Volume 12; Issue 11

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Bioorganic & Medicinal Chemistry Letters
Volume 12; Issue 11

Bioorganic & Medicinal Chemistry Letters

Volume 12; Issue 11

1

Synthesis and cytotoxicity of 2α-amido docetaxel analogues

Wei-Shuo Fang, Ying Liu, Hong-Yan Liu, Shao-Feng Xu, Liang Wang, Qi-Cheng Fang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 119 KB

english, 2002

2

Scaffold hopping and optimization towards libraries of glycogen synthase kinase-3 inhibitors

Lars Nærum, Leif Nørskov-Lauritsen, Preben H Olesen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 117 KB

english, 2002

3

Identification of novel antifungal nonapeptides through the screening of combinatorial peptide libraries based on a hexapeptide motif

B Kundu, T Srinivasan, A. P Kesarwani, A Kavishwar, S. K Raghuwanshi, S Batra, P. K Shukla

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 145 KB

english, 2002

4

Nicotinanilides as inhibitors of neutrophil chemotaxis

Neil S. Cutshall, Kristin A. Kucera, Rocky Ursino, John Latham, Nathan C. Ihle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 126 KB

english, 2002

5

CoMFA and HQSAR of acylhydrazide cruzain inhibitors

Carlos R. Rodrigues, Terrence M. Flaherty, Clayton Springer, James H. McKerrow, Fred E. Cohen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 182 KB

english, 2002

6

Discovery of L-791,943: A potent, selective, non emetic and orally active phosphodiesterase-4 inhibitor

Daniel Guay, Pierre Hamel, Marc Blouin, Christine Brideau, Chi Chung Chan, Nathalie Chauret, Yves Ducharme, Zheng Huang, Mario Girard, Tom R. Jones, France Laliberté, Paul Masson, Malia McAuliffe, Han

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 151 KB

english, 2002

7

Tricarbocyanine cholesteryl laurates labeled LDL: new near infrared fluorescent probes (NIRFs) for monitoring tumors and gene therapy of familial hypercholesterolemia

Gang Zheng, Hui Li, Kathy Yang, Dana Blessington, Kai Licha, Sissel Lund-Katz, Britton Chance, Jerry D. Glickson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 170 KB

english, 2002

8

Novel bicyclic oxazolone derivatives as anti-Angiogenic agents

Françoise M Perron-Sierra, Alain Pierré, Mike Burbridge, Nicolas Guilbaud

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 126 KB

english, 2002

9

Design, synthesis, and SAR of substituted acrylamides as factor Xa inhibitors

Yonghong Song, Lane Clizbe, Chhaya Bhakta, Willy Teng, Wenhao Li, Yanhong Wu, Zhaozhong Jon Jia, Penglie Zhang, Lingyan Wang, Brandon Doughan, Ting Su, James Kanter, John Woolfrey, Paul Wong, Brian Hu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 169 KB

english, 2002

10

Glycosidation of alkylamino-alkan-1-ol. A simple and convenient synthesis of glycosylated cationic lipids

Christophe Jacopin, Marie-José Egron, Daniel Scherman, Jean Herscovici

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 124 KB

english, 2002

11

CDP840. A prototype of a novel class of orally active anti-Inflammatory phosphodiesterase 4 inhibitors

R.P. Alexander, G.J. Warrellow, M.A.W. Eaton, E.C. Boyd, J.C. Head, J.R. Porter, J.A. Brown, J.T. Reuberson, B. Hutchinson, P. Turner, B. Boyce, D. Barnes, B. Mason, A. Cannell, R.J. Taylor, A. Zomaya

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 166 KB

english, 2002

12

Novel phthalimide derivatives, designed as leukotriene D4 receptor antagonists

Lı́dia M. Lima, Fernanda C.F. de Brito, Simone D. de Souza, Ana L.P. Miranda, Carlos R. Rodrigues, Carlos A.M. Fraga, Eliezer J. Barreiro

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 145 KB

english, 2002

13

Synthesis of more potent analogues of the acetylcholinesterase inhibitor, huperzine B

