Volume 6; Issue 24

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Bioorganic & Medicinal Chemistry Letters
Volume 6; Issue 24

Bioorganic & Medicinal Chemistry Letters

Volume 6; Issue 24

1

Chemistry and pharmacokinetics of diarylthiophenes and terphenyls as selective COX-2 inhibitors

Donald J.P. Pinto, Robert A. Copeland, Maryanne B. Covington, William J. Pitts, Douglas G. Batt, Michael J. Orwat, Gilbert N. Lam, Amita Joshi, Yuk-Charn Chan, Shuaige Wang, James M. Trzaskos, Ronald

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 330 KB

english, 1996

2

(N-acyl-N-alkyl)glycyl borolysine analogs: A new class of potent thrombin inhibitors

Robert A. Galemmo Jr., John M. Fevig, David J. Carini, Joseph Cacciola, Brian L. Wells, Gregory L. Hillyer, Joseph Buriak Jr., Karen A. Rossi, Pieter F.W. Stouten, Richard S. Alexander, Richard Hilmer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 372 KB

english, 1996

3

Potent cyclic urea HIV protease inhibitors with benzofused heterocycles as P2/P2′ groups

James D. Rodgers, Barry L. Johnson, Haisheng Wang, Roger A. Greenberg, Susan Erickson-Viitanen, Ronald M. Klabe, Beverly C. Cordova, Marlene M. Rayner, Gilbert N. Lam, Chong-Hwan Chang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 274 KB

english, 1996

4

Asiaticoside mimetics as wound healing agent

Pil-Jong Shim, Jae-Ho Park, Min-Sun Chang, Min-Jung Lim, Do-Ha Kim, Young Hoon Jung, Sang-Sup Jew, Eun Hee Park, Hee-Doo Kim

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 224 KB

english, 1996

5

The nature of interaction between the carboxylate of substrates and the guanidinium moiety of Arg-145 in carboxypeptidase A probed by inhibitors of the enzyme

Dong H. Kim, Jeong- il Park

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 231 KB

english, 1996

6

Novel inhibitors of influenza sialidases related to GG167 structure-activity, crystallographic and Molecular dynamics studies with 4H-pyran-2-carboxylic acid 6-carboxamides

Paul W. Smith, Steven L. Sollis, Peter D. Howes, Peter C. Cherry, Kevin N. Cobley, Helen Taylor, Andrew R. Whittington, Jan Scicinski, Richard C. Bethell, Neil Taylor, Tadeusz Skarzynski, Anne Cleasby

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 289 KB

english, 1996

7

Enzymatic fucosylations with purine-diphosphate-fucoses (PDP-Fucoses)

Gabi Baisch, Reinhold Öhrlein, Andreas Katopodis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 163 KB

english, 1996

8

Synthesis and evaluation of novel 1,5-Benzodiazepines as potent and selective CCK-B ligands. Effect of the substitution of the N-5 phenyl with alkyl groups

Gabriella Finizia, Daniele Donati, Beatrice Oliosi, Maria Elvira Tranquillini, Antonella Ursini

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 247 KB

english, 1996

9

Stereoselective synthesis of 2-amino-1-hydroxy-3-phenylpropylphosphonic acid

Jan Zygmunt, Roman Gancarz, Barbara Lejczak, Piotr Wieczorek, Pawel Kafarski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 212 KB

english, 1996

10

Identification and biological activity of novel peptidomimetic gastrin/CCK-B receptor agonists

Graeme Semple, Hamish Ryder, David A. Kendrick, Andrzej R. Batt, Elizabeth Mathews, David P. Rooker, Michael Szelke, Akito Nishida, Keiji Miyata

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 310 KB

english, 1996

11

Enantioselective synthesis of a pyrrolo-benzothiadiazine derivative S 18986, a new AMPA receptor positive modulator

P. Desos, B. Serkiz, P. Morain, J. Lepagnol, A. Cordi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 314 KB

english, 1996

12

Functional groups positioned in unusual asymmetric microenvironments

Christian M. Rojas, Julius Rebek Jr.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 252 KB

english, 1996

13

Solid-phase synthesis of carbohydrate and phosphodiester modified 2′–5′ oligoadenylate analogs

Stephanie A. Hartsel, William S. Marshall

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 331 KB

english, 1996

14

Inhibition of calpain by peptidyl heterocycles

Ming Tao, Ron Bihovsky, James C. Kauer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 187 KB

english, 1996

15

Synthesis and structure-activity relationships of 9-substituted acridines as endothelin-A receptor antagonists

