Volume 13; Issue 8

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Bioorganic & Medicinal Chemistry Letters
Volume 13; Issue 8

Bioorganic & Medicinal Chemistry Letters

Volume 13; Issue 8

1

Phenylbutyrates as potent, orally bioavailable vitronectin receptor (integrin αvβ3) antagonists

William H Miller, Peter J Manley, Russell D Cousins, Karl F Erhard, Dirk A Heerding, Chet Kwon, Stephen T Ross, James M Samanen, Dennis T Takata, Irene N Uzinskas, Catherine C.K Yuan, R.Curtis Haltiwa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 161 KB

english, 2003

2

Photo-oxidation of duplex DNA with the stable trioxatriangulenium ion

Arti Pothukuchy, Sampathkumar Ellapan, Karickal R. Gopidas, Miguel Salazar

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 184 KB

english, 2003

3

Oxyguanidines: application to non-peptidic phenyl-based thrombin inhibitors

Bruce Tomczuk, Tianbao Lu, Richard M Soll, Cynthia Fedde, Aihua Wang, Larry Murphy, Carl Crysler, Malini Dasgupta, Stephen Eisennagel, John Spurlino, Roger Bone

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 183 KB

english, 2003

4

Synthesis and estrogen receptor binding affinities of 7-hydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-ones containing a basic side chain

Young-Woo Kim, James A. Mobley, Robert W. Brueggemeier

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 159 KB

english, 2003

5

Analogues of dealanylalahopcin are inhibitors of human HIF prolyl hydroxylases

Imre Schlemminger, David R Mole, Luke A McNeill, Anupma Dhanda, Kirsty S Hewitson, Ya-Min Tian, Peter J Ratcliffe, Christopher W Pugh, Christopher J Schofield

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 154 KB

english, 2003

6

Leporin B: a novel hexokinase II gene inducing agent from an unidentified fungus

Chaowei Zhang, Liang Jin, Belinda Mondie, Scott S Mitchell, Arlindo L Castelhano, Weizhong Cai, Nils Bergenhem

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 155 KB

english, 2003

7

3-Amino-4-sulfonylpyridinone acetamide and related pyridothiadiazine thrombin inhibitors

Philip E.J. Sanderson, Kellie J. Cutrona, Kelly L. Savage, Adel M. Naylor-Olsen, Denise J. Bickel, Dennis L. Bohn, Franklin C. Clayton, Julie A. Krueger, S.Dale Lewis, Bobby J. Lucas, Elizabeth A. Lyl

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 216 KB

english, 2003

8

High-throughput synthesis and optimization of thrombin inhibitors via urazole α-addition and Michael addition

P.Douglas Boatman, Jan Urban, Minh Nguyen, Maher Qabar, Michael Kahn

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 223 KB

english, 2003

9

Design, synthesis and biological activity of β-carboline-based type-5 phosphodiesterase inhibitors

Graham N. Maw, Charlotte M.N. Allerton, Eugene Gbekor, William A. Million

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 190 KB

english, 2003

10

Design and synthesis of S-(−)-2-[[4-(napht-1-yl)piperazin-1-yl]methyl]-1,4-dioxoperhydropyrrolo[1,2-a]pyrazine (CSP-2503) using computational simulation. A 5-HT1A receptor agonist

Marı́a L López-Rodrı́guez, Ma José Morcillo, Esther Fernández, Bellinda Benhamú, Ignacio Tejada, David Ayala, Alma Viso, Mireia Olivella, Leonardo Pardo, Mercedes Delgado, Jorge Manzanares, José A Fue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 214 KB

english, 2003

11

Identification of a broad-Spectrum azasordarin with improved pharmacokinetic properties

Michael H. Serrano-Wu, Denis R.St. Laurent, Tina M. Carroll, Marco Dodier, Qi Gao, Patrice Gill, Claude Quesnelle, Anne Marinier, Charles E. Mazzucco, Alicia Regueiro-Ren, Terry M. Stickle, Dedong Wu,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 194 KB

english, 2003

12

Discovery and SAR of novel Naphthyridines as potent inhibitors of spleen tyrosine kinase (SYK)

