Volume 12; Issue 13

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Bioorganic & Medicinal Chemistry Letters
Volume 12; Issue 13

Bioorganic & Medicinal Chemistry Letters

Volume 12; Issue 13

1

CCR3 antagonists: a potential new therapy for the treatment of asthma. Discovery and structure–activity relationships

Dean A Wacker, Joseph B Santella, III, Daniel S Gardner, Jeffrey G Varnes, Melissa Estrella, George V DeLucca, Soo S Ko, Keiichi Tanabe, Paul S Watson, Patricia K Welch, Maryanne Covington, Nicole C S

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 136 KB

english, 2002

2

Structure-based design and synthesis of HIV-1 protease inhibitors employing β-d-mannopyranoside scaffolds

Paul V. Murphy, Julie L. O'Brien, Lorraine J. Gorey-Feret, Amos B. Smith III

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 133 KB

english, 2002

3

Discovery of substituted 3,4-Diphenyl-thiazoles as a novel class of monoamine transporter inhibitors through 3-D pharmacophore search using a new pharmacophore model derived from mazindol

Istvan J Enyedy, Jiansuo Wang, Wahiduz A Zaman, Kenneth M Johnson, Shaomeng Wang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 160 KB

english, 2002

4

4,4-Disubstituted cyclohexylamine NK1 receptor antagonists I

Jason M Elliott, Jose L Castro, Gary G Chicchi, Laura C Cooper, Kevin Dinnell, Gregory J Hollingworth, Mark P Ridgill, Wayne Rycroft, Marc M Kurtz, Duncan E Shaw, Christopher J Swain, Kwei-Lan Tsao, L

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 144 KB

english, 2002

5

4,4-Disubstituted cyclohexylamine NK1 receptor antagonists II

Laura C Cooper, Emma J Carlson, Jose L Castro, Gary G Chicchi, Kevin Dinnell, Jerry Di Salvo, Jason M Elliott, Gregory J Hollingworth, Marc M Kurtz, Mark P Ridgill, Wayne Rycroft, Kwei-Lan Tsao, Chris

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 148 KB

english, 2002

6

Synthesis of triazole-Tethered pyrrolidine libraries: novel ECE inhibitors

Eric A Kitas, Bernd-Michael Löffler, Stefan Daetwyler, Henrietta Dehmlow, Johannes D Aebi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 106 KB

english, 2002

7

Efficient chemoenzymatic synthesis of (S)- and (R)-5-(1-Aminoethyl)-2-(cyclohexylmethoxy)benzamide: key intermediate for Src-SH2 inhibitor

Ahmed Kamal, Mahendra Sandbhor

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 119 KB

english, 2002

8

Synthesis and antifungal activity of the 2,2,5-tetrahydrofuran regioisomers of SCH 51048

Raymond G Lovey, Anil K Saksena, Viyyoor M Girijavallabhan, Paul Blundell, Henry Guzik, David Loebenberg, Raulo M Parmegiani, Anthony Cacciapuoti

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 151 KB

english, 2002

9

Discovery of imidazole glycerol phosphate dehydratase inhibitors through 3-D database searching

Barbara A Schweitzer, Paul J Loida, Claire A CaJacob, Robert C Chott, Elizabeth M Collantes, Shridhar G Hegde, Philip D Mosier, Salvatore Profeta

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 117 KB

english, 2002

10

Discovery of potent and selective small molecule NPY Y5 receptor antagonists

Imadul Islam, Dale Dhanoa, John Finn, Ping Du, Mary W Walker, John A Salon, Jack Zhang, Charles Gluchowski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 134 KB

english, 2002

11

Design, synthesis, and evaluation of postulated transient intermediate and substrate analogues as inhibitors of 4-hydroxyphenylpyruvate dioxygenase

Yun-Loung Lin, Jian-Lin Huang, Chung-Shieh Wu, Hung-Ge Liu, Ding-Yah Yang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 143 KB

english, 2002

12

A convenient synthetic pathway for multivalent assembly of aminoglycoside antibiotics starting from amikacin

Hidehiko Tanaka, Yoshihiro Nishida, Yousuke Furuta, Kazukiyo Kobayashi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 128 KB

english, 2002

13

Antifungal sordarins. Part 4: synthesis and structure–activity relationships of 3′,4′-fused alkyl-tetrahydrofuran derivatives

José M Bueno, Jesús Chicharro, José M Fiandor, Federico Gómez de las Heras, Sophie Huss

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 147 KB

english, 2002

14

Pyrrolidine-5,5-trans-lactams as novel mechanism-based inhibitors of human cytomegalovirus protease. Part 3: potency and plasma stability

Alan D Borthwick, Anne M Exall, Terry M Haley, Deborah L Jackson, Andrew M Mason, Gordon G Weingarten

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 129 KB

english, 2002

15

Graphical abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 164 KB

english, 2002

16

The synthesis and structure–activity relationships of 4-aryl-3-aminoquinolin-2-ones: a new class of calcium-Dependent, large conductance, potassium (maxi-K) channel openers targeted for post-stroke neuroprotection

Piyasena Hewawasam, Wenhong Fan, Jay Knipe, Sandra L Moon, Christopher G Boissard, Valentin K Gribkoff, John E Starrett Jr.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 127 KB

english, 2002

17

A new lipophilic fluorescent probe for interaction studies of bioactive lipopeptides with membrane models

Elisa Peroni, Gabriella Caminati, Piero Baglioni, Francesca Nuti, Mario Chelli, Anna M Papini

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 136 KB

english, 2002

18

A Library Construction of 2,5-Disubstituted Pyrrole Compounds by Using Solid/Solution-Phase Syntheses

Naoki Kobayashi, Yumiko Kaku, Kunizo Higurashi, Toshihiko Yamauchi, Akira Ishibashi, Yasushi Okamoto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 146 KB

english, 2002

19

Side-chain homologation of nodulisporic acid: synthesis of potent new dienyl derivatives

Dong Ok, Chunshi Li, Thomas L. Shih, Steve Salva, Michelle B. Ayer, Steven L. Colletti, Prasun K. Chakravarty, Matthew J. Wyvratt, Michael H. Fisher, Lynn Gregory, Michelle Zakson-Aiken, Wesley L. Sho

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 126 KB

english, 2002

20

High-throughput synthesis optimization of sulfonamide NPY Y5 antagonists

John Finn, David Pelham, Mary W. Walker, Charles Gluchowski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 120 KB

english, 2002

21

Antimalarial activities of ring-substituted bioimidazoles

Rahul Jain, Suryanarayana Vangapandu, Meenakshi Jain, Navneet Kaur, Savita Singh, Prati Pal Singh

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 98 KB

english, 2002

22

Synthesis and evaluation of N-substituted 1,4-oxazepanyl sordaricins as selective fungal EF-2 inhibitors

Satoru Kaneko, Masami Arai, Takuya Uchida, Tamako Harasaki, Takashi Fukuoka, Toshiyuki Konosu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 132 KB

english, 2002

23

New ketosteroids from the red alga Hypnea musciformis

V. Bultel-Poncé, S. Etahiri, M. Guyot

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 99 KB

english, 2002

24

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 40 KB

english, 2002

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