Volume 11; Issue 6

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Bioorganic & Medicinal Chemistry Letters
Volume 11; Issue 6

Bioorganic & Medicinal Chemistry Letters

Volume 11; Issue 6

1

An improved synthesis of 1,2,4-oxadiazoles on solid support

Kenneth D. Rice, John M. Nuss

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 100 KB

english, 2001

2

The synthesis of cyclic tetrapeptoid analogues of the antiprotozoal natural product apicidin

Peter J Murray, Michael Kranz, Mark Ladlow, Stephen Taylor, Frédéric Berst, Andrew B Holmes, Kenneth N Keavey, Albert Jaxa-Chamiec, Peter W Seale, Paul Stead, Richard J Upton, Simon L Croft, William C

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 235 KB

english, 2001

3

Synthesis of phenylglycine derivatives as potent and selective antagonists of group III metabotropic glutamate receptors

Stuart J Conway, Jacqueline C Miller, Patrick A Howson, Barry P Clark, David E Jane

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 291 KB

english, 2001

4

Peptidomimetic inhibitors of protein farnesyltransferase show potent antimalarial activity

Junko Ohkanda, Jeffrey W. Lockman, Kohei Yokoyama, Michael H. Gelb, Simon L. Croft, Howard Kendrick, Maria Isabel Harrell, Jean E. Feagin, Michelle A. Blaskovich, Said M. Sebti, Andrew D. Hamilton

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 129 KB

english, 2001

5

Bisphosphonates derived from fatty acids are potent growth inhibitors of Trypanosoma cruzi

Sergio H. Szajnman, Brian N. Bailey, Roberto Docampo, Juan B. Rodriguez

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 141 KB

english, 2001

6

Phenylcyclohexene and phenylcyclohexadiene substituted compounds having retinoid antagonist activity

Richard L. Beard, Elliott S. Klein, Andrew M. Standeven, Maria Escobar, Roshantha A.S. Chandraratna

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 135 KB

english, 2001

7

Discovery of zoniporide: A potent and selective sodium–hydrogen exchanger type 1 (NHE-1) inhibitor with high aqueous solubility

Angel Guzman-Perez, Ronald T. Wester, Mary C. Allen, Janice A. Brown, Allan R. Buchholz, Ewell R. Cook, Wesley W. Day, Ernest S. Hamanaka, Scott P. Kennedy, Delvin R. Knight, Paul J. Kowalczyk, Ravi B

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 162 KB

english, 2001

8

Anti-MRSA cephems. Part 1: C-3 substituted thiopyridinium derivatives

Dane M. Springer, Bing-Yu Luh, Joanne J. Bronson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 224 KB

english, 2001

9

A novel fluorinated tryptamine with highly potent serotonin 5-HT1A receptor agonist properties

Uroš Laban, Deborah Kurrasch-Orbaugh, Danuta Marona-Lewicka, David E. Nichols

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 99 KB

english, 2001

10

2,4-thiazolidinediones as potent and selective human β3 agonists

Baihua Hu, John Ellingboe, Iwan Gunawan, Stella Han, Elwood Largis, Zenan Li, Michael Malamas, Ruth Mulvey, Alexander Oliphant, Fuk-Wah Sum, Jeff Tillett, Victoria Wong

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 149 KB

english, 2001

11

Design, synthesis, and intracellular localization of a fluorescently labeled DNA binding polyamide related to the antibiotic distamycin

Sanjay K. Sharma, Andrew T. Morrissey, Gerald G. Miller, William H. Gmeiner, J.William Lown

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 547 KB

english, 2001

12

Synthesis of metabolically blocked paclitaxel analogues

Mark D. Wittman, Thomas J. Altstadt, Craig Fairchild, Stephen Hansel, Kathy Johnston, John F. Kadow, Byron H. Long, William C. Rose, Dolatrai M. Vyas, Mu-Jen Wu, Mary E. Zoeckler

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 108 KB

english, 2001

13

Synthesis and antitumor activity of novel paclitaxel–chlorambucil hybrids

Mark D. Wittman, John F. Kadow, Dolatrai M. Vyas, Francis L. Lee, William C. Rose, Byron H. Long, Craig Fairchild, Kathy Johnston

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 194 KB

english, 2001

14

Effects of two-carbon bridge region methoxylation of benztropine: discovery of novel chiral ligands for the dopamine transporter

