Volume 12; Issue 5

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Bioorganic & Medicinal Chemistry Letters
Volume 12; Issue 5

Bioorganic & Medicinal Chemistry Letters

Volume 12; Issue 5

1

New 2-(1-adamantylcarbonyl)pyridine and 1-acetyladamantane thiosemicarbazones–thiocarbonohydrazones: cell growth inhibitory, antiviral and antimicrobial activity evaluation

Antonios Kolocouris, Kostas Dimas, Christophe Pannecouque, Myriam Witvrouw, George B. Foscolos, George Stamatiou, George Fytas, Grigoris Zoidis, Nicolas Kolocouris, Graciela Andrei, Robert Snoeck, Eri

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 154 KB

english, 2002

2

Novel potent antagonists of human neuropeptide Y Y5 receptors. Part 2: substituted benzo[a]cycloheptene derivatives

Hiromichi Itani, Harunobu Ito, Yoshihiko Sakata, Yoshifumi Hatakeyama, Hiroko Oohashi, Yoshinari Satoh

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 154 KB

english, 2002

3

Anti-HIV-1 Activities and Pharmacokinetics of New Arylpiperazinyl Fluoroquinolones

Toshinori Ohmine, Tetsushi Katsube, Yasunori Tsuzaki, Miho Kazui, Nobuhiro Kobayashi, Tomoaki Komai, Masahiko Hagihara, Takashi Nishigaki, Aikichi Iwamoto, Tomio Kimura, Hiroto Kashiwase, Makoto Yamas

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 118 KB

english, 2002

4

Synthesis of an α-Fucosidase Inhibitor, 5a-Carba-β-l-fucopyranosylamine, and Fucose-Type α- and β-dl-Valienamine Unsaturated Derivatives

Seiichiro Ogawa, Maiko Watanabe, Ayako Maruyama, Seiichi Hisamatsu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 124 KB

english, 2002

5

Novel Agents Combining Platelet Activating Factor (PAF) Receptor Antagonist with Thromboxane Synthase Inhibitor (TxSI)

Masakazu Fujita, Taketsugu Seki, Haruaki Inada, Kazuhiro Shimizu, Akane Takahama, Tetsuro Sano

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 126 KB

english, 2002

6

Peptidomimetics of Efflux Pump Inhibitors Potentiate the Activity of Levofloxacin in Pseudomonas aeruginosa

Thomas E. Renau, Roger Léger, Rose Yen, Miles W. She, Eric M. Flamme, Joan Sangalang, Carla L. Gannon, Suzanne Chamberland, Olga Lomovskaya, Ving J. Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 156 KB

english, 2002

7

Benzamide-Based Thiolcarbamates: A New Class of HIV-1 NCp7 Inhibitors

Atul Goel, Sharlyn J. Mazur, Rasem J. Fattah, Tracy L. Hartman, Jim A. Turpin, Mingjun Huang, William G. Rice, Ettore Appella, John K. Inman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 104 KB

english, 2002

8

Structure-Based Design, Synthesis, and Biological Evaluation of Irreversible Human Rhinovirus 3C Protease Inhibitors. Part 7: Structure–Activity Studies of Bicyclic 2-Pyridone-Containing Peptidomimetics

Peter S. Dragovich, Thomas J. Prins, Ru Zhou, Theodore O. Johnson, Edward L. Brown, Fausto C. Maldonado, Shella A. Fuhrman, Leora S. Zalman, Amy K. Patick, David A. Matthews, Xinjun Hou, James W. Mead

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 181 KB

english, 2002

9

The Synthesis and Selective IL-2 Inhibitory Activity of Bis Piperazine–Phenol Mannich Adducts

Bolin Geng, Paul R Fleming, Scott Umlauf, Augustine Lin, Peter V Pallai

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 115 KB

english, 2002

10

Synthesis and Activity of a New Methoxytetrahydropyran Derivative as Dual Cyclooxygenase-2/5-Lipoxygenase Inhibitor

Sabine Barbey, Laurence Goossens, Thierry Taverne, Joséphine Cornet, Valérie Choesmel, Céline Rouaud, Gilles Gimeno, Sylvie Yannic-Arnoult, Catherine Michaux, Caroline Charlier, Raymond Houssin, Jean-

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 160 KB

english, 2002

11

Synthesis and Vasorelaxant Activity of New Coumarin and Furocoumarin Derivatives

Manuel Campos-Toimil, Francisco Orallo, Lourdes Santana, Eugenio Uriarte

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 131 KB

english, 2002

12

Assamicin I and II, Novel Triterpenoid Saponins with Insulin-Like Activity from Aesculus assamica Griff.

