Volume 26; Issue 3

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Bioorganic & Medicinal Chemistry Letters
Volume 26; Issue 3

Bioorganic & Medicinal Chemistry Letters

Volume 26; Issue 3

1

The influence of 5-HT2A activity on a 5-HT2C specific in vivo assay used for early identification of multiple acting SERT and 5-HT2C receptor ligands

Éliás, Olivér, Nógrádi, Katalin, Domány, György, Szakács, Zoltán, Kóti, János, Szántay, Csaba, Tarcsay, Ákos, Keserű, György M., Gere, Anikó, Kiss, Béla, Kurkó, Dalma, Kolok, Sándor, Némethy, Zsolt, K

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 722 KB

english, 2016

2

Molecular insights to the bioactive form of BV02, a reference inhibitor of 14-3-3σ protein–protein interactions

Valensin, Daniela, Cau, Ylenia, Calandro, Pierpaolo, Vignaroli, Giulia, Dello Iacono, Lucia, Chiariello, Mario, Mori, Mattia, Botta, Maurizio

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 795 KB

english, 2016

3

Sequence selective naked-eye detection of DNA harnessing extension of oligonucleotide-modified nucleotides

Verga, Daniela, Welter, Moritz, Marx, Andreas

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 701 KB

english, 2016

4

Mitochondrial drug targets in neurodegenerative diseases

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 495 KB

english, 2016

5

Bioactive lignan derivatives from the stems of Firmiana simplex

Woo, Kyeong Wan, Suh, Won Se, Subedi, Lalita, Kim, Sun Yeou, Kim, Aejung, Lee, Kang Ro

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 470 KB

english, 2016

6

Identification of allosteric ERK2 inhibitors through in silico biased screening and competitive binding assay

Kinoshita, Takayoshi, Sugiyama, Hajime, Mori, Yurika, Takahashi, Naruhide, Tomonaga, Atsushi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 876 KB

english, 2016

7

Synthesis and biological evaluation of quinoxaline di-N-oxide derivatives with in vitro trypanocidal activity

Pérez-Silanes, Silvia, Torres, Enrique, Arbillaga, Leire, Varela, Javier, Cerecetto, Hugo, González, Mercedes, Azqueta, Amaya, Moreno-Viguri, Elsa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 1.35 MB

english, 2016

8

Lead optimization of the VU0486321 series of mGlu1 PAMs. Part 2: SAR of alternative 3-methyl heterocycles and progress towards an in vivo tool

Garcia-Barrantes, Pedro M., Cho, Hyekyung P., Metts, Adam M., Blobaum, Anna L., Niswender, Colleen M., Conn, P. Jeffrey, Lindsley, Craig W.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 3.20 MB

english, 2016

9

Novel hydroxyamides and amides containing d-glucopyranose or d-fructose units: Biological assays in MCF-7 and MDST8 cell lines

Carreiro, Elisabete P., Costa, Ana R., Cordeiro, Maria M., Martins, Rute, Pires, Tiago O., Saraiva, Mafalda, Antunes, Célia M., Burke, Anthony J.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 1.08 MB

english, 2016

10

Salicylates are interference compounds in TR-FRET assays

Hanley, Ronan P., Horvath, Shanti, An, Jianghong, Hof, Fraser, Wulff, Jeremy E.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 1.41 MB

english, 2016

11

2-Amino-4-bis(aryloxybenzyl)aminobutanoic acids: A novel scaffold for inhibition of ASCT2-mediated glutamine transport

Schulte, Michael L., Khodadadi, Alexandra B., Cuthbertson, Madison L., Smith, Jarrod A., Manning, H. Charles

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 873 KB

english, 2016

12

Alkenes with antioxidative activities from Murraya koenigii (L.) Spreng

Ma, Qin-Ge, Xu, Kun, Sang, Zhi-Pei, Wei, Rong-Rui, Liu, Wen-Min, Su, Ya-Lun, Yang, Jian-Bo, Wang, Ai-Guo, Ji, Teng-Fei, Li, Lu-Jun

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 405 KB

english, 2016

13

Gene silencing by 2′-O-methyldithiomethyl-modified siRNA, a prodrug-type siRNA responsive to reducing environment

Ochi, Yosuke, Imai, Mieko, Nakagawa, Osamu, Hayashi, Junsuke, Wada, Shun-ichi, Urata, Hidehito

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 1.00 MB

english, 2016

14

Synthesis of a norcantharidin-tethered guanosine: Protein phosphatase-1 inhibitors that change alternative splicing

Kwiatkowski, Stefan, Sviripa, Vitaliy M., Zhang, Zhaiyi, Wendlandt, Alison E., Höbartner, Claudia, Watt, David S., Stamm, Stefan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 621 KB

english, 2016

15

A stepwise dechlorination/cross-coupling strategy to diversify the vancomycin ‘in-chloride’

Wadzinski, Tyler J., Gea, Katherine D., Miller, Scott J.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 1018 KB

english, 2016

16

Gambogic acid induces apoptotic cell death in T98G glioma cells

Thida, Mya, Kim, Dae Won, Tran, Thi Thu Thuy, Pham, Minh Quan, Lee, Heesu, Kim, Inki, Lee, Jae Wook

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 1.08 MB

english, 2016

17

Discovery of highly potent dual EP2 and EP3 agonists with subtype selectivity

Kinoshita, Akihiro, Higashino, Masato, Aratani, Yoshiyuki, Kakuuchi, Akito, Matsuya, Hidekazu, Ohmoto, Kazuyuki

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 752 KB

english, 2016

18

Editorial board

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 30 KB

english, 2016

19

Design, radiosynthesis, and evaluation of radiotracers for positron emission tomography imaging of stearoyl-CoA desaturase-1

Silvers, William C., Cai, Hancheng, Öz, Orhan K., Sun, Xiankai

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 538 KB

english, 2016

20

Multimodal formyl peptide receptor 1 targeted inflammation imaging probe: cFLFLF-MHI-DOTA

Li, Jie, Zhang, Yi, Chordia, Mahendra D., Wu, Hua, Shao, Li, Pan, Dongfeng

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 678 KB

english, 2016

21

Growth inhibitory effect of d-arabinose against the nematode Caenorhabditis elegans: Discovery of a novel bioactive monosaccharide

Sakoguchi, Hirofumi, Yoshihara, Akihide, Shintani, Tomoya, Okuma, Kazuhiro, Izumori, Ken, Sato, Masashi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 804 KB

english, 2016

22

Synthesis and positive inotropic activity evaluation of liguzinediol metabolites

Zhu, Hao-hao, Chen, Yu-qing, Cheng, Dong, Li, Wei, Wang, Tian-lin, Wen, Hong-mei, Chen, Long, Liu, Jian

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 568 KB

english, 2016

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