Volume 4; Issue 20

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Bioorganic & Medicinal Chemistry Letters
Volume 4; Issue 20

Bioorganic & Medicinal Chemistry Letters

Volume 4; Issue 20

1

Graphical abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 338 KB

english, 1994

2

Synthesis and 5-HT3 receptor antagonist potency of novel (endo) 3,9-diazabicyclo[3.3.1]nonan-7-amino derivatives

J. Bermudez, L. Gaster, J. Gregory, J. Jerman, G.F. Joiner, F.D. King, S.K. Rahman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 181 KB

english, 1994

3

DNA-binding ability of non-diynene class of dynemicins and Aza-anthraquinones

Rumiko Shimazawa, Ryuichi Shirai, Yuichi Hashimoto, Shigeo Iwasaki

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 451 KB

english, 1994

4

Design of pyrrolo-1,4-benzoxazine derivatives as inhibitors of 5-lipoxygenase and PAF antagonists with anthihistaminic properties

Patrice Demonchaux, Patrick Lenoir, Guy Augert, Pierre Dupassieux

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 257 KB

english, 1994

5

Synthesis and structure-activity relationships of pyrrolidine-modified analogs of the potent cholinergic channel activator, ABT 418

Nan-Horng Lin, Yun He, Anderson David J., James T. Wasicak, Richard Kasson, David Sweeny, Sullivan James P.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 281 KB

english, 1994

6

Synthesis of new thiazinoindole derivatives and their evaluation as inhibitors of human leukocyte elastase and other related serine proteases

Giuseppe Romeo, Filippo Russo, Salvatore Guccione, Renee Chabin, David Kuo, W.B. Knight

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 341 KB

english, 1994

7

Conformationally constrained analogues of diacylglycerol. 9.1 the effect of side-chain orientation on the protein kinase C (PK-C) binding affinity of σ-lactones

Jeewoo Lee, Nancy E. Lewin, Peter M. Blumberg, Victor E. Marquez

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 318 KB

english, 1994

8

DNA topoisomerase II inhibition by substituted 1,2,3,4-tetrahydro-β-carboline derivatives

Erich K. Lehnert, Kelli E. Miller, Jose S. Madalengoitia, Timothy J. Guzi, Timothy L. Macdonald

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 818 KB

english, 1994

9

Diphenylborinic acid is a strong inhibitor of serine proteases

Steven J. Steiner, Jeffrey T. Bien, Bradley D. Smith

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 227 KB

english, 1994

10

Pimolin, a new class of natural product from Pimpinella monoica: A novel dimeric furochromone

Padmanava Pradhan, Devanand L. Luthria, Banerji Asoke

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 181 KB

english, 1994

11

Multiple binding modes with DNA of anthracene-9-carbonyl-N1-spermine probed by LD, CD, normal absorption, and molecular modelling compared with those of spermidine and spermine

Gareth Adlam, Ian S. Blagbrough, Steven Taylor, Harriet C. Latham, Ian S. Haworth, Alison Rodger

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 338 KB

english, 1994

12

Synthesis and antiviral activity of a novel class of HIV-1 protease inhibitors containing a heterocyclic P1′-P2′ amide bond isostere

Scott K. Thompson, Alecia M. Eppley, James S. Frazee, Michael G. Darcy, Robert T. Lum, Thaddeus A. Tomaszek Jr., Lucinda A. Ivanoff, Jane F. Morris, Edmund J. Sternberg, Dennis M. Lambert, Annabellee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 300 KB

english, 1994

13

Penazetidine A, an alkaloid inhibitor of protein kinase C

Khisal A. Alvi, Marcel Jaspars, Phillip Crews, Berta Strulovici, Edwin Oto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 248 KB

english, 1994

14

Selective inhibitors of protein kinase C in a model of graft-vs-host disease

James P. Demers, William E. Hageman, Sigmond G. Johnson, Dieter H. Klaubert, Richard A. Look, John B. Moore

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 464 KB

english, 1994

15

Synthesis of cis-δ-phenylmethyl-d-proline using a nitrogen-centered radical derived from a chiral oxaziridine

Jeffrey Aubé, Belgin Gülgeze, Xin Peng

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 248 KB

english, 1994

16

Highly water soluble taxol derivatives: 2′-polyethyleneglycol esters as potential prodrugs

Richard B. Greenwald, Annapurna Pendri, Durgadas Bolikal, Carl W. Gilbert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 218 KB

english, 1994

17

Stereospecific bio-reversibility of dinucleoside S-alkyl phosphorothiolates to dinucleoside phosphorothioates

Radhakrishnan P. Iyer, Dong Yu, Sudhir Agrawal

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 301 KB

english, 1994

18

Synthesis and preliminary pharmacological evaluation of 2-benzyloxy substituted aryl ketones as 5-HT4 receptor antagonists

R.D. Clark, A. Jahangir, J.A. Langston, K.K. Weinhardt, A.B. Miller, E. Leung, D.W. Bonhaus, E.H.F. Wong, R.M. Eglen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 174 KB

english, 1994

19

Structure-activity studies of N-cyano-3-pyridinecarboxamidines and their amide and thioamide congeners

Tatsuo Nakajima, Tomoko Kashiwabara, Toshio Izawa, Shohachi Nakajima

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 171 KB

english, 1994

20

Structure and synthesis of clausenaquinone-a. A novel carbazolequinone alkaloid and bioactive principle from Clausena excavata

Tian-Shung Wu, Shiow-Chyn Huang, Pei-Lin Wu, Kuo-Hsiung Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 145 KB

english, 1994

21

Probing the importance of the second chloroethyl arm of a benzoic acid mustard derivative of an imidazole-containing analogue of distamycin

John A. Hartley, Michael D. Wyatt, Bonnie J. Garbiras, Celese Richter, Moses Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 462 KB

english, 1994

22

An immunosensor for the detection of human B-lymphocytes

Bernd König, Michael Grätzel

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 278 KB

english, 1994

23

Synthesis and neuraminidase inhibition studies of 4-azido, amino, and acetamido substituted sialosides

Subramaniam Sabesan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 199 KB

english, 1994

24

Ketones related to the benzoate 5-HT4 receptor antagonist RS-23597 are high affinity partial agonists

R.D. Clark, A. Jahangir, J.A. Langston, K.K. Weinhardt, A.B. Miller, E. Leung, R.M. Eglen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 200 KB

english, 1994

25

Additions and corrections

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

File:

PDF, 15 KB

1994