Takashi Sakurai, Toshio Nishimura, Noboru Otake, Yao Xinsheng, Keiichi Abe, Mitsuhiro Zeida, Hiromichi Nagasawa, Shohei Sakuda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 93 KB

english, 2002

13

Synthesis and antiplatelet activity of gemfibrozil chiral analogues

Alessandra Ammazzalorso, Rosa Amoroso, Mario Baraldi, Giancarlo Bettoni, Daniela Braghiroli, Barbara De Filippis, Andrea Duranti, Marco Moretti, Paolo Tortorella, Maria Luisa Tricca, Francesca Vezzali

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 132 KB

english, 2002

14

Substituted 2-(R)-Methyl piperazines as muscarinic M2 selective ligands

Joseph A Kozlowski, Guowei Zhou, Jayaram R Tagat, Sue-Ing Lin, Stuart W McCombie, Vilma B Ruperto, Ruth A Duffy, Robert A McQuade, Gordon Crosby Jr., Lisa A Taylor, William Billard, Herbert Binch III,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 127 KB

english, 2002

15

Synthesis and structure–Activity relationships of M2-Selective muscarinic receptor ligands in the 1-[4-(4-Arylsulfonyl)-phenylmethyl]-4-(4-piperidinyl)-piperazine family

Stuart W McCombie, Sue-Ing Lin, Jayaram R Tagat, Dennis Nazareno, Susan Vice, Jennifer Ford, Theodros Asberom, Daria Leone, Joseph A Kozlowski, Guowei Zhou, Vilma B Ruperto, Ruth A Duffy, Jean E Lacho

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 118 KB

english, 2002

16

2-Arylindoles as gonadotropin releasing hormone (GnRH) antagonists: optimization of the tryptamine side chain

Jonathan R. Young, Song X. Huang, Thomas F. Walsh, Matthew J. Wyvratt Jr., Yi Tien Yang, Joel B. Yudkovitz, Jisong Cui, George R. Mount, Rena Ning Ren, Tsuei-Ju Wu, Xiaolan Shen, Kathryn A. Lyons, An-

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 217 KB

english, 2002

17

Structure–Activity relationships of oxime neurokinin antagonists: oxime modifications

Gregory A Reichard, James Spitler, Robert Aslanian, Mwangi wa Mutahi, Neng-Yang Shih, Ling Lin, Pauline C Ting, John C Anthes, John J Piwinski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 117 KB

english, 2002

18

Instructions to Contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 97 KB

english, 2002

19

Contributors to this Issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 41 KB

english, 2002

20

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 189 KB

english, 2002

21

N-Aryl 2,6-Dimethoxybiphenylalanine Analogues as VLA-4 Antagonists

George A Doherty, Theodore Kamenecka, Ermenegilda McCauley, Gail Van Riper, Richard A Mumford, Sharon Tong, William K Hagmann

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 122 KB

english, 2002

22

Novel, Potent Non-Covalent Thrombin Inhibitors Incorporating P3-Lactam Scaffolds

Jonathan Z Ho, Tony S Gibson, J.Edward Semple

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 175 KB

english, 2002

23

Anionic Cyclophanes as Potential Reversal Agents of Muscle Relaxants by Chemical Chelation

Kenneth S. Cameron, Lee Fielding, Rona Mason, Alan W. Muir, David C. Rees, Simon Thorn, Ming-Qiang Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 107 KB

english, 2002

24

Novel Potent Antagonists of Human Neuropeptide Y Y5 Receptors. Part 3: 7-Methoxy-1-hydroxy-1-substituted Tetraline Derivatives

Hiromichi Itani, Harunobu Ito, Yoshihiko Sakata, Yoshifumi Hatakeyama, Hiroko Oohashi, Yoshinari Satoh

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 145 KB

english, 2002

25

Synthesis of Sordaricin Analogues as Potent Antifungal Agents against Candida albicans

Satoru Kaneko, Takuya Uchida, Satoshi Shibuya, Takeshi Honda, Isao Kawamoto, Tamako Harasaki, Takashi Fukuoka, Toshiyuki Konosu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 128 KB

english, 2002

26

Cytotoxic, antifouling bromotyramines: A synthetic study on simple marine natural products and Their analogues

Ryan C. Schoenfeld, Susan Conova, Daniel Rittschof, Bruce Ganem

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 95 KB

english, 2002

27

Potent nonsteroidal progesterone receptor agonists: Synthesis and SAR study of 6-aryl benzoxazines

Puwen Zhang, Eugene A. Terefenko, Andrew Fensome, Zhiming Zhang, Yuan Zhu, Jeffrey Cohen, Richard Winneker, Jay Wrobel, John Yardley

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 120 KB

english, 2002

28

Syntheses and binding affinities of 6-nitroquipazine analogues for serotonin transporter. part 2: 4-Substituted 6-nitroquipazines

Byoung Se Lee, Soyoung Chu, Bon-Su Lee, Dae Yoon Chi, Yun Seon Song, Changbae Jin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 134 KB

english, 2002

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