Daniele Simoni, Marinella Roberti, Riccardo Rondanin, Riccardo Baruchello, Marcello Rossi, Francesco Paolo Invidiata, Stefania Merighi, Katia Varani, Stefania Gessi, Pier Andrea Borea, Silvia Marino,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 153 KB

english, 2001

15

Synthesis and use of FSCPX, an irreversible adenosine A1 antagonist, as a ‘Receptor Knock-Down’ tool

Jacqueline E.van Muijlwijk-Koezen, Henk Timmerman, Richard P.van der Sluis, Andrea C van de Stolpe, Wiro M.P.B Menge, Margot W Beukers, Piet H van der Graaf, Miriam de Groote, Adriaan P IJzerman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 159 KB

english, 2001

16

Synthesis and characterization of Bis(μ-hydroxo)diiron(III) complex of N-(4-Nitro-2-hydroxy)phenylmethyl-N-(2-pyridylethyl)-N-(2-pyridylmethyl)amine and hydroxylation reaction of alkane

Hiromasa Kurosaki, Hiroyuki Yoshida, Masami Ito, Hiroyuki Koike, Eiko Higuchi, Masafumi Goto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 280 KB

english, 2001

17

An efficient conversion of 5-nitroisatin into 5-nitroindole derivative

Yasuhiro Torisawa, Takao Nishi, Jun-Ichi Minamikawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 172 KB

english, 2001

18

Structure elucidation and conformational properties of a novel bioactive clerodane diterpene using a combination of high field NMR spectroscopy, computational analysis and X-ray diffraction

Antonios Kolocouris, Thomas Mavromoustakos, Costas Demetzos, Aris Terzis, Simona Golic Grdadolnik

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 257 KB

english, 2001

19

NO-Independent stimulators of soluble guanylate cyclase

Alexander Straub, Johannes-Peter Stasch, Cristina Alonso-Alija, Jordi Benet-Buchholz, Bernhard Ducke, Achim Feurer, Chantal Fürstner

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 263 KB

english, 2001

20

Spatial requirements of the antagonist binding site of the NK2 receptor

Mohammed A. Ali, Nirmala Bhogal, Colin W.G. Fishwick, John B.C. Findlay

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 267 KB

english, 2001

21

Diaryl ester prodrugs of fR900098 with improved in vivo antimalarial activity

Armin Reichenberg, Jochen Wiesner, Claus Weidemeyer, Erhard Dreiseidler, Silke Sanderbrand, Boran Altincicek, Ewald Beck, Martin Schlitzer, Hassan Jomaa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 127 KB

english, 2001

22

N-Aminoindoline derivatives as inhibitors of 5-lipoxygenase

Corinne Audouin, Nathalie Mestdagh, Marie-Agnès Lassoie, Raymond Houssin, Jean-Pierre Hénichart

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 166 KB

english, 2001

23

7-Alkyl- and 7-Cycloalkyl-5-aryl-pyrrolo[2,3-d]pyrimidines—potent inhibitors of the tyrosine kinase c-Src

Leo Widler, Jonathan Green, Martin Missbach, Mira Šuša, Eva Altmann

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 142 KB

english, 2001

24

7-Pyrrolidinyl- and 7-piperidinyl-5-aryl-pyrrolo[2,3-d]pyrimidines—potent inhibitors of the tyrosine kinase c-Src

Eva Altmann, Martin Missbach, Jonathan Green, Mira Šuša, Hans-Achim Wagenknecht, Leo Widler

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 127 KB

english, 2001

25

Synthesis and in vitro cytotoxicity of novel long chain busulphan analogues

George Kokotos, Violetta Constantinou-Kokotou, José M Padrón, Godefridus J Peters

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 101 KB

english, 2001

26

Access to the inaccessible sequence of Cpn 60.1 (195–217) by temporary oxazolidine protection of selected amide bonds

Michael Keller, Andrew D. Miller

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 99 KB

english, 2001

27

Novel inhibitors of the enzyme estrone sulfatase (ES)

Sabbir Ahmed, Karen James, Caroline P Owen, Chirag K Patel, Mijal Patel

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 135 KB

english, 2001

28

Contributors to this Issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 37 KB

english, 2001

29

Instructions to Contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 94 KB

english, 2001

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