Charles L Cywin, Bao-Ping Zhao, Daniel W McNeil, Matt Hrapchak, Anthony S Prokopowicz III, Daniel R Goldberg, Tina M Morwick, Amy Gao, Scott Jakes, Mohammed Kashem, Ronald L Magolda, Richard M Soll, M

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 168 KB

english, 2003

13

Synthesis and evaluation of a novel series of farnesyl protein transferase inhibitors as non-peptidic CAAX tetrapeptide analogues

Michel Perez, Catherine Maraval, Stephan Dumond, Marie Lamothe, Philippe Schambel, Chantal Etiévant, Bridget Hill

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 203 KB

english, 2003

14

3D-QSAR Studies on thieno[3,2-d]pyrimidines as Phosphodiesterase IV Inhibitors

Asit K Chakraborti, B Gopalakrishnan, M.Elizabeth Sobhia, Alpeshkumar Malde

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 307 KB

english, 2003

15

Contents List - 2 pages

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 222 KB

english, 2003

16

Contributors to this Issue - 2 page

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

File:

PDF, 40 KB

2003

17

Graphical Abstracts - 6 pages

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 268 KB

english, 2003

18

Instructions to Contributors and GA example

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 119 KB

english, 2003

19

Synthesis and SAR of bicyclic heteroaryl hydroxamic acid MMP and TACE inhibitors

A. Zask, Y. Gu, J.D. Albright, X. Du, M. Hogan, J.I. Levin, J.M. Chen, L.M. Killar, A. Sung, J.F. DiJoseph, M.A. Sharr, C.E. Roth, S. Skala, G. Jin, R. Cowling, K.M. Mohler, D. Barone, R. Black, C. Ma

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 203 KB

english, 2003

20

First enantiodivergent Baeyer–Villiger oxidation by recombinant whole-Cells expressing two monooxygenases from Brevibacterium

Marko D Mihovilovic, Florian Rudroff, Bernhard Müller, Peter Stanetty

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 144 KB

english, 2003

21

Novel Openers of Ca2+-Dependent Large-Conductance Potassium Channels: Symmetrical Pharmacophore and Electrophysiological Evaluation of Bisphenols

Yi Li, Graham Johnson, Jeffrey L Romine, Nicholas A Meanwell, Scott W Martin, Steven I Dworetzky, Christopher G Boissard, Valentin K Gribkoff, John E Starrett Jr

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 128 KB

english, 2003

22

Peptoid mimics of agouti related protein

Darren A. Thompson, Biao-Xin Chai, Hilary L.E. Rood, Michael A. Siani, Nicholai R. Douglas, Ira Gantz, Glenn L. Millhauser

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 211 KB

english, 2003

23

Structure-based design of inhibitors of human l-xylulose reductase modelled into the active site of the enzyme

Vincenzo Carbone, Connie Darmanin, Shuhei Ishikura, Akira Hara, Ossama El-Kabbani

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 425 KB

english, 2003

24

Design, synthesis, and structure–activity relationship of a new class of amidinophenylurea-based factor VIIa inhibitors

Otmar Klingler, Hans Matter, Manfred Schudok, S.Paul Bajaj, Joerg Czech, Martin Lorenz, Hans Peter Nestler, Herman Schreuder, Peter Wildgoose

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 229 KB

english, 2003

25

From pure FPP to mixed FPP and CAAX competitive inhibitors of farnesyl protein transferase

Marc Lannuzel, Marie Lamothe, Philippe Schambel, Chantal Etiévant, Bridget Hill, Michel Perez

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 191 KB

english, 2003

26

Peptide nucleic acid–metal complex conjugates: facile modulation of PNA–DNA duplex stability

Andriy Mokhir, Roman Stiebing, Roland Kraemer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 204 KB

english, 2003

27

Editorial board

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 54 KB

english, 2003

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