Volume 6; Issue 23

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Bioorganic & Medicinal Chemistry Letters
Volume 6; Issue 23

Bioorganic & Medicinal Chemistry Letters

Volume 6; Issue 23

1

Protein-ligand interactions. 6 nicotinic acetylcholine receptor agonist activity of isoquinoline alkaloids

C.G. Whiteley, S. Daya

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 364 KB

english, 1996

2

Nucleosides and nucleotides. 161. Incorporation of 5-(N-aminoalkyl)carbamoyl-2′-deoxycytidines into oligodeoxyribonucleotides by a convenient post-synthetic modification method

Yukari Nomura, Noriyasu Haginoya, Yoshihito Ueno, Akira Matsuda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 336 KB

english, 1996

3

Nucleosides and nucleotides. 162. Facile synthesis of 5′-5′-linked oligodeoxyribonucleotides with the potential for triple-helix formation

Yoshihito Ueno, Akira Ogawa, Aiko Nakagawa, Akira Matsuda

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 344 KB

english, 1996

4

Synthesis of novel ellipticine analogues and their inhibition of Moloney leukaemia reverse transcriptase

Géza Timári, Tibor Soós, György Hajós, András Messmer, János Nacsa, József Molnár

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 305 KB

english, 1996

5

Antitumor agents 171. Cytotoxicities of lobatosides B, C, D, and E, cyclic bisdesmosides isolated from Actinostemma lobatum maxim

Toshihiro Fujioka, Yoshiki Kashiwada, Hikaru Okabe, Kunihide Mihashi, Kuo-Hsiung Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 198 KB

english, 1996

6

Application of the Heck reaction in the synthesis of truncated naphthoic acid retinoids

Kuo-Long Yu, Simon Chen, Jacek Ostrowski, Kenneth M. Tramposch, Peter R. Reczek, Muzammil M. Mansuri, John E. Starrett Jr.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 286 KB

english, 1996

7

Structural modifications of 6-naphthalene-2-carboxylate retinoids

Kuo-Long Yu, Jacek Ostrowski, Simon Chen, Kenneth M. Tramposch, Peter R. Reczek, Muzammil M. Mansuri, John E. Starrett Jr.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 325 KB

english, 1996

8

Coumarin-based prodrugs 2. Synthesis and bioreversibility studies of an esterase-sensitive cyclic prodrug of dadle, an opioid peptide

Binghe Wang, Wei Wang, Huijuan Zhang, Daxian Shan, Terrill D. Smith

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 245 KB

english, 1996

9

New simplified inhibitors of EPSP synthase: The importance of ring size for recognition at the shikimate 3-phosphate site

Mark L. Peterson, Susan D. Corey, Jose L. Font, Mark C. Walker, James A. Sikorski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 291 KB

english, 1996

10

Evaluation of furofuran as a P2 ligand for symmetry-based HIV protease inhibitors

Xiaoqi Chen, Lin Li, Dale J. Kempf, Hing Sham, Norman E. Wideburg, Ayda Saldivar, Sudthida Vasavanonda, Kennan C. Marsh, Edith McDonald, Daniel W. Norbeck

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 313 KB

english, 1996

11

Dual inhibition of angiotensin-converting enzyme and neutral endopeptidase by tricyclic benzazepinone thiols

Stéphane De Lombaert, Louis Blanchard, Lisa B. Stamford, Yumi Sakane, Carol Berry, Rajendra D. Ghai, Angelo J. Trapani

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 320 KB

english, 1996

12

Conformationally restricted 1,5-diarylpyrazoles are selective COX-2 inhibitors

Stephen R. Bertenshaw, John J. Talley, D.J. Rogier, Matthew J. Graneto, Carol M. Koboldt, Yan Zhang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 208 KB

english, 1996

13

Peptidomimetic inhibitors of herpes virus ribonucleotide reductase. Correlation between herpes simplex and varicella zoster virus

Montse Llinàs-Brunet, Neil Moss, Erika Scouten, Michel Liuzzi, Robert Déziel

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 259 KB

english, 1996

14

Retropane — a new rhenium complex as a potential ligand to label the dopamine transporter

Alexander Hoepping, Hartmut Spies, Bernd Johannsen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 159 KB

english, 1996

15

Pyrrolylquinoxalinediones: A new class of AMPA receptor antagonists

W. Lubisch, B. Behl, H.P. Hofmann

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 295 KB

english, 1996

16

Solid phase synthesis of polylactosamine oligosaccharide

Hiroki Shimizu, Yukishige Ito, Osamu Kanie, Tomoya Ogawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 291 KB

english, 1996

17

Peptidyl epoxides as inhibitors of α-chymotrypsin: Remarkable change from irreversible to reversible competitive inhibitor as a consequence of the improvement of binding affinity

Dong H. Kim, Zhi-Hong Li, Soo Suk Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 200 KB

english, 1996

18

Small peptidic aldehyde inhibitors of human rhinovirus 3C protease

Timothy A. Shepherd, Gregory A. Cox, Emma McKinney, Joseph Tang, Mark Wakulchik, Ronald E. Zimmerman, Elcira C. Villarreal

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 231 KB

english, 1996

19

Specific and nonspecific inhibition of transcription by DNA, PNA, and phosphorothioate promoter analog duplexes

Susan E. Hamilton, Mridula Iyer, James C. Norton, David R. Corey

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 277 KB

english, 1996

20

1-(Dihydroxyphosphynyl)vinyl phosphate: The phosphonate analogue of phosphoenolpyruvate is a pH-dependent substrate of Kdo8P synthase

Yaakov Benenson, Valery Belakhov, Timor Baasov

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 346 KB

english, 1996