Volume 12; Issue 6

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Bioorganic & Medicinal Chemistry Letters
Volume 12; Issue 6

Bioorganic & Medicinal Chemistry Letters

Volume 12; Issue 6

1

Stereoselective Synthesis of Ψ[CH2O] Pseudodipeptides and Conformational Analysis of a PheΨ[CH2O]Ala Containing Analogue of the Drug Desmopressin

Mattias Hedenström, Lotta Holm, ZhongQing Yuan, Hans Emtenäs, Jan Kihlberg

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 144 KB

english, 2002

2

Benzene fused monocyclic enediynyl amides: synthesis, reactivity and DNA-Cleavage activity in comparison to the corresponding sulfonamides

Amit Basak, Subrata Mandal, Amit Kumar Das, Valerio Bertolasi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 257 KB

english, 2002

3

Biphenyls as potential mimetics of protein α-helix

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 120 KB

english, 2002

4

Structure–Activity Study of l-Cysteine-Based N-Type Calcium Channel Blockers: Optimization of N- and C-Terminal Substituents

Takuya Seko, Masashi Kato, Hiroshi Kohno, Shizuka Ono, Kazuya Hashimura, Hideyuki Takimizu, Katsuhiko Nakai, Hitoshi Maegawa, Nobuo Katsube, Masaaki Toda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 124 KB

english, 2002

5

Chemical synthesis and calcium release activity of N1-ether strand substituted cADPR mimic

Li-Jun Huang, Yong-Yuan Zhao, Lan Yuan, Ji-Mei Min, Li-He Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 120 KB

english, 2002

6

Synthesis, Characterization and Antiamoebic Activity of Benzimidazole Derivatives and Their Vanadium and Molybdenum Complexes

Neelam Bharti, Shailendra, M.T. Gonzalez Garza, Delia E. Cruz-Vega, J. Castro-Garza, Kishwar Saleem, Fehmida Naqvi, Mannar R. Maurya, Amir Azam

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 102 KB

english, 2002

7

Highly Potent Inhibitors of TNF-α Production. Part 1: Discovery of Chemical Leads

Toshiaki Matsui, Takashi Kondo, Yoshitaka Nishita, Satoshi Itadani, Shingo Nakatani, Nagashige Omawari, Masaru Sakai, Shuichi Nakazawa, Akihito Ogata, Hiroyuki Ohno, Takaaki Obata, Hisao Nakai, Masaak

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 96 KB

english, 2002

8

Highly potent inhibitors of TNF-α production. Part 2: identification of drug candidates

Toshiaki Matsui, Takashi Kondo, Yoshitaka Nishita, Satoshi Itadani, Hiroshi Tsuruta, Setsuko Fujita, Nagashige Omawari, Masaru Sakai, Shuichi Nakazawa, Akihito Ogata, Hideaki Mori, Hiroyuki Ohno, Taka

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 121 KB

english, 2002

9

Evaluation of Morphogenic Regulatory Activity of Farnesoic acid and Its Derivatives against Candida albicans Dimorphism

Sanghee Kim, Eunkyung Kim, Dong-Sun Shin, Heonjoong Kang, Ki-Bong Oh

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 118 KB

english, 2002

10

QSAR study on adenosine kinase inhibition of pyrrolo[2,3-d]pyrimidine nucleoside analogues using the hansch approach

K Srikanth, Bikash Debnath, Tarun Jha

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 99 KB

english, 2002

11

Synthesis and antibacterial activity of linezolid analogues

Du Yu, Guo Huiyuan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 93 KB

english, 2002

12

Hydrophobic modifications at 1-phosphate of inositol 1,4,5-Trisphosphate analogues enhance receptor binding

Waka Nakanishi, Kazuya Kikuchi, Takanari Inoue, Kenzo Hirose, Masamitsu Iino, Tetsuo Nagano

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 120 KB

english, 2002

13

Parallel suspension polymerization for high-throughput resin synthesis

Thomas S Reger, Kim D Janda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 113 KB

english, 2002

14

Synthesis of iodinated 3β-aryltropanes with selective binding to either the dopamine or serotonin transporters

Huw M.L Davies, Pingda Ren, Norman X Kong, Tammy Sexton, Steven R Childers

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 110 KB

english, 2002

15

Antibacterial activity of G6-quaternary ammonium derivatives of a lipophilic vancomycin analogue

Timothy A Blizzard, Ronald M Kim, Jerry D Morgan II, Jiang Chang, Joyce Kohler, Ruth Kilburn, Kevin Chapman, Milton L Hammond

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 137 KB

english, 2002

16

Synthesis and photochemical protein crosslinking studies of hydrophilic naphthalimides

Jianxing Zhang, R.Jeremy Woods, Philip B Brown, Kap Duk Lee, Robert R Kane

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 243 KB

english, 2002

17

Tricyclic isoxazoles are novel inhibitors of the multidrug resistance protein (MRP1)

Bryan H. Norman, Joseph M. Gruber, Sean P. Hollinshead, Joseph W. Wilson, James J. Starling, Kevin L. Law, Tracy D. Self, Linda B. Tabas, Daniel C. Williams, Donald C. Paul, Margaret M. Wagner, Anne H

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 139 KB

english, 2002

18

Oxal hydroxamic acid derivatives with inhibitory activity against matrix metalloproteinases

Dirk Krumme, Harald Tschesche

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 131 KB

english, 2002

19

Probing the overlap of chorismate mutase and prephenate dehydrogenase sites in the escherichia coli T-protein: a dehydrogenase-selective inhibitor

Sarah Vincent, Shuqing Chen, David B. Wilson, Bruce Ganem

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 119 KB

english, 2002

20

Identification of a novel, orally bioavailable histamine H3 receptor antagonist based on the 4-benzyl-(1H-imidazol-4-yl) template

