Volume 4; Issue 7

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Bioorganic & Medicinal Chemistry Letters
Volume 4; Issue 7

Bioorganic & Medicinal Chemistry Letters

Volume 4; Issue 7

1

Stereoselective synthesis of novel analogues of 2′-deoxy- and 2′,3′-dideoxynucleosides with potential antiviral activity

Daniel O. Cicero, Philippe J.S. Neuner, Ornella Franzese, Chiara D'Onofrio, Adolfo M. Iribarren

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 372 KB

english, 1994

2

Replacement of the phosphodiester linkage in oligonucleotides: Comparison of two structural amide isomers

Alain De Mesmaeker, Jacques Lebreton, Adrian Waldner, Valérie Fritsch, Romain M. Wolf

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 424 KB

english, 1994

3

Simple synthesis of O,N-protected tunicamine - the undecose part of tunicamycins

Wojciech Karpiesiuk, Anna Banaszek

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 267 KB

english, 1994

4

Synthesis of a dermatan sulphate-like hexasaccharide with a “non-glycosamino” glycan structure

J.E.M. Basten, C.A.A. van Boeckel, G. Jaurand, M. Petitou, N.M. Soijker, P. Westerduin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 397 KB

english, 1994

5

Chemical and plasma hydrolyses of a diphenyl α-aminomethyl phosphonate prodrug inhibitor of neutral endopeptidase 24.11

Stéphane De Lombaert, Kuldeep Singh, Louis Blanchard, Victor F. Soliman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 313 KB

english, 1994

6

Enantioselective reduction of ethyl 3-methyl-2-oxobutanoate by an enzymatic system from callus of catharanthus roseus

Hiroki Hamada, Nobuyoshi Nakajima, Yoshiko Shisa, Makoto Funahashi, Kaoru Nakamura

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 206 KB

english, 1994

7

Synthesis and in vitro cytotoxicity of 1,3-dioxolane-2-(2-ethanamine)-2-methanamine platinum(II) complexes

Dae-Kee Kim, Jongsik Gam, Key H. Kim

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 485 KB

english, 1994

8

A thermostable chymotrypsin derivative soluble in toluene

Hyung Soon Park, Junghun Suh

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 270 KB

english, 1994

9

Alkyl ether analogs of the FK-506 related, immunosuppressive macrolide L-683,590 (ascomycin)

Mark T. Goulet, Derek W. Hodkey, Mary Jo Staruch, Francis J. Dumont, John G. Cryan, William H. Parsons, Matthew J. Wyvratt

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 433 KB

english, 1994

10

Alkyl ether derivatives of the FK-506 related, immunosuppressive macrolide L-683,742 (C31-O-desmethyl ascomycin)

Mark T. Goulet, Derek W. Hodkey, Mary Jo Staruch, Francis J. Dumont, Shirley Lin, Shirley H.Y. Hung, John J. Siekierka, Matthew J. Wyvratt

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 374 KB

english, 1994

11

Synthesis and in vitro anti-human immunodeficiency virus activity of artemisinin (qinghaosu)-related trioxanes

Mankil Jung, Raymond F. Schinazi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 248 KB

english, 1994

12

The relative ability of BSO and other γ-glutamylcysteine synthetase inhibitors to both deplete glutathione and alter drug metabolizing enzyme activities

Michael R. Franklin, Jeanette C. Roberts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 435 KB

english, 1994

13

Dehydrolysine containing analogues of tuftsin: Synthesis and bioactivity

Sunanda D. Gupta, Ratanmani Jain, Virender S. Chauhan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 317 KB

english, 1994

14

N-chloromethyl quinuclidinium derivatives: A new class of irreversible ligands for 5-HT3 receptors.

M. Langlois, J.L. Soulier, M. Mathé-Allainmat, C. Gallais, B. Brémont, S. Shen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 327 KB

english, 1994

15

1,3-Oxazino[4,5-b]indole-2,4-(1H,9H)-diones and 5,6-dimethylpyrrolo-[2,3-d]-1,3-oxazin-2,4-(1H,7H)-diones as serine protease inhibitors

Mark R. Player, J.Walter Sowell Sr., Girish S. Patil, Kam Chih-Min, James C. Powers

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 312 KB

english, 1994

16

Graphical abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 397 KB

english, 1994

17

Novel cholecystokinin receptor ligands: Oxopiperazines derived from Boc-CCK-4

Andrzej R Batt, David A Kendrick, Elizabeth Mathews, David P Rooker, Hamish Ryder, Graeme Semple, Michael Szelke

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 314 KB

english, 1994

18

Evaluation of (2S,4S)/(2R,4R) and (2S,4R)/(2R,4S) 6,6-N,N-dimethyl-2-methyl-2-oxo-1,3-dioxa-4-hexadecyl-6,aza-2-phosphacyclooctane bromide as inhibitors for protein kinase C, carnitine octanoyltransferase, and carnitine palmitoyltransferase

G. Kumaravel, N. Nic a' Bháird, F.R. Fronczek, R.R. Ramsay, C.L. Ashendel, R.D. Gandour

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 245 KB

english, 1994

19

Peptide based P21RAS farnesyl transferase inhibitors: systematic modification of the tetrapeptide CA1A2X motif

K. Leftheris, T. Kline, S. Natarajan, M.K. DeVirgilio, Y.H. Cho, J. Pluscec, C. Ricca, S. Robinson, B.R. Seizinger, V. Manne, C.A. Meyers

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 349 KB

english, 1994

20

Asymmetric synthesis of cis- and trans-γ-lactones useful in HIV-1 protease inhibitor synthesis

Michael P. Trova, Allan Wissner, Wellington T. Casscles Jr., Grace C. Hsu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 289 KB

english, 1994