Volume 25; Issue 18

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Bioorganic & Medicinal Chemistry Letters
Volume 25; Issue 18

Bioorganic & Medicinal Chemistry Letters

Volume 25; Issue 18

1

Chemical constituents of Miliusa balansae leaves and inhibition of nitric oxide production in lipopolysaccharide-induced RAW 264.7 cells

Thao, Nguyen Phuong, Luyen, Bui Thi Thuy, Tai, Bui Huu, Cuong, Nguyen Manh, Kim, Youn Chul, Minh, Chau Van, Kim, Young Ho

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 660 KB

english, 2015

2

N-Aryl benzenesulfonamide inhibitors of [3H]-thymidine incorporation and β-catenin signaling in human hepatocyte-derived Huh-7 carcinoma cells

Kril, Liliia M., Vilchez, Valery, Jiang, Jieyun, Turcios, Lilia, Chen, Changguo, Sviripa, Vitaliy M., Zhang, Wen, Liu, Chunming, Spear, Brett, Watt, David S., Gedaly, Roberto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 277 KB

english, 2015

3

Synthesis and validation of novel cholesterol-based fluorescent lipids designed to observe the cellular trafficking of cationic liposomes

Kim, Bieong-Kil, Seu, Young-Bae, Choi, Jong-Soo, Park, Jong-Won, Doh, Kyung-Oh

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 1.11 MB

english, 2015

4

Total synthesis of cordatanine, structural reassignment of drymaritin, and anti-inflammatory activity of synthetic precursors

Fang, Hsin Wei, Liao, Yu-Ren, Hwang, Tsong-Long, Shieh, Po-Chuen, Lee, Kuo-Hsiung, Hung, Hsin-Yi, Wu, Tian-Shung

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 359 KB

english, 2015

5

Biarylmethoxy 2-nitroimidazooxazine antituberculosis agents: Effects of proximal ring substitution and linker reversal on metabolism and efficacy

Thompson, Andrew M., Blaser, Adrian, Palmer, Brian D., Franzblau, Scott G., Wan, Baojie, Wang, Yuehong, Ma, Zhenkun, Denny, William A.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 703 KB

english, 2015

6

Structure-based de novo design and synthesis of aminothiazole-based p38 MAP kinase inhibitors

Park, Hwangseo, Lee, Soyoung, Hong, Sungwoo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 760 KB

english, 2015

7

Synthesis and in vitro evaluation of [18F]FECIMBI-36: A potential agonist PET ligand for 5-HT2A/2C receptors

Prabhakaran, Jaya, Underwood, Mark D., Kumar, J.S. Dileep, Simpson, Norman R., Kassir, Suham A., Bakalian, Mihran J., Mann, J. John, Arango, Victoria

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 588 KB

english, 2015

8

Identification of dialkyl diacetylene diols with potent cancer chemopreventive activity

Lee, Chang-Yong, Yun, Ji Ho, Kang, Kyungsu, Nho, Chu-Won, Shin, Dongyun

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 570 KB

english, 2015

9

Synthesis and characterization of oligodeoxyribonucleotides modified with 2′-thio-2′-deoxy-2′-S-(pyren-1-yl)methyluridine

Anderson, Brooke A., Hrdlicka, Patrick J.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 752 KB

english, 2015

10

Hydrogen deuterium mass spectrometry in drug discovery

Campobasso, Nino, Huddler, Donald

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 1.94 MB

english, 2015

11

Discovery of indolizines containing triazine moiety as new leads for the development of antitumoral agents targeting mitotic events

Lucescu, Liliana, Ghinet, Alina, Belei, Dalila, Rigo, Benoît, Dubois, Joëlle, Bîcu, Elena

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 885 KB

english, 2015

12

Re-exploring the N-phenylpicolinamide derivatives to develop mGlu4 ligands with improved affinity and in vitro microsomal stability

Zhang, Zhaoda, Kil, Kun-Eek, Poutiainen, Pekka, Choi, Ji-Kyung, Kang, Hye-Jin, Huang, Xi-Ping, Roth, Bryan L., Brownell, Anna-Liisa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 1.60 MB

english, 2015

13

Dietziamides, novel tetramic acid dimers from Dietzia timorensis MZ-3 with antioxidative activity

Hoshino, Shotaro, Wakimoto, Toshiyuki, Zhang, Huiping, Hayashi, Fumiaki, Okada, Masahiro, Abe, Ikuro

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 459 KB

english, 2015

14

Strongylophorines, new protein tyrosine phosphatase 1B inhibitors, from the marine sponge Strongylophora strongilata collected at Iriomote Island

Lee, Jong-Soo, Abdjul, Delfly B., Yamazaki, Hiroyuki, Takahashi, Ohgi, Kirikoshi, Ryota, Ukai, Kazuyo, Namikoshi, Michio

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 433 KB

english, 2015

15

The effect of complexation of 3-formylrifamycin SV macrocyclic ether derivatives with metal cations and small nitrogen-containing organic molecules on antibacterial activity against S. aureus and S. epidermidis

Przybylski, Piotr, Pyta, Krystian, Czerwonka, Dominika, Kubicka, Marcelina M., Gajecka, Marzena

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 2.16 MB

english, 2015

16

Synthesis and biological evaluation of levofloxacin core-based derivatives with potent antibacterial activity against resistant Gram-positive pathogens

Huang, Xiaoguang, Bao, Yingxia, Zhu, Shaoxuan, Zhang, Xiaona, Lan, Shilong, Wang, Ting