X.-M. Cheng, C. Lee, S. Klutchko, T. Winters, E.E. Reynolds, K.M. Welch, M.A. Flynn, A.M. Doherty

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 241 KB

english, 1996

16

Lipophilic bis-arylsulfonates as inhibitors of the CD4-gp120 interaction

Raymond J. Patch, John C. Roberts, Huai Gao, Zhan Shi, Ariamala Gopalsamy, Azis Kongsjahju, Kevin Daniels, Paul J. Kowalczyk, Marie-Rose van Schravendijk, Kristin A. Gordon, Peter V. Pallai

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 355 KB

english, 1996

17

A comparative SAR and computer modeling study of benzisothiazolone, mechanism-based inhibitors with porcine pancreatic and human leukocyte elastase

Dennis J. Hlasta, John J. Court, Ranjit C. Desai, Timothy G. Talomie, Jian Shen, Richard P. Dunlap, Catherine A. Franke, Albert J. Mura

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 332 KB

english, 1996

18

Novel thrombin inhibitors that are based on a macrocyclic tripeptide motif

Michael N. Greco, Eugene T. Powell, Leonard R. Hecker, Patricia Andrade-Gordon, Jack A. Kauffman, Joan M. Lewis, Venkatapathy Ganesh, Alexander Tulinsky, Bruce E. Maryanoff

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 280 KB

english, 1996

19

A model for the taxol (paclitaxel)/epothilone pharmacophore

Jeffrey D. Winkler, Paul H. Axelsen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 222 KB

english, 1996

20

Additions and corrections

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

File:

PDF, 14 KB

1996

21

Anti-pneumocystis activity of bis-amidoximes and bis-o-alkylamidoximes prodrugs

David W. Boykin, Arvind Kumar, James E. Hall, Brendan C. Bender, Richard R. Tidwell

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 213 KB

english, 1996

22

Novel tricyclic aminoacetyl and sulfonamide inhibitors of Ras farnesyl protein transferase

F.George Njoroge, Bancha Vibulbhan, Carmen S. Alvarez, W.Robert Bishop, Joanne Petrin, Ronald J. Doll, V. Girijavallabhan, Ashit K. Ganguly

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 275 KB

english, 1996

23

Peptide inhibitors of IKB protease: Modification of the C-termini of Z-LLF-CHO

Mark J. Suto, Robert W. Sullivan, Lynn J. Ransone

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 263 KB

english, 1996

24

Discovery of antirhinoviral leads by screening a combinatorial library of ureas prepared using covalent scavengers

Stephen W Kaldor, James E Fritz, Joseph Tang, Emma R McKinney

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 176 KB

english, 1996

25

Recognition of a G-C base pair by α-N7-deoxyinosine within the pyrimidine-purine-pyrimidine DNA triple helical motif

Judith Marfurt, Jürg Hunziker, Christian Leumann

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 254 KB

english, 1996

26

6-(4-Phenyl-benzyloxy-methyl) guvacine. Synthesis, GABA uptake inhibitor and muscarinic properties

Philippe Bisel, Jean Pierre Gies, Gilbert Schlewer, Camille G. Wermuth

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 170 KB

english, 1996

27

SAR of 2-benzyl-4-aminopiperidines NK1 antagonists. Part 21. synthesis of CGP 49823

Siem J. Veenstra, Kathleen Hauser, Walter Schilling, Claudia Betschart, Silvio Ofner

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 316 KB

english, 1996

28

Synthesis and antiangiogenic activity of new carbohydrate derivatives

G. Dorey, P. Léon, S. Sciberras, S. Léonce, N. Guilbaud, A. Pierré, G. Atassi, D.C. Billington

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 329 KB

english, 1996

29

Solid-phase synthesis of peptidosulfonamide containing peptides derived from Leu-enkephalin

Dries B.A de Bont, Gerard D.H Dijkstra, Jack A.J den Hartog, Rob M.J Liskamp

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 377 KB

english, 1996

30

Benzolactam growth hormone secretagogues: Replacement of the C-3 amide bond in L-692,429

Hyun O Ok, John L Szumiloski, George A Doldouras, William R Schoen, Kang Cheng, Wanda W.-S Chan, Bridget S Butler, Roy G Smith, Michael H Fisher, Matthew J Wyvratt

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 253 KB

english, 1996

31

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 91 KB

english, 1996

32

Graphical abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 485 KB

english, 1996

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