Volume 5; Issue 11

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Bioorganic & Medicinal Chemistry Letters
Volume 5; Issue 11

Bioorganic & Medicinal Chemistry Letters

Volume 5; Issue 11

1

In search of the non-polar amopyroquin metabolite. A consideration of polonovski-type reactivity

David J. Aitken, Isabelle Jobet-Hermelin, Henri-Philippe Husson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 206 KB

english, 1995

2

Synthesis and antiviral activity of phosphonate derivatives of enantiomeric dihydro-2H-pyranyl nucleosides

María-Jesús Pérez-Pérez, Jan Balzarini, Jef Rozenski, Erik De Clercq, Piet Herdewijn

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 212 KB

english, 1995

3

A PNA-DNA linker synthesis of N-((4,4′-dimethoxytrityloxy)ethyl)-N-(thymin-1-ylacetyl)glycine

Kenneth H. Petersen, Dorte K. Jensen, Michael Egholm, Peter E. Nielsen, Ole Buchardt

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 250 KB

english, 1995

4

Active-site conformation of 17-(3-pyridyl)androsta-5,16-dien-3β-ol, a potent inhibitor of the P450 enzyme C17α-hydroxylase/C17-20 lyase

David F. Burke, Charles A. Laughton, Chris F. Snook, Stephen Neidle, Gerard A. Potter, Michael Jarman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 228 KB

english, 1995

5

Acetylcholinesterase inhibition by alkaloids of the ant's venom Monomorium minutum

Nello Ronzani, Maryse Lajat

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 98 KB

english, 1995

6

Enzymatic synthesis of Thia-L-tryptophans

Robert S. Phillips, Louis A. Cohen, Ulf Annby, David Wensbo, Salo Gronowitz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 112 KB

english, 1995

7

16,19-cis-murisolin and murisolin a, two novel bioactive mono-tetrahydrofuran annonaceous acetogenins from Asimina triloba seeds

Mi Hee Woo, Lu Zeng, Qing Ye, Zhe-Ming Gu, Geng-Xian Zhao, Jerry L. McLaughlin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 347 KB

english, 1995

8

α-Phenoxyphenylacetic acid derived angiotensin II antagonists with low nanomolar AT1/AT2 receptor subtype affinity (Part II)

Thomas F. Walsh, Kenneth J. Fitch, Raymond S.L. Chang, Kristie A. Faust, Tsing-Bau Chen, Salah D. Kivlighn, Gloria J. Zingaro, Victor J. Lotti, Peter K.S. Siegl, Arthur A. Patchett, William J. Greenle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 212 KB

english, 1995

9

Synthesis of peptide nucleic acids (PNA) by submonomer solid-phase synthesis

Lutz S. Richter, Ronald N. Zuckermann

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 250 KB

english, 1995

10

The effect of Pyrrolo[3,4-c]carbazole derivatives on spinal cord ChAT activity

David P. Rotella, Marcie A. Glicksman, J.Eric Prantner, Nicola T. Neff, Robert L. Hudkins

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 198 KB

english, 1995

11

2,4,5- triarylimidazole inhibitors of IL-1 biosynthesis

Timothy F. Gallagher, Susan M. Fier-Thompson, Ravi.S. Garigipati, Margaret E. Sorenson, Juanita M. Smietana, Dennis Lee, Paul E. Bender, John C. Lee, Jeffrey T. Laydon, Don E. Griswold, Marie C. Chabo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 316 KB

english, 1995

12

Synthetic studies on the furan ring of wortmannin

Bryan H. Norman, Jonathan Paschal, Chris J. Vlahos

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 185 KB

english, 1995

13

An unusually facile SnAr 14-membered biaryl ether macrocyclization reaction suitable for preparation of the cycloisodityrosine subunit of bouvardin, deoxybouvardin and related agents

Dale L. Boger, Robert M. Borzilleri

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 229 KB

english, 1995

14

A single precursor approach to new DNA cleaving and crosslinking agents

David J. Jebaratnam, Dev P. Arya, Hang Chen, S. Kugabalasooriar, Duc Vo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 327 KB

english, 1995

15

Synthesis and evaluation of diacylhydrazines as inhibitors of the interleukin-1β converting enzyme (ICE)

Todd L. Graybill, Roland E. Dolle, Carla T. Helaszek, Mark A. Ator, Joost Strasters

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 374 KB

english, 1995

16

Preparation of neurotensin analogs with a novel pro-tyr replacement

David A. Nugiel, Wagner Regina M., William K. Schmidt

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 181 KB

english, 1995

17

Graphical abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 297 KB

english, 1995

18

Stereochemical differentiation of anticonvulsant and antihypertensive effects in 4-(fluorobenzoylamino)-benzopyrans

Thomas P. Blackburn, Robin E. Buckingham, Wai N. Chan, John M. Evans, Michael S. Hadley, Mervyn Thompson, Neil Upton, Tania O. Stean, Geoffrey Stemp, Antonio K. Vong

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 193 KB

english, 1995

19

Synthesis and structure-activity relationships of 2′-(R) and (S) pyrrolidine-modified analogs of the cholinergic channel activator, ABT-418

Nan-Horng Lin, Yun He, Stephen P. Arneric, James P. Sullivan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 322 KB

english, 1995

20

A medicinal chemistry evaluation of the autoinhibitory domain of calcineurin

Meheryar N. Rivetna, Scott P. Salowe, Richard L. Tolman, A.Brian Jones

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 251 KB

english, 1995

21

Potent dual antagonists of endothelin and angiotensin II receptors derived from α-phenoxyphenylacetic acids (Part III)

Thomas F. Walsh, Kenneth J. Fitch, David L. Williams Jr., Kathryn L. Murphy, Nancy A. Nolan, Douglas J. Pettibone, Raymond S.L. Chang, Stacey S. O'Malley, Bradley V. Clineschmidt, Daniel F. Veber, Wil

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 243 KB

english, 1995

22

Octahydro-1,2,3,4,4a,5,11,11a-pyrido[3,4-c][1,5]benzoxazepines: conformationally restricted fentanyl analogs

Linas V. Kudzma, Suzanne M. Evans, Stanhope P. Turnbull Jr., Sherry A. Severnak, Edward F. Ezell

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 210 KB

english, 1995

23

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 65 KB

english, 1995