books search
books
articles search
articles
Donate
Log In
Log In
to access more features
personal recommendations
Telegram Bot
download history
send to Email or Kindle
manage booklists
save to favorites
Explore
Journals
Contribution
Donate
Litera Library
Donate paper books
Add paper books
Open LITERA Point
Volume 30; Issue 11
Main
Bioorganic & Medicinal Chemistry Letters
Volume 30; Issue 11
Bioorganic & Medicinal Chemistry Letters
Volume 30; Issue 11
1
Design, synthesis and anti-influenza A virus activity of novel 2,4-disubstituted quinazoline derivatives
Wang, Minghua
,
Zhang, Guoning
,
Wang, Yujia
,
Wang, Juxian
,
Zhu, Mei
,
Cen, Shan
,
Wang, Yucheng
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 809 KB
Your tags:
2020
2
Design, synthesis and biological evaluation of novel hybrids of N-aryl pyrrothine-base α-pyrone as bacterial RNA polymerase inhibitors
Tan, Xiangduan
,
Huang, Mohan
,
Nian, Siyun
,
Peng, Yanfen
,
Qin, Jianli
,
Kong, Bo
,
Duan, Xiaoqun
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 2.87 MB
Your tags:
2020
3
S1P1-selective agonist prodrug IMMH002 is phosphorylated in rats to form an S-configured enantiomer: Synthesis, verification, and biological activity of the in vivo active metabolite
Xiao, Qiong
,
Hu, Minwan
,
Chen, Si
,
Jin, Jing
,
Li, Li
,
Hu, Jinping
,
Xie, Ping
,
Yin, Dali
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 1.90 MB
Your tags:
2020
4
Chalcones bearing a 3,4,5-trimethoxyphenyl motif are capable of selectively inhibiting oncogenic K-Ras signaling
Kovar, Sarah E.
,
Fourman, Cody
,
Kinstedt, Christine
,
Williams, Brandon
,
Morris, Christopher
,
Cho, Kwang-jin
,
Ketcha, Daniel M.
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 3.35 MB
Your tags:
2020
5
Two new secondary metabolites, saccharochlorines A and B, from a marine bacterium Saccharomonospora sp. KCTC-19160
Le, Tu Cam
,
Katila, Nikita
,
Park, Songhee
,
Lee, Jihye
,
Yang, Inho
,
Choi, Hyukjae
,
Choi, Dong-Young
,
Nam, Sang-Jip
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 910 KB
Your tags:
2020
6
Dithiocarbamate prodrugs activated by prostate specific antigen to target prostate cancer
Bakthavatsalam, Subha
,
Wiangnak, Petpailin
,
George, Daniel J.
,
Zhang, Tian
,
Franz, Katherine J.
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 750 KB
Your tags:
2020
7
Ultrasounds-mediated 10-seconds synthesis of chalcones as potential farnesyltransferase inhibitors
Homerin, Germain
,
Nica, Adrian Sorin
,
Farce, Amaury
,
Dubois, Joëlle
,
Ghinet, Alina
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 5.33 MB
Your tags:
2020
8
Finding the mechanism of esterase D activation by a small molecule
Chen, Xinpeng
,
Yang, Yuejun
,
Su, Le
,
Cui, Xiaoling
,
Shao, Jing
,
Liu, Shuyan
,
Zhao, Baoxiang
,
Miao, Junying
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 5.76 MB
Your tags:
2020
9
Synthesis of novel tryptanthrin derivatives as dual inhibitors of indoleamine 2,3-dioxygenase 1 and tryptophan 2,3-dioxygenase
Li, Yuanyuan
,
Zhang, Shengnan
,
Wang, Rong
,
Cui, Menghan
,
Liu, Wei
,
Yang, Qing
,
Kuang, Chunxiang
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 670 KB
Your tags:
2020
10
Design, synthesis and biological evaluation of spiropyrazolopyridone derivatives as potent dengue virus inhibitors
Xu, Jimin
,
Xie, Xuping
,
Chen, Haiying
,
Zou, Jing
,
Xue, Yu
,
Ye, Na
,
Shi, Pei-Yong
,
Zhou, Jia
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 620 KB
Your tags:
2020
11
Direct modifications of the cyclic peptide Polymyxin B leading to analogues with enhanced in vitro antibacterial activity
Brown, Pamela
,
Abdulle, Omar
,
Boakes, Steven
,
Duperchy, Esther
,
Moss, Stephen
,
Simonovic, Mona
,
Stanway, Steven
,
Wilson, Antoinette
,
Dawson, Michael J.
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 554 KB
Your tags:
2020
12
Ansamycin derivatives from the marine-derived Streptomyces sp. SCSGAA 0027 and their cytotoxic and antiviral activities
Nong, Xu-Hua
,
Tu, Zheng-Chao
,
Qi, Shu-Hua
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 1.27 MB
Your tags:
2020
13
Synthesis and biological evaluation of heterocyclic bis-aryl amides as novel Src homology 2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors
Satheeshkumar, Rajendran
,
Zhu, Rui
,
Feng, Bo
,
Huang, Chao
,
Gao, Ya
,
Gao, Li-Xin
,
Shen, Chao
,
Hou, Ting-Jun
,
Xu, Lei
,
Li, Jia
,
Zhu, Yun-Long
,
Zhou, Yu-Bo
,
Wang, Wen-Long
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 1.74 MB
Your tags:
2020
14
Substituted sulfonamide bioisosteres of 8-hydroxyquinoline as zinc-dependent antibacterial compounds
McGowan, John E.
