Volume 12; Issue 2

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Bioorganic & Medicinal Chemistry Letters
Volume 12; Issue 2

Bioorganic & Medicinal Chemistry Letters

Volume 12; Issue 2

1

Effects of the incorporation of IBTM β-turn mimetics into the dipeptoid CCK1 receptor agonist PD 170292

Mercedes Martı́n-Martı́nez, Miriam Latorre, M.Teresa Garcı́a-López, Edurne Cenarruzabeitia, Joaquı́n Del Rı́o, Rosario González-Muñiz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 122 KB

english, 2002

2

The design and synthesis of a novel series of indole derived selective ETA antagonists

David J Rawson, Kevin N Dack, Roger P Dickinson, Kim James

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 131 KB

english, 2002

3

Anti-MRSA activity of alkyl gallates

Isao Kubo, Ping Xiao, Ken'ichi Fujita

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 97 KB

english, 2002

4

Synthesis and biological activity of 8β-substituted hydrocodone indole and hydromorphone indole derivatives

Han Yu, Thomas Prisinzano, Christina M. Dersch, Jamila Marcus, Richard B. Rothman, Arthur E. Jacobson, Kenner C. Rice

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 112 KB

english, 2002

5

Mixed lineage kinase activity of indolocarbazole analogues

Chikara Murakata, Masami Kaneko, George Gessner, Thelma S Angeles, Mark A Ator, Teresa M O'Kane, Beth Ann W McKenna, Beth Ann Thomas, Joanne R Mathiasen, Michael S Saporito, Donna Bozyczko-Coyne, Robe

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 164 KB

english, 2002

6

3-Aryl pyridone derivatives. Potent and selective kappa opioid receptor agonists

Graeme Semple, Britt-Marie Andersson, Vijay Chhajlani, Jennie Georgsson, Magnus Johansson, Marcel Lindschoten, Fritof Pontén, Åsa Rosenquist, Henrik Sörensen, Lars Swanson, Marianne Swanson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 113 KB

english, 2002

7

Solid-Phase synthesis of new saphenamycin analogues with antimicrobial activity

Jane B Laursen, Peter C de Visser, Henrik K Nielsen, Knud J Jensen, John Nielsen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 126 KB

english, 2002

8

Synthesis and pharmacology of isoquinuclidine derivatives as 5-HT3 ligands

Isabel Iriepa, Francisco J Villasante, Enrique Gálvez, Luis Labeaga, Ana Innerarity, Aurelio Orjales

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 113 KB

english, 2002

9

An improved procedure for the synthesis of branched polyethylene glycols (PEGs) with the reporter dipeptide met-βala for protein conjugation

Andrea Guiotto, Michela Pozzobon, Chiara Sanavio, Oddone Schiavon, Piero Orsolini, Francesco M Veronese

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 114 KB

english, 2002

10

Selective urokinase-type plasminogen activator (uPA) inhibitors. Part 1: 2-Pyridinylguanidines

Christopher G Barber, Roger P Dickinson, Valerie A Horne

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 151 KB

english, 2002

11

Selective urokinase-type plasminogen activator (uPA) inhibitors. Part 2: (3-Substituted-5-halo-2-pyridinyl)guanidines

Christopher G Barber, Roger P Dickinson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 107 KB

english, 2002

12

Oxyaniliniums as acetylcholinesterase inhibitors for the reversal of neuromuscular block

Simon J.A. Grove, Jasmit Kaur, Alan W. Muir, Eleanor Pow, Gary J. Tarver, Ming-Qiang Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 107 KB

english, 2002

13

Specific and dual antagonists of α4β1 and α4β7 integrins

Linus S. Lin, Thomas Lanza Jr., Ermenegilda McCauley, Gail Van Riper, Usha Kidambi, Jin Cao, Linda A. Egger, Richard A. Mumford, John A. Schmidt, Malcolm MacCoss, William K. Hagmann

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 129 KB

english, 2002

14

Synthesis and biological activities of ykfa analogues: effects of position 4 substitutions and altered ring size on In vitro opioid activity

John E Burden, Peg Davis, Frank Porreca, Arno F Spatola

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 97 KB

english, 2002

15

Synthesis of an immunoconjugate of camptothecin

Michael A Walker, Gene M Dubowchik, Sandra J Hofstead, Pamela A Trail, Raymond A Firestone

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 112 KB

english, 2002

16

Facile synthesis of β-Cyclodextrin dithiols

Jerry Yang, David K Leung

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 130 KB

english, 2002

17

Synthesis and structure–activity relationships of oxime neurokinin antagonists: discovery of potent arylamides

Neng-Yang Shih, Margaret Albanese, John C Anthes, Nicholas I Carruthers, Cheryl A Grice, Ling Lin, Pietro Mangiaracina, Gregory A Reichard, John Schwerdt, Vera Seidl, Shing-Chung Wong, John J Piwinski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 160 KB

english, 2002

18

The discovery of small molecule carbamates as potent dual α4β1/α4β7 integrin antagonists

Linda L. Chang, Quang Truong, Richard A. Mumford, Linda A. Egger, Usha Kidambi, Kathryn Lyons, Ermengilda McCauley, Gail Van Riper, Stella Vincent, John A. Schmidt, Malcolm MacCoss, William K. Hagmann

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 132 KB

english, 2002

19

N-Acyl-l-phenylalanine derivatives as potent VLA-4 antagonists that mimic a cyclic peptide conformation

Li Chen, Jefferson Tilley, Richard V. Trilles, Weiya Yun, David Fry, Charles Cook, Karen Rowan, Virginia Schwinge, Robert Campbell

