptide

Yixin Lu, Grazyna Weltrowska, Carole Lemieux, Nga N Chung, Peter W Schiller

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 112 KB

english, 2001

14

The development of a potential single photon emission computed tomography (SPECT) imaging agent for the corticotropin-releasing hormone receptor type 1

Xinrong Tian, Ling-Wei Hsin, Elizabeth L Webster, Carlo Contoreggi, George P Chrousos, Philip W Gold, Kamal Habib, Alejandro Ayala, William C Eckelman, Arthur E Jacobson, Kenner C Rice

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 127 KB

english, 2001

15

Trifluoromethyl-containing 3-alkoxymethyl- and 3-aryloxymethyl-2-pyridinones are potent inhibitors of hIV-1 non-nucleoside reverse transcriptase

Jeffrey W. Corbett, Kristen J. Kresge, Senliang Pan, Beverly C. Cordova, Ronald M. Klabe, James D. Rodgers, Susan K. Erickson-Viitanen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 178 KB

english, 2001

16

Synthesis and photodynamic activity of a cationic zinc monoazaporphyrin bearing a nitrogen atom at the peripheral position

Shigeo Kai, Seiji Hiramitsu, Mikio Suzuki, Yukio Masaki

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 114 KB

english, 2001

17

Conformational study of a highly specific CXCR4 inhibitor, T140, disclosing the close proximity of its intrinsic pharmacophores associated with strong anti-HIV activity

Hirokazu Tamamura, Makiko Sugioka, Yoshihiko Odagaki, Akane Omagari, Yukiko Kan, Shinya Oishi, Hideki Nakashima, Naoki Yamamoto, Stephen C Peiper, Nobuyuki Hamanaka, Akira Otaka, Nobutaka Fujii

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 231 KB

english, 2001

18

Enkephalin analogues with 2′,6′-dimethylphenylalanine replacing phenylalanine in position 4

Yusuke Sasaki, Mariko Hirabuki, Akihiro Ambo, Hidekazu Ouchi, Yutaka Yamamoto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 116 KB

english, 2001

19

Selective reaction to a flipping cytidine of the duplex DNA mediated by triple helix formation

Fumi Nagatsugi, Daisaku Usui, Takeshi Kawasaki, Minoru Maeda, Shigeki Sasaki

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 166 KB

english, 2001

20

Specific binding of 2-amino-1,8-naphthyridine into a single guanine bulge as evidenced by photooxidation of GG doublet

Kazuhiko Nakatani, Shinsuke Sando, Kohzo Yoshida, Isao Saito

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 217 KB

english, 2001

21

Design and synthesis of tricyclic derivatives as high density lipoprotein cholesterol enhancers

Hassan Elokdah, Sie-Yearl Chai, Douglas Ho, Theodore Sulkowski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 230 KB

english, 2001

22

Human β3 adrenergic receptor agonists containing cyanoguanidine and nitroethylenediamine moieties

Linda L Brockunier, Mari R Candelore, Margaret A Cascieri, Yong Liu, Laurie Tota, Matthew J Wyvratt, Michael H Fisher, Ann E Weber, Emma R Parmee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 142 KB

english, 2001

23

The 5-HT3 antagonist tropisetron (ICS 205-930) is a potent and selective α7 nicotinic receptor partial agonist

John E Macor, David Gurley, Thomas Lanthorn, James Loch, Robert A Mack, George Mullen, Oahn Tran, Nicole Wright, John C Gordon

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 123 KB

english, 2001

24

Anti-Helicobacter pylori agents endowed with H2-antagonist properties

Giovanni Sorba, Massimo Bertinaria, Antonella Di Stilo, Alberto Gasco, Maria M Scaltrito, Maria I Brenciaglia, Francesco Dubini

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 146 KB

english, 2001

25

Bicyclic nucleoside inhibitors of Varicella-Zoster virus (VZV): the effect of terminal unsaturation in the side chain

Sheila Srinivasan, Christopher McGuigan, Graciela Andrei, Robert Snoeck, Erik De Clercq, Jan Balzarini

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 114 KB

english, 2001

26

Solid-phase synthesis of oligonucleotides containing a Bipyridine ligand at the 3′-3′ inversion of polarity site