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 418 KB

english, 2015

17

Synthesis and inhibitory activity of substrate-analog fructosyl peptide oxidase inhibitors

Watanabe, Bunta, Ichiyanagi, Atsushi, Hirokawa, Kozo, Gomi, Keiko, Nakatsu, Toru, Kato, Hiroaki, Kajiyama, Naoki

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 739 KB

english, 2015

18

Indolylpiperidine derivatives as potent and selective α1B adrenoceptor antagonists

Hayashi, Ryoji, Ohmori, Eiji, Moriwaki, Mitsuhiro, Kumagai, Hiroki, Isogaya, Masafumi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 505 KB

english, 2015

19

Discovery and structure-guided optimization of tert-butyl 6-(phenoxymethyl)-3-(trifluoromethyl)benzoates as liver X receptor agonists

Matsui, Yumi, Yamaguchi, Takahiro, Yamazaki, Takanori, Yoshida, Masayuki, Arai, Masami, Terasaka, Naoki, Honzumi, Shoko, Wakabayashi, Kenji, Hayashi, Shinko, Nakai, Daisuke, Hanzawa, Hiroyuki, Tamaki,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 1.86 MB

english, 2015

20

Cytotoxic triterpenoid glycosides (saikosaponins) from the roots of Bupleurum chinense

Li, Dan-Qi, Wu, Jie, Liu, Li-Yin, Wu, Ying-Ying, Li, Ling-Zhi, Huang, Xiao-Xiao, Liu, Qing-Bo, Yang, Jing-Yu, Song, Shao-Jiang, Wu, Chun-Fu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 531 KB

english, 2015

21

Efficient synthesis of the intermediate of abacavir and carbovir using a novel (+)-γ-lactamase as a catalyst

Gao, Shuaihua, Zhu, Shaozhou, Huang, Rong, Lu, Yingxiu, Zheng, Guojun

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 855 KB

english, 2015

22

New phenolic compounds from the seeds of Nigella glandulifera and their inhibitory activities against human cancer cells

Sun, Lu, Liu, Yu-Ming, Chen, Bao-Quan, Liu, Qing-Hua

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 395 KB

english, 2015

23

Synthesis of [11C]CX-6258 as a new PET tracer for imaging of Pim kinases in cancer

Wang, Min, Tzintzun, Reynaldo, Gao, Mingzhang, Xu, Zhidong, Zheng, Qi-Huang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 501 KB

english, 2015

24

Design, synthesis, and in vivo activity of novel inhibitors of delta-5 desaturase for the treatment of metabolic syndrome

Baugh, Simon D.P., Pabba, Praveen K., Barbosa, Joseph, Coulter, Eric, Desai, Urvi, Gay, Jason P., Gopinathan, Suma, Han, Qiang, Hari, Rajee, Kimball, S. David, Nguyen, Huy V., Ni, Chi-You, Powell, Dav

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 820 KB

english, 2015

25

Antiviral activity and interaction mechanisms study of novel glucopyranoside derivatives

Chen, Meihang, Hu, Deyu, Li, Xiangyang, Yang, Song, Zhang, Weiying, Li, Pei, Song, Baoan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 1.34 MB

english, 2015

26

Eight new cycloartane triterpenoids from Beesia calthifolia with hepatoprotective effects against d-galactosamine induced L02 cell damage

Gan, Li-She, Zheng, Dan-Jun, Liu, Qian, Zhou, Jing, Zhang, Min-Zhe, Yao, Wei, Shao, Bai-Hao, Mo, Jian-Xia, Zhou, Chang-Xin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 505 KB

english, 2015

27

Isolation and structure elucidation of bioactive compounds from the roots of the Tunisian Ononis angustissima L.

Ghribi, Lotfi, Waffo-Téguo, Pierre, Cluzet, Stéphanie, Marchal, Axel, Marques, Jessica, Mérillon, Jean-Michel, Ben Jannet, Hichem

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 648 KB

english, 2015

28

Novel antibacterial active quinolone–fluoroquinolone conjugates and 2D-QSAR studies

Panda, Siva S., Liaqat, Sumaira, Girgis, Adel S., Samir, Ahmed, Hall, C. Dennis, Katritzky, Alan R.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 712 KB

english, 2015

29

Mechanism studies on anti-HepG2 cell proliferation of phenanthroline derivatives as G-quadruplex DNA stabilizers

Li, Huiqing, Wei, Chunying

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 1.52 MB

english, 2015

30

Corrigendum to “Novel monobactams utilizing a siderophore uptake mechanism for the treatment of Gram-negative infections” [Bioorg. Med. Chem. Lett. 22/18 (2012) 5989–5994]

Mitton-Fry, Mark J., Arcari, Joel T., Brown, Matthew F., Casavant, Jeffrey M., Finegan, Steven M., Flanagan, Mark E., Gao, Hongying, George, David M., Gerstenberger, Brian S., Han, Seungil, Hardink, J

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 246 KB

english, 2015

31

Corrigendum to “Design, synthesis and RNase A inhibition activity of catechin and epicatechin and nucleobase chimeric molecules” [Bioorg. Med. Chem. Lett. 18 (2008) 5411–5414]

Roy, Basab, Dutta, Sansa, Choudhary, Anupma, Basak, Amit, Dasgupta, Swagata

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

File:

PDF, 174 KB

2015

32

Editorial board

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 30 KB

english, 2015

33

Graphical contents list

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 4.37 MB

english, 2015

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