,
Harper, Andrew D.
,
Davison, Emma K.
,
Jeong, Joo Young
,
Mros, Sonya
,
Harbison-Price, Nichaela
,
Van Zuylen, Essie M.
,
Knottenbelt, Melanie K.
,
Heikal, Adam
,
Ferguson, Scott A.
,
McConne
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 808 KB
Your tags:
2020
15
Hypolipidemic constituents from the aerial portion of Sibiraea angustata
Liu, Hongdong
,
Zhang, Ting
,
Jiang, Piao
,
Zhu, Weifeng
,
Yu, Songhua
,
Liu, Yong
,
Li, Bin
,
Li, Fei
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 1.27 MB
Your tags:
2020
16
Screening of chalcone analogs with anti-depressant, anti-inflammatory, analgesic, and COX-2-inhibiting effects
Huang, Zhe-Hao
,
Yin, Li-Quan
,
Guan, Li-Ping
,
Li, Zhao-Hui
,
Tan, Cheng
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 1.60 MB
Your tags:
2020
17
Influence of side-chain changes on histone deacetylase inhibitory and cytotoxicity activities of curcuminoid derivatives
Somsakeesit, La-or
,
Senawong, Thanaset
,
Kumboonma, Pakit
,
Saenglee, Somprasong
,
Samankul, Arunta
,
Senawong, Gulsiri
,
Yenjai, Chavi
,
Phaosiri, Chanokbhorn
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 2.61 MB
Your tags:
2020
18
A hypoxia-activated antibacterial prodrug
Yeoh, Yuan Qi
,
Horsley, John R.
,
Polyak, Steven W.
,
Abell, Andrew D.
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 421 KB
Your tags:
2020
19
New 8-amino-1,2,4-triazolo[4,3-a]pyrazin-3-one derivatives. Evaluation of different moieties on the 6-aryl ring to obtain potent and selective human A2A adenosine receptor antagonists
Falsini, Matteo
,
Ceni, Costanza
,
Catarzi, Daniela
,
Varano, Flavia
,
Dal Ben, Diego
,
Marucci, Gabriella
,
Buccioni, Michela
,
Martà Navia, Aleix
,
Volpini, Rosaria
,
Colotta, Vittoria
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 2.90 MB
Your tags:
2020
20
Alanine scan-guided synthesis and biological evaluation of analogues of culicinin D, a potent anticancer peptaibol
Kavianinia, Iman
,
Stubbing, Louise A.
,
Abbattista, Maria R.
,
Harris, Paul W.R.
,
Smaill, Jeff B.
,
Patterson, Adam V.
,
Brimble, Margaret A.
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 899 KB
Your tags:
2020
21
In silico and in vitro studies on interaction of novel non-imidazole histamine H3R antagonists with CYP3A4
Podlewska, Sabina
,
Latacz, Gniewomir
,
Åażewska, Dorota
,
KieÄ-Kononowicz, Katarzyna
,
Handzlik, Jadwiga
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 5.14 MB
Your tags:
2020
22
Synthesis and evaluation of Al18F-NODA complex conjugated 2-(4-aminophenyl)benzothiazole as a potential tumor imaging agent
Wang, Liang
,
Niu, Mengda
,
He, Yujia
,
Tian, Chuanhuizi
,
Peng, Zhiping
,
Jia, Jianhua
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 5.70 MB
Your tags:
2020
23
An osteoinductive effect of phytol on mouse mesenchymal stem cells (C3H10T1/2) towards osteoblasts
Sanjeev, Ganesh
,
Sidharthan, D. Saleth
,
Pranavkrishna, S.
,
Pranavadithya, S.
,
Abhinandan, R.
,
Akshaya, R.L.
,
Balagangadharan, K.
,
Siddabathuni, Nishitha
,
Srinivasan, Swathi
,
Selvamurugan, N.
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 2.38 MB
Your tags:
2020
24
Identification of a new class of non-electrophilic TRPA1 agonists by a structure-based virtual screening approach
Araki, Mitsugu
,
Kanda, Naoto
,
Iwata, Hiroaki
,
Sagae, Yukari
,
Masuda, Katsuyoshi
,
Okuno, Yasushi
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 4.14 MB
Your tags:
2020
25
Inhibitory effects of biseokeaniamide A against lipopolysaccharide-induced signal transduction
Ohno, Osamu
,
Terasaki, Takuro
,
Sano, Takuya
,
Hitomi, Yuki
,
Miyamoto, Junichiro
,
Matsuno, Kenji
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 1.11 MB
Your tags:
2020
26
The EZMTT cell proliferation assay provides precise measurement for drug combinations and better correlation between in vitro and in vivo efficacy
Rui, Jingjing
,
Xu, Ning
,
Yin, JianBing
,
Yu, Yan
,
Bai, Ruisong
,
Su, Weike
,
Ruan, Benfang
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 3.37 MB
Your tags:
2020
27
Graphical abstract TOC
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 367 KB
Your tags:
2020
28
Editorial Board
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 37 KB
Your tags:
2020
29
Graphical Abstract Contents Continued
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 1.27 MB
Your tags:
2020
30
Graphical abstract TOC
Journal:
Bioorganic & Medicinal Chemistry Letters
Year:
2020
File:
PDF, 234 KB
Your tags:
2020
1
Follow
this link
or find "@BotFather" bot on Telegram
2
Send /newbot command
3
Specify a name for your chatbot
4
Choose a username for the bot
5
Copy an entire last message from BotFather and paste it here
×
×