Volume 30; Issue 16

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Bioorganic & Medicinal Chemistry Letters
Volume 30; Issue 16

Bioorganic & Medicinal Chemistry Letters

Volume 30; Issue 16

1

N-[18F]-Fluoroacetylcrizotinib: A potentially potent and selective PET tracer for molecular imaging of non-small cell lung cancer

Buck, Jason R., Saleh, Samir, Claus, Trey, Lovly, Christine, Hight, Matthew R., Nickels, Michael L., Noor Tantawy, M., Charles Manning, H.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.52 MB

2020

2

Synthesis and biological evaluation of a novel photo-activated histone deacetylase inhibitor

Sama, Gopal R., Liu, Hongbin, Mountford, Simon, Thompson, Phillip, Robinson, Andrea, Dear, Anthony E.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 813 KB

2020

3

Potent dual EGFR/Her4 tyrosine kinase inhibitors containing novel (1,2-dithiolan-4-yl)acetamides

Mansour, Tarek S., Pallepati, Ranga R., Basetti, Vishnu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 623 KB

2020

4

N-(4-(2-chloro-4-(trifluoromethyl)phenoxy)phenyl)picolinamide as a new inhibitor of mitochondrial complex III: Synthesis, biological evaluation and computational simulations

Cheng, Hua, Yang, Lu, Liu, Hong-Fu, Zhang, Rui, Chen, Cheng, Wu, Yuan, Jiang, Wen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 2.80 MB

2020

5

Synthesis and dopamine receptor pharmacological evaluations on ring C ortho halogenated 1-phenylbenzazepines

Giri, Rajan, Namballa, Hari K., Sarker, Ananta, Alberts, Ian, Harding, Wayne W.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 2.15 MB

2020

6

Design, synthesis and biological evaluation of novel pteridinone derivatives possessing a hydrazone moiety as potent PLK1 inhibitors

Li, Zhiwei, Xu, Le, Zhu, Liangyu, Zhao, Yanfang, Hu, Tao, Yin, Bixi, Liu, Yajing, Hou, Yunlei

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 6.68 MB

2020

7

Decaturenol A and known oxalicine related meroterpenoids isolated from Penicillium decaturense RO050, and their new biological activities

Ishiuchi, Kan'ichiro, Amber Syed, Ayesha, Kosuge, Yasuhiro, Fujiwara, Yukio, Makino, Toshiaki, Hirose, Dai

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 544 KB

2020

8

Exploring the newer oxadiazoles as real inhibitors of human SIRT2 in hepatocellular cancer cells

Dukanya,, Shanmugam, Muthu K., Rangappa, Shobith, Metri, Prashant K., Mohan, Surender, Basappa,, Rangappa, Kanchugarakoppal S.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.28 MB

2020

9

SAR of non-hydrolysable analogs of pyridoxal 5â²-phosphate against low molecular weight protein tyrosine phosphatase isoforms

DeSouza, Shirin R., Olson, Maxwell C., Tinucci, Samantha L., Sinner, Erica K., Flynn, Rebecca S., Marshall, Quinlen F., Jakubowski, Henry V., McIntee, Edward J.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.52 MB

2020

10

Novel anticancer drug curaxin CBL0137 impairs DNA methylation by eukaryotic DNA methyltransferase Dnmt3a

Sergeev, Alexander, Vorobyov, Andrey, Yakubovskaya, Marianna, Kirsanova, Olga, Gromova, Elizaveta

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 716 KB

2020

11

Structure-activity relationship study of cytotoxic neolignan derivatives using multivariate analysis and computation-aided drug design

de Sousa, Fernanda S., Baldim, JoÃ£o L., Azevedo, Ricardo A., Figueiredo, Carlos R., Pieper, Pauline, Sear, Claire E., Anderson, Edward A., Lago, JoÃ£o Henrique G.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.12 MB

2020

12

Discovery of ASP5286: A novel non-immunosuppressive cyclophilin inhibitor for the treatment of HCV

Makino, Takuya, Yoshimura, Seiji, Neya, Masahiro, Yamanaka, Toshio, Sawada, Masae, Tsujii, Eisaku, Barrett, David

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 891 KB

2020

13

Development of a new class of liver receptor homolog-1 (LRH-1) agonists by photoredox conjugate addition

Cornelison, Jeffery L., Cato, Michael L., Johnson, Alyssa M., D'Agostino, Emma H., Melchers, Diana, Patel, Anamika B., Mays, Suzanne G., Houtman, RenÃ©, Ortlund, Eric A., Jui, Nathan T.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 3.48 MB

2020

14

Single-crystal structure and intracellular localization of Zn(II)-thiosemicarbazone complex targeting mitochondrial apoptosis pathways

Qi, Jinxu, Zhao, Wei, Zheng, Yunyun, Wang, Ruiya, Chen, Qiu, Wang, Fu-An, Fan, Weiwei, Gao, Huashan, Xia, Xichao

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 4.33 MB

2020

15

A chalcone derivative binds a putative allosteric site of YopH: Inhibition of a virulence factor of Yersinia

de Souza, Ana C.A., Mori, Mattia, Sens, Larissa, Rocha, Ruth F., Tizziani, Tiago, de Souza, Luiz F.S., Domeneghini Chiaradia-Delatorre, Louise, Botta, Maurizio, Nunes, Ricardo J., Terenzi, HernÃ¡n, Me

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.21 MB

2020

16

Non-food bioactive products for insecticides (II): Investigation on stress responses of Tetranychus cinnabarinus Boisduval against a derivative of the alkaloid matrine

Lv, Min, Sun, Zhiqiang, Li, Shaochen, Zhang, Shaoyong, Xu, Hui

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.51 MB

2020

17

Direct monitoring of live human pluripotent stem cells by a highly selective pluripotency sensor

Park, Myung Rae, Nam, Donggyu, Lee, Hyunah, Chang, Young-Tae, Zaehres, Holm, Kim, Jeong Beom

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 10.40 MB

2020

18

Improving NK1R-targeted gene delivery of stearyl-antimicrobial peptide CAMEL by conjugating it with substance P

Song, Jingjing, Huang, Sujie, Ma, Panpan, Zhang, Bao, Jia, Bo, Zhang, Wei

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.44 MB

2020

19

Structural basis for the stabilization of amyloidogenic immunoglobulin light chains by hydantoins

Yan, Nicholas L., Santos-Martins, Diogo, Rennella, Enrico, Sanchez, Brittany B., Chen, Jason S., Kay, Lewis E., Wilson, Ian A., Morgan, Gareth J., Forli, Stefano, Kelly, Jeffery W.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 3.89 MB

2020

20

Editorial Board

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 35 KB

2020

21

Graphical abstract TOC

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 357 KB

2020

22

Graphical Abstract Contents Continued

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 247 KB

2020

23

Signaling pathways associated with macrophage-activating polysaccharide isolated from the fermentation liquor of Rhizopus nigricans

Yu, Zhidan, Li, Xiaoqin, Zhou, Fang, Zhang, Pengying, Chen, Kaoshan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.38 MB

2020

24

Corrigendum to âDesign of selective PI3KÎ´ inhibitors using an iterative scaffold-hopping workflowâ [Bioorg. Med. Chem. Lett. 29 (2019) 2575â2580]

Fradera, Xavier, Methot, Joey L., Achab, Abdelghani, Christopher, Matthew, Altman, Michael D., Zhou, Hua, McGowan, Meredeth A., Kattar, Sam D., Wilson, Kevin, Garcia, Yudith, Augustin, Martin A., Lesb

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 252 KB

2020

25

Graphical abstract TOC

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 123 KB

2020

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