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 152 KB

english, 2002

20

An N1–Hydrogen bonding model for flavin coenzyme

Fengli Guo, Bryan H. Chang, Carmelo J. Rizzo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 153 KB

english, 2002

21

Evaluation of isotryptamine derivatives at 5-HT2 serotonin receptors

Jean Chang-Fong, James Addo, Małgorzata Dukat, Carol Smith, Nicholas A. Mitchell, Katharine Herrick-Davis, Milt Teitler, Richard A. Glennon

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 115 KB

english, 2002

22

Potent In vitro methicillin-resistant Staphylococcus aureus activity of 2-(1H-indol-3-yl)tetrahydroquinoline derivatives

Michael Z. Hoemann, Roger L. Xie, Richard F. Rossi, Sylvia Meyer, Alban Sidhu, Gregory D. Cuny, James R. Hauske

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 173 KB

english, 2002

23

Structure-based design and protein X-ray analysis of a protein kinase inhibitor

Pascal Furet, Thomas Meyer, André Strauss, Sylvie Raccuglia, Jean-Michel Rondeau

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 219 KB

english, 2002

24

New series of aryloxypropanolamines with both human β3-adrenoceptor agonistic activity and free radical scavenging properties

Silvère Aubriot, Edwige Nicolle, Mireille Lattier, Cécile Morel, Wenhong Cao, Kiefer W. Daniel, Sheila Collins, Gérard Leclerc, Patrice Faure

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 117 KB

english, 2002

25

Biphenyls as potent vitronectin receptor antagonists

Klaus Urbahns, Michael Härter, Markus Albers, Delf Schmidt, Beatrix Stelte-Ludwig, Ulf Brüggemeier, Andrea Vaupel, Christoph Gerdes

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 127 KB

english, 2002

26

Cyclic acid anhydrides as a new class of potent, selective and non-peptidic inhibitors of geranylgeranyl transferase

Charles M. Marson, Alphonso S. Rioja, Greg Brooke, R.Charles Coombes, David M. Vigushin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 135 KB

english, 2002

27

Polyhydroxylated azepanes as new motifs for DNA minor groove binding agents

Heather A Johnson, Neil R Thomas

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 126 KB

english, 2002

28

Synthesis of 4-(8-benzo[1,2,5]oxadiazol-5-yl-[1,7]naphthyridine-6-yl)-benzoic acid: a potent and selective phosphodiesterase type 4D inhibitor

Rene Hersperger, Janet Dawson, Thomas Mueller

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 128 KB

english, 2002

29

Synthesis and structure–activity relationship of 2-(aminoalkyl)-2,3,3a,8-tetrahydrodibenzo[c,f]isoxazolo[2,3-a]azepine derivatives: a novel series of 5-HT2A/2C receptor antagonists. Part 1

J.Ignacio Andrés, Jesús Alcázar, José M Alonso, Adolfo Dı́az, Javier Fernández, Pilar Gil, Laura Iturrino, Encarna Matesanz, Theo F Meert, Anton Megens, Victor K Sipido

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 145 KB

english, 2002

30

Synthesis and structure–Activity relationship of 2-(aminoalkyl)-2,3,3a,8-tetrahydrodibenzo[c,f]isoxazolo[2,3-a]azepine derivatives: a novel series of 5-HT2A/2C receptor antagonists. Part 2

J Ignacio Andrés, Jesús Alcázar, José M Alonso, Adolfo Dı́az, Javier Fernández, Pilar Gil, Laura Iturrino, Encarna Matesanz, Theo F Meert, Anton Megens, Victor K Sipido

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 134 KB

english, 2002

31

N-Methylbenzanilide derivatives as a novel class of selective V1A receptor antagonists

Akio Kakefuda, Junko Tsukada, Toshiyuki Kusayama, Atsuo Tahara, Shin-ichi Tsukamoto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 140 KB

english, 2002

32

Theoretical elucidation on structure–Antioxidant activity relationships for indolinonic hydroxylamines

Hong-Yu Zhang, Lan-Fen Wang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 93 KB

english, 2002

33

DNA cleavage by pentadentate iron(II) complexes containing fluoro-substituted phenyl groups

Hiromasa Kurosaki, Aoi Maruyama, Hiroyuki Koike, Naoko Kuroda, Yoshinobu Ishikawa, Masafumi Goto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 150 KB

english, 2002

34

First dual NK1 antagonists–serotonin reuptake inhibitors: synthesis and SAR of a new class of potential antidepressants

Thomas Ryckmans, Laurent Balançon, Olivier Berton, Christophe Genicot, Yves Lamberty, Benedicte Lallemand, Patrick Pasau, Nathalie Pirlot, Luc Quéré, Patrice Talaga

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 113 KB

english, 2002

35

Increase of the adenallene anti-HIV activity in cell culture using its bis(tBuSATE) phosphotriester derivative

David Egron, Christian Périgaud, Gilles Gosselin, Anne-Marie Aubertin, Hiroyuki Gatanaga, Hiroaki Mitsuya, Jiri Zemlicka, Jean-Louis Imbach

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 81 KB

english, 2002

36

Antifungal sordarins. Synthesis and structure–activity relationships of 3′-O-Substituted derivatives

Enrique M Arribas, Julia Castro, Ian R Clemens, Juan C Cuevas, Jesús Chicharro, Mª Teresa Fraile, Silvestre Garcı́a-Ochoa, Federico Gómez de las Heras, José R Ruiz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 115 KB

english, 2002

37

Antifungal sordarins. Synthesis and structure–activity relationships of 3′,4′-Fused dioxolane and dioxane derivatives

José M Bueno, Juan C Cuevas, José M Fiandor, Silvestre Garcı́a-Ochoa, Federico Gómez de las Heras

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 138 KB

english, 2002

38

Instructions to Contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 96 KB

english, 2002

39

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 262 KB

english, 2002

40

Contributors to this Issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 44 KB

english, 2002

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