V. Rajendran, Ashima Saxena, Bhupendra P. Doctor, Alan P. Kozikowski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 104 KB

english, 2002

14

Structure–Activity studies for a novel series of tricyclic dihydropyrimidines as KATP channel openers (KCOs)

Irene Drizin, Mark W. Holladay, Lin Yi, Henry Q. Zhang, Sujatha Gopalakrishnan, Murali Gopalakrishnan, Kristi L. Whiteaker, Steven A. Buckner, James P. Sullivan, William A. Carroll

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 121 KB

english, 2002

15

Synthesis of TDP-3-amino-3,4,6-trideoxy-α-d-xylo-hexopyranose—The immediate precursor of TDP-α-d-desosamine

Cheng-Wei T. Chang, Hung-wen Liu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 152 KB

english, 2002

16

Substituted tetrahydrofuroyl-1-phenylalanine derivatives as potent and specific VLA-4 antagonists

George A. Doherty, Ginger X. Yang, Edite Borges, Linda L. Chang, Malcolm MacCoss, Sharon Tong, Usha Kidambi, Linda A. Egger, Ermenegilda McCauley, Gail Van Riper, Richard A. Mumford, John A. Schmidt,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 147 KB

english, 2002

17

2-Amino-α-2′-deoxyadenosine increased duplex stability of methoxyethylphosphoramidate α-Oligodeoxynucleotides with RNA target

Magali Naval, Thibaut Michel, Jean-Jacques Vasseur, Françoise Debart

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 120 KB

english, 2002

18

Novel lipoic acid analogues that inhibit nitric oxide synthase

Jeremiah J Harnett, Michel Auguet, Isabelle Viossat, Christine Dolo, Dennis Bigg, Pierre-E Chabrier

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 108 KB

english, 2002

19

Design and synthesis of some new pyranoxanthenone aminoderivatives with cytotoxic activity

George Kolokythas, Ioannis K. Kostakis, Nicole Pouli, Panagiotis Marakos, Alexios-Leandros Skaltsounis, Harris Pratsinis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 122 KB

english, 2002

20

Contributors to this Issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 42 KB

english, 2002

21

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 182 KB

english, 2002

22

Cytotoxic alpha-Bromoacrylic derivatives of low molecular weight

Italo Beria, Marina Caldarelli, Cristina Geroni, Nicola Mongelli, Benedetta Reinach, Luisella Vignati, Paolo Cozzi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 113 KB

english, 2002

23

Electrochemical and peroxidase oxidation study of N′-Hydroxyguanidine derivatives as NO donors

Tingwei Cai, Ming Xian, Peng George Wang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 116 KB

english, 2002

24

9-[(Hydroxymethyl)phenyl]adenines: new aryladenine substrates of adenosine deaminase

Mohamed Brakta, Devangachinta Murthy, L'Ouverture Ellis, Shashikant Phadtare

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 120 KB

english, 2002

25

Doxorubicin immunoconjugates containing bivalent, lysosomally-Cleavable dipeptide linkages

Gene M Dubowchik, Shilpa Radia, Harold Mastalerz, Michael A Walker, Raymond A Firestone, H Dalton King, Sandra J Hofstead, David Willner, Shirley J Lasch, Pamela A Trail

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 133 KB

english, 2002

26

SAR and species/stereo-selective metabolism of the sorbitol dehydrogenase inhibitor, CP-470,711

Margaret Y. Chu-Moyer, William E. Ballinger, David A. Beebe, James B. Coutcher, Wesley W. Day, Jiancheng Li, Peter J. Oates, R.Matthew Weekly

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 132 KB

english, 2002

27

N-Tetrahydrofuroyl-(l)-phenylalanine derivatives as potent VLA-4 antagonists

Ginger X. Yang, Linda L. Chang, Quang Truong, George A. Doherty, Plato A. Magriotis, Stephen E. de Laszlo, Bing Li, Malcolm MacCoss, Usha Kidambi, Linda A. Egger, Ermengilda McCauley, Gail Van Riper,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 133 KB

english, 2002