Aldo Galeone, Luciano Mayol, Giorgia Oliviero, Daniela Rigano, Michela Varra

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 150 KB

english, 2001

27

Securiosides A and B, novel acylated triterpene bisdesmosides with selective cytotoxic activity against M-CSF-stimulated macrophages

Minpei Kuroda, Yoshihiro Mimaki, Yutaka Sashida, Mikio Kitahara, Masatoshi Yamazaki, Satoru Yui

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 163 KB

english, 2001

28

Active site geometry of porcine pancreatic lipase: an interesting switchover from Jones' to Seebach's model

Amit Basak, Kakali Rani Rudra, Hussam Moh'd Bdour, Jyotishman Dasgupta

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 143 KB

english, 2001

29

A model of photoprobe docking with β1,4-galactosyltransferase identifies a possible carboxylate involved in glycosylation steps

Yasumaru Hatanaka, Masaji Ishiguro, Makoto Hashimoto, Louis Noël Gastinel, Kazuya Nakagomi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 297 KB

english, 2001

30

FR131535, a novel water-soluble echinocandin-like lipopeptide: synthesis and biological properties

Akihiko Fujie, Toshiro Iwamoto, Bunji Sato, Hideyuki Muramatsu, Chiyoshi Kasahara, Takahisa Furuta, Yasuhiro Hori, Motohiro Hino, Seiji Hashimoto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 126 KB

english, 2001

31

Synthesis and antifungal activities of novel 1,3-β-d-glucan synthase inhibitors. Part 1

Kazunao Masubuchi, Takehiro Okada, Masami Kohchi, Masahiro Sakaitani, Eisaku Mizuguchi, Haruyoshi Shirai, Masahiro Aoki, Takahide Watanabe, Osamu Kondoh, Toshikazu Yamazaki, Yasuko Satoh, Kazuko Kobay

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 167 KB

english, 2001

32

Solid-phase synthesis of pyrrolo[2,1-c]benzodiazepine-5,11-diones

Ahmed Kamal, G.Suresh Kumar Reddy, Sadagopan Raghavan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 113 KB

english, 2001

33

Orally active docetaxel analogue: synthesis of 10-deoxy-10-C-morpholinoethyl docetaxel analogues

Shin Iimura, Kouichi Uoto, Satoru Ohsuki, Jun Chiba, Toshiharu Yoshino, Michio Iwahana, Takeshi Jimbo, Hirofumi Terasawa, Tsunehiko Soga

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 209 KB

english, 2001

34

Synthesis and transfecting properties of a glycosylated polycationic DNA vector

Christophe Jacopin, Hans Hofland, Daniel Scherman, Jean Herscovici

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 213 KB

english, 2001

35

Structure–activity relationships of novel anti-malarial agents. Part 2: cinnamic acid derivatives

Jochen Wiesner, Andreas Mitsch, Pia Wißner, Hassan Jomaa, Martin Schlitzer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 107 KB

english, 2001

36

Non-peptidic, non-prenylic inhibitors of the prenyl protein-specific protease Rce1

Martin Schlitzer, Ann Winter-Vann, Patrick J Casey

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 171 KB

english, 2001

37

Cytotoxic michael-type amine adducts of α-methylene lactones alantolactone and isoalantolactone

Nicholas J. Lawrence, Alan T. McGown, Jane Nduka, John A. Hadfield, Robin G. Pritchard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 138 KB

english, 2001

38

Nipecotic and iso-nipecotic amides as potent and selective somatostatin subtype-2 receptor agonists

Changyou Zhou, Liangqin Guo, Greg Morriello, Alex Pasternak, Yanping Pan, Susan P Rohrer, Elizebeth T Birzin, Su-Er Wu Huskey, Tom Jacks, Klaus D Schleim, Kang Cheng, James M Schaeffer, Arthur A Patch

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 172 KB

english, 2001

39

Equilibrium and kinetics studies of transnitrosation between S-nitrosothiols and thiols

Kun Wang, Zhong Wen, Wei Zhang, Ming Xian, Jin-Pei Cheng, Peng George Wang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 137 KB

english, 2001

40

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

File:

PDF, 44 KB

2001

41

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 555 KB

english, 2001

42

Instructions to contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 98 KB

english, 2001

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