Robert Aslanian, Mwangi W. Mutahi, Neng-Yang Shih, Kevin D. McCormick, John J. Piwinski, Pauline C. Ting, Margaret M. Albanese, Michael Y. Berlin, Xiaohong Zhu, Shing-Chun Wong, Stuart B. Rosenblum, Y

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 150 KB

english, 2002

21

Benzimidazoles and isosteric compounds as potent and selective factor Xa inhibitors

Wei He, Barbara Hanney, Michael R Myers, Stephen Condon, Michael R Becker, Alfred P Spada, Christopher Burns, Karen Brown, Dennis Colussi, Valeria Chu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 103 KB

english, 2002

22

Diaryl-dialkyl-substituted pyrazoles: regioselective synthesis and binding affinity for the estrogen receptor

Gisele A. Nishiguchi, Alice L. Rodriguez, John A. Katzenellenbogen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 189 KB

english, 2002

23

Soluble polymer-supported synthesis of benzodiazepinones

Cheng-Yi Wu, Chung-Ming Sun

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 113 KB

english, 2002

24

Formation of thomasidioic acid from dehydrosinapinic acid dilactone under neutral conditions, and a remaining inhibitory activity against peroxynitrite-mediated protein nitration

Toshio Niwa, Umeyuki Doi, Toshihiko Osawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 112 KB

english, 2002

25

Novel N-[1-(1-substituted 4-piperidinylmethyl)-4-piperidinyl]benzamides as potent colonic prokinetic agents

Hiroshi Harada, Hiroshi Yamazaki, Yoshihito Toyotomi, Hirotaka Tateishi, Yukiko Mine, Naoyuki Yoshida, Shiro Kato

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 181 KB

english, 2002

26

Design, synthesis and bioactivity evaluation of tribactam β lactamase inhibitors

Anton Copar, Tadeja Prevec, Borut Anžič, Tomaž Mesar, Lovro Selič, Mateja Vilar, Tom Solmajer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 144 KB

english, 2002

27

Bivalent inhibition of β-Tryptase: distance scan of neighboring subunits by dibasic inhibitors

Norbert Schaschke, Andreas Dominik, Gabriele Matschiner, Christian P. Sommerhoff

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 169 KB

english, 2002

28

Benzimidazole-4,7-diones as Inhibitors of Protozoal (Toxoplasma gondii) Purine Nucleoside Phosphorylase

Frédéric Alvarez, Arnaud Ghérardi, Pascal Nebois, Marie-Elizabeth Sarciron, Anne-Françoise Pétavy, Nadia Walchshofer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 102 KB

english, 2002

29

Construction of the novel conformationally-restricted peptide library for screening of peptides that control the interaction Between nucleobases

Mizuki Takahashi, Akihiko Ueno, Hisakazu Mihara

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 279 KB

english, 2002

30

Design and synthesis of antiangiogenic/heparin-binding arginine dendrimer mimicking the surface of endostatin

Soko Kasai, Hideko Nagasawa, Mariko Shimamura, Yoshihiro Uto, Hitoshi Hori

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 139 KB

english, 2002

31

Substrate spectrum of tyrocidine thioesterase probed with randomized peptide N-acetylcysteamine thioesters

Guiyang Xie, Mahesh Uttamchandani, Grace Y.J Chen, Xianzhang Bu, San San Lin, Ka Man Wong, Weili Yan, Shao Q Yao, Zhihong Guo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 151 KB

english, 2002

32

Instructions to Contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 97 KB

english, 2002

33

Imidazo[5,1-f]triazin-4(3H)-ones, a new class of potent PDE 5 inhibitors

Helmut Haning, Ulrich Niewöhner, Thomas Schenke, Mazen Es-Sayed, Gunter Schmidt, Thomas Lampe, Erwin Bischoff

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 111 KB

english, 2002

34

Dermorphin and deltorphin heptapeptide analogues: replacement of Phe residue by Dmp greatly improves opioid receptor affinity and selectivity

Akihiro Ambo, Harumi Murase, Hideko Niizuma, Hidekazu Ouchi, Yutaka Yamamoto, Yusuke Sasaki

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 80 KB

english, 2002

35

Synthesis and evaluation of pseudopeptide analogues of a specific CXCR4 inhibitor, T140: The insertion of an (E)-alkene dipeptide isostere into the βII′-turn moiety

Hirokazu Tamamura, Kenichi Hiramatsu, Kazuhide Miyamoto, Akane Omagari, Shinya Oishi, Hideki Nakashima, Naoki Yamamoto, Yoshihiro Kuroda, Terumichi Nakagawa, Akira Otaka, Nobutaka Fujii

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 367 KB

english, 2002

36

Antibody-catalyzed cleavage of the d-Ala-d-Lac depsipeptide: An immunological approach to the problem of vancomycin resistance

Shigeki Isomura, Jon A Ashley, Peter Wirsching, Kim D Janda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 158 KB

english, 2002

37

Oxime derivatives of sordaricin as potent antifungal agents

Michael H. Serrano-Wu, Denis R. St. Laurent, Charles E. Mazzucco, Terry M. Stickle, John F. Barrett, Dolatrai M. Vyas, Balu N. Balasubramanian

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 112 KB

english, 2002

38

Binding properties of oligonucleotides containing a modified 2′-deoxyuridine with a thymine ended linker to pair with 2′-deoxyadenosine

Pascal Savy, Rachid Benhida, Jean-Louis Fourrey, Rosalie Maurisse, Jian-Sheng Sun

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 100 KB

english, 2002

39

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 254 KB

english, 2002

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