Volume 13; Issue 9

Main
Bioorganic & Medicinal Chemistry Letters
Volume 13; Issue 9

Bioorganic & Medicinal Chemistry Letters

Volume 13; Issue 9

1

A new model of the tautomycin–PP1 complex that is not analogous to the corresponding okadaic acid structure

David A. Colby, Wen Liu, James E. Sheppeck II, Hsien-Bin Huang, Angus C. Nairn, A.Richard Chamberlin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 399 KB

english, 2003

2

Controlling the intracellular localization of fluorescent polyamide analogues in cultured cells

Kathleen S Crowley, Dennis P Phillion, Scott S Woodard, Barbara A Schweitzer, Megh Singh, Hossein Shabany, Barry Burnette, Paul Hippenmeyer, Monique Heitmeier, James K Bashkin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 382 KB

english, 2003

3

Design, synthesis, and activity of novel cis- and trans-3,6-disubstituted pyran biomimetics of 3,6-disubstituted piperidine as potential ligands for the dopamine transporter

Shijun Zhang, Maarteen E.A. Reith, Aloke K. Dutta

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 176 KB

english, 2003

4

Macrocyclic inhibitors of the bacterial cell wall biosynthesis enzyme mur D

James R. Horton, Julieanne M. Bostock, Ian Chopra, Lars Hesse, Simon E.V. Phillips, David J. Adams, A.Peter Johnson, Colin W.G. Fishwick

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 164 KB

english, 2003

5

Unique spirocyclopiperazinium salt I: synthesis and structure–Activity relationship of spirocyclopiperazinium salts as analgesics

Feng-Li Gao, Xin Wang, Hong-Mei Zhang, Tie-Ming Cheng, Run-Tao Li

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 144 KB

english, 2003

6

5-Imidazolyl-quinolinones, -quinazolinones and -benzo-azepinones as farnesyltransferase inhibitors

Patrick Angibaud, Xavier Bourdrez, Ann Devine, David W End, Eddy Freyne, Yannick Ligny, Philippe Muller, Geert Mannens, Isabelle Pilatte, Virginie Poncelet, Stacy Skrzat, Gerda Smets, Jacky Van Dun, P

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 231 KB

english, 2003

7

Nonpeptide RGD antagonists: A novel class of mimetics, the 5,8-disubstituted 1-azabicyclo[5.2.0]nonan-2-one lactam

Erika Bourguet, Jean-Louis Banères, Joseph Parello, Xavier Lusinchi, Jean-Pierre Girard, Jean-Pierre Vidal

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 150 KB

english, 2003

8

Preparation and pharmacological profile of 7-(α-Azolylbenzyl)-1H-indoles and indolines as new aromatase inhibitors

Pascal Marchand, Marc Le Borgne, Martina Palzer, Guillaume Le Baut, Rolf W. Hartmann

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 150 KB

english, 2003

9

A novel metal-Chelating inhibitor of protein farnesyltransferase

Akiyuki Hamasaki, Hayato Naka, Fuyuhiko Tamanoi, Kazuo Umezawa, Masami Otsuka

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 214 KB

english, 2003

10

Discovery of potent imidazole and cyanophenyl containing farnesyltransferase inhibitors with improved oral bioavailability

Yunsong Tong, Nan-Horng Lin, Le Wang, Lisa Hasvold, Weibo Wang, Nicholas Leonard, Tongmei Li, Qun Li, Jerry Cohen, Wen-Zhen Gu, Haiying Zhang, Vincent Stoll, Joy Bauch, Kennan Marsh, Saul H. Rosenberg

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 242 KB

english, 2003

11

Synthesis and collateral dilator activity of nitroxyalkylamides having direct or latent sulfhydryl moieties

Sadao Ishihara, Fujio Saito, Yasuo Ohhata, Marie Kanai, Hiroshi Mizuno, Michio Fujisawa, Ryosuke Yorikane, Hiroyuki Koike

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 201 KB

english, 2003

12

Anti-HIV Agents. Part 55: 3′R,4′R-Di-(O)-(−)-camphanoyl-2′,2′-dimethyldihydropyrano[2,3-f]chromone (DCP), a Novel Anti-HIV agent

Donglei Yu, Arnold Brossi, Nicole Kilgore, Carl Wild, Graham Allaway, Kuo-Hsiung Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 116 KB

english, 2003

13

Effects of 8-chlorodeoxyadenosine on DNA synthesis by the klenow fragment of DNA polymerase I

Lisa S. Chen, Michael H. Bahr, Terry L. Sheppard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 190 KB

english, 2003

14

Novel selective small molecule agonists for peroxisome proliferator-activated receptor δ (PPARδ)—synthesis and biological activity

