Volume 6; Issue 14

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Bioorganic & Medicinal Chemistry Letters
Volume 6; Issue 14

Bioorganic & Medicinal Chemistry Letters

Volume 6; Issue 14

1

SAR of 2-benzyl-4-aminopiperidines: CGP 49823, an orally and centrally active non-peptide NK1 antagonist

Silvio Ofner, Kathleen Hauser, Walter Schilling, Annick Vassout, Siem J. Veenstra

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 331 KB

english, 1996

2

New heteroaryl-spaced phosphono α-amino acids are competitive NMDA antagonists with analgesic activity

Britt-Marie Swahn, Alf Claesson, Benjamin Pelcman, Yevgeni Besidski, Håkan Molin, Mats P. Sandberg, Odd-Geir Berge

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 308 KB

english, 1996

3

Design, synthesis and binding affinities of novel non-peptide mimics of somatostatin/sandostatin®

Dominique Damour, Michel Barreau, Jean-Charles Blanchard, Marie-Claude Burgevin, Adam Doble, Frederic Herman, Guy Pantel, Evelyne James-Surcouf, Marc Vuilhorgne, Serge Mignani, Lydie Poitout, Yves Le

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 317 KB

english, 1996

4

Tripeptidyl pyridinium methyl ketones as potent active site inhibitors of thrombin

Torsten Steinmetzer, Yasuo Konishi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 295 KB

english, 1996

5

Anti-human immunodeficiency and anti-hepatitis B virus activities of β-l-2′,3′-dideoxy purine nucleosides

Pascal J. Bolon, Peiyuan Wang, Chung K. Chu, Gilles Gosselin, Valérie Boudou, Claire Pierra, Christophe Mathé, Jean-Louis Imbach, Abdesselem Faraj, Abdelaziz el Alaoui, Jean-Pierre Sommadossi, S.Balak

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 305 KB

english, 1996

6

Application of the “trimethyl lock”1 to Ganciclovir, a pro-prodrug with increased oral bioavailability

Michael P. Dillon, Haiying Cai, Hans Maag

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 193 KB

english, 1996

7

Decapitation of a 5' capped RNA by an antisense copper complex conjugate

Brenda F. Baker, Kanda Ramasamy, John Kiely

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 367 KB

english, 1996

8

Design and synthesis of phosphinic acids that triply inhibit endothelin converting enzyme, angiotensin converting enzyme and neutral endopeptidase 24.11

Brian A. McKittrick, Andrew W. Stamford, Xiaoyu Weng, Ke Ma, Samuel Chackalamannil, Michael Czarniecki, ReneéM. Cleven, Ahmad B. Fawzi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 304 KB

english, 1996

9

Co-electropolymerization of a viologen oligomer and lipoamide dehydrogenase on an electrode surface. Application to cofactor regeneration

Mihaela Draganoiu Leonida, Albert J. Fry, Susan B. Sobolov, Kamen I. Voivodov

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 242 KB

english, 1996

10

Thromboxane modulating agents. 2. Thromboxane receptor antagonists derived from the thromboxane synthase inhibitor dazmegrel.

Roger P. Dickinson, Kevin N. Dack, John Steele, Michael S. Tute

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 306 KB

english, 1996

11

Synthesis of CD-ring modified 1α,25-dihydroxy vitamin D analogues : E-ring analogues

K. Sabbe, C. D'Hallewyn, P. De Clercq, M. Vandewalle, R. Bouillon, A. Verstuyf

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 281 KB

english, 1996

12

Synthesis of CD-ring modified 1α,25-dihydroxy vitamin D analogues: C-ring analogues

Gui-Dong Zhu, Yongjun Chen, Xiaoming Zhou, Maurits Vandewalle, Pierre J. De Clercq, R. Bouillon, A. Verstuyf

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 317 KB

english, 1996

13

Drupangtonine, a novel antileukemic alkaloid from Cephalotaxus harringtonia var. drupacea

Ichiro Takano, Ichiro Yasuda, Motohiro Nishijima, Yukio Hitotsuyanagi, Koichi Takeya, Hideji Itokawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 123 KB

english, 1996

14

Inhibitors of MMP-1: an examination of P1′ Cα gem-disubstitution in the succinamide hydroxamate series

Ralph P. Robinson, John A. Ragan, Brian J. Cronin, Kathleen M. Donahue, Lori L. Lopresti-Morrow, Peter G. Mitchell, Lisa M. Reeves, Sue A. Yocum

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 259 KB

english, 1996

15

Inhibitors of MMP-1: an examination of P1′ Cα gem-disubstitution in the N-carboxyalkylamine and glutaramide carboxylate series

Ralph P. Robinson, Brian J. Cronin, Kathleen M. Donahue, Brian P. Jones, Lori L. Lopresti-Morrow, Peter G. Mitchell, James P. Rizzi, Lisa M. Reeves, Sue A. Yocum

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 342 KB

english, 1996

16

Peptidomimetic growth hormone secretagogues: synthesis and biological activities of analogs varied at the indole nucleus of the prototypical spiropiperidine L-162,752

Ravi P. Nargund, Meng-Hsin Chen, David B.R. Johnston, Khaled J. Barakat, James R. Tata, Kang Cheng, Thomas M. Jacks, Wanda W.-S. Chan, Liente Wei, Bridget R. Butler, Gerard J. Hickey, Roy G. Smith, Ar

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 297 KB

english, 1996

17

GPI membrane anchors: synthesis and functional evaluation of aminoglucosyl phosphatidylinositol core analogs

Jianhua Ye, William T. Doerrler, Mark A. Lehrman, J.R. Falck

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 249 KB

english, 1996

18

A study of 3-amino-N-hydroxypropanesulfonamide derivatives as potential GABAB agonists and their fragmentation to 3-aminopropanesulfinic acid

Ho-Jane Shue, Xiao Chen, David J. Blythin, Nicholas I. Carruthers, James M. Spitler, Shing-Chun Wong, Richard W. Chapman, Charles Rizzo, Robert West, Hoyan S. She

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 307 KB

english, 1996

19

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 74 KB

english, 1996

20

Graphical abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 316 KB

english, 1996

21

Synthesis of α-difluoro and α-difluoro-β-trifluoroketo-derivatives as potential inhibitors for Cholesterol Ester Hydrolase

Béatrice David, Francis Schuber

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 229 KB

english, 1996

22

Synthesis and antimicrobial activity of 4-amino trinems

Maria Elvira Tranquillini, Gian Luca Araldi, Daniele Donati, Giorgio Pentassuglia, Anna Pezzoli, Antonella Ursini

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 231 KB

english, 1996

23

N-Benzylated benzimidazol-2-one derivatives: activators of large-conductance Ca2+-dependent K+ channels

Nicholas A. Meanwell, Sing-Yuen Sit, Jinnian Gao, Christopher G. Boissard, Janet Lum-Ragan, Steven I. Dworetzky, Valentin K. Gribkoff

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 286 KB

english, 1996

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