Marcos L. Sznaidman, Curt D. Haffner, Patrick R. Maloney, Adam Fivush, Esther Chao, Donna Goreham, Michael L. Sierra, Christelle LeGrumelec, H.Eric Xu, Valerie G. Montana, Millard H. Lambert, Timothy

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 237 KB

english, 2003

15

Phosphate ester serum albumin affinity tags greatly improve peptide half-life in vivo

Kerry Zobel, Michael F.T. Koehler, Maureen H. Beresini, Lisa D. Caris, Daniel Combs

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 169 KB

english, 2003

16

Editorial board

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 54 KB

english, 2003

17

Contents List

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 222 KB

english, 2003

18

Contributors to this Issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 39 KB

english, 2003

19

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 206 KB

english, 2003

20

Instructions to Contributors and GA example

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 119 KB

english, 2003

21

The selective inhibition of phosphatases by natural toxins: the anhydride domain of tautomycin is not a primary factor in controlling PP1/PP2A selectivity

Wen Liu, James E. Sheppeck II, David A. Colby, Hsien-Bin Huang, Angus C. Nairn, A.Richard Chamberlin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 191 KB

english, 2003

22

5-Aryl-pyrazolo[3,4-b]pyridines: potent inhibitors of glycogen synthase kinase-3 (GSK-3)

Jason Witherington, Vincent Bordas, Stephen L Garland, Deirdre M.B Hickey, Robert J Ife, John Liddle, Martin Saunders, David G Smith, Robert W Ward

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 171 KB

english, 2003

23

5-Aryl-pyrazolo[3,4-b]pyridazines: potent inhibitors of glycogen synthase kinase-3 (GSK-3)

Jason Witherington, Vincent Bordas, David Haigh, Deirdre M.B Hickey, Robert J Ife, Anthony D Rawlings, Brian P Slingsby, David G Smith, Robert W Ward

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 188 KB

english, 2003

24

Corrigendum to ‘Synthesis of Aminoglycoside–DNA Conjugates’ [Bioorg. Med. Chem. Lett. 12 (2002) 1259]

I. Charles, Liang Xue, Dev P. Arya

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 58 KB

english, 2003

25

Chain-Branched acyclic phenethylthiocarbamates as vanilloid receptor antagonists

JungWha Yoon, HyeYoung Choi, Hyun Joo Lee, Chong Hyun Ryu, Hyeung-geun Park, Young-ger Suh, Uhtaek Oh, Yeon Su Jeong, Jin Kyu Choi, Young-Ho Park, Hee-Doo Kim

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 163 KB

english, 2003

26

Structure–Activity relationships of novel anti-malarial agents. Part 6: N-(4-Arylpropionylamino-3-benzoylphenyl)-[5-(4-nitrophenyl)-2-furyl]acrylic acid amides

Jochen Wiesner, Katharina Fucik, Katja Kettler, Jacek Sakowski, Regina Ortmann, Hassan Jomaa, Martin Schlitzer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 154 KB

english, 2003

27

New scaffolds in the development of Mu opioid-receptor ligands

Daniel Pagé, Natalie Nguyen, Sylvain Bernard, Martin Coupal, Mylène Gosselin, Julie Lepage, Lynda Adam, William Brown

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 198 KB

english, 2003

28

Efficient synthesis of 3-trifluoromethylphenyldiazirinyl oleic acid derivatives and Their biological activity for protein kinase C

Makoto Hashimoto, Kensuke Nabeta, Kentaro Murakami

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 125 KB

english, 2003

29

Synthesis, in vitro, and in vivo evaluation of phosphate ester derivatives of combretastatin A-4

Mallinath B. Hadimani, Jianyi Hua, M.Devan Jonklaas, Raymond J. Kessler, Yezhou Sheng, Adrian Olivares, Rajendra P. Tanpure, Aimee Weiser, Jianxing Zhang, Klaus Edvardsen, Robert R. Kane, Kevin G. Pin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 188 KB

english, 2003

To build up a library is to create a life. It’s never just a random collection of books.

— Carlos María Domínguez

Official channel

Z-Library Desktop Launcher

Tor version

Z-Library

Z-Library Since 2009 support@z-lib.do

EnglishРусскийEspañolItalianoελληνικάاللغة العربيةBahasa IndonesiaBahasa Malaysiaहिन्दीDeutschFrançaisPortuguêsУкраїнськаPolski中文繁體中文日本語Tiếng ViệtAzərbaycan DiliՀայոց լեզուภาษาไทยTürk Diliქართველიবাংলাپښتوతెలుగుاردو한국어SrpskiБългарски