Volume 7; Issue 17

Main
Bioorganic & Medicinal Chemistry Letters
Volume 7; Issue 17

Bioorganic & Medicinal Chemistry Letters

Volume 7; Issue 17

1

Synthesis of 7-membered cyclic hydroxyguanidines: Novel HIV-1 protease inhibitors

Prabhakar K. Jadhav, Francis J. Woerner, Hon-Wah Man

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 233 KB

english, 1997

2

Synthesis and structural characterization of conjugates of adenosine and tetra-aspartate, novel analogs of ATP

Tõnis Pehk, Asko Uri

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 365 KB

english, 1997

3

Synthesis and in vitro cytotoxicity of aminocoumarin platinum(II) complexes

George Kokotos, Vassiliki Theodorou, Chryssa Tzougraki, Dieter L.D. Deforce, Elfreide G. Van den Eeckhout

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 197 KB

english, 1997

4

Parallel-stranded duplex DNA formed by a new base pair between guanine and 5-aza-7-deazaguanine

Frank Seela, Alexander Melenewski, Changfu Wei

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 189 KB

english, 1997

5

Novel hydroxyphosphonate inhibitors of CD-45 tyrosine phosphatase

Roger F. Frechette, Caridad Ackerman, Scott Beers, Rich Look, John Moore

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 219 KB

english, 1997

6

Hemisynthesis of rhazinilam analogues: structure - activity relationships on tubulin-microtubule system

Bruno David, Thierry Sévenet, Odile Thoison, Khalijah Awang, Mary Païs, Michel Wright, Daniel Guénard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 242 KB

english, 1997

7

Synthesis and receptor binding studies of quinolinic derivatives as melatonin receptor ligands

Pui-Kai Li, Guo-Hua Chu, Megan L. Gillen, Paula A. Witt-Enderby

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 185 KB

english, 1997

8

Synthesis and evaluation of a designed inhibitor for nonactin biosynthesis in S. griseus ETH A7796

Martyn J. Earle, Nigel D. Priestley

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 250 KB

english, 1997

9

Structure-based design of non-peptidic pyridone aldehydes as inhibitors of interleukin-1β converting enzyme

Julian M.C. Golec, Michael D. Mullican, Mark A. Murcko, Keith P. Wilson, David P. Kay, Stuart D. Jones, Robert Murdoch, Guy W. Bemis, Scott A. Raybuck, Yu-Ping Luong, David J. Livingston

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 383 KB

english, 1997

10

Solid phase synthesis of C-terminal carbohydrate modified enkephalins

Bruno Drouillat, Barrie Kellam, Gyula Dekany, Mike S. Starr, Istvan Toth

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 256 KB

english, 1997

11

Synthesis of rhenium(I) and technetium(I) carbonyl/dithioether ligand complexes bearing 3,17β-estradiol

Martina Reisgys, Frank Wüst, Roger Alberto, Roger Schibli, Paul August Schubiger, Hans-Jürgen Pietzsch, Hartmut Spies, Bernd Johannsen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 184 KB

english, 1997

12

11,21-Bisphenyl-19-norpregnane derivatives are selective antiglucocorticoids

R. Gebhard, H. van der Voort, W. Schuts, W. Schoonen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 283 KB

english, 1997

13

BN 80245: An E-ring modified camptothecin with potent antiproliferative and topoisomerase I inhibitory activities

Olivier Lavergne, Laurence Lesueur-Ginot, Francesc Pla Rodas, Dennis C.H. Bigg

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 199 KB

english, 1997

14

Novel inhibitors of influenza sialidases related to zanamivir. Heterocyclic replacements of the glycerol sidechain

Paul W. Smith, Andrew R. Whittington, Steven L. Sollis, Peter D. Howes, Neil R. Taylor

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 201 KB

english, 1997

15

Discovery of Ro 48-5695: A potent mixed endothelin receptor antagonist optimized from bosentan

Werner Neidhart, Volker Breu, Kaspar Burri, Martine Clozel, Georges Hirth, Uwe Klinkhammer, Thomas Giller, Henri Ramuz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 312 KB

english, 1997

16

Synthesis and biological activity of novel penem sulfoxides and sulfones

Hans Rudolf Pfaendler, Ralf Weishaupt, Claus Medicus

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 208 KB

english, 1997

17

4-Heterocyclyl tetrahydropyridines as selective ligands for the human dopamine D4 receptor

K.E. Haworth, T. Harrison, J.J. Kulagowski, P.D. Leeson, A.P. Owens, M.P. Ridgill, M.R. Teall, M. Fielding, K. Chapman, F. Emms, R. Marwood, S. Patel, K.L. Moss

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 202 KB

english, 1997

18

Design and synthesis of conformationally constrained arginal thrombin inhibitors

Aldo Salimbeni, Fabio Paleari, Renato Canevotti, Marco Criscuoli, Marco Criscuoli, Annalisa Lippi, Mauro Angiolini, Laura Belvisi, Carlo Scolastico, Lino Colombo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 324 KB

english, 1997

19

A conformational study of ligands for omega modulatory sites of GABAa receptors by NOESY NMR spectroscopy and distance geometry

Anne Olivier, Mireille Sevrin, François Durant, Pascal George

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 256 KB

english, 1997

20

Synthesis and biological activities of new heterocyclic aromatic retinoids

P. Diaz, S. Michel, L. Stella, B. Charpentier

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 295 KB

english, 1997

21

Arylacetamide kappa-selective opioid ligands

Anthony D. Pechulis, Sydney Archer, Mark P. Wentland, Ann M. Colasurdo, Jean M. Bidlack

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 263 KB

english, 1997

22

Orevactaene,1 a novel binding inhibitor of HIV-1 rev protein to Rev response element (RRE) from Epicoccum nigrum WC47880

Yue-Zhong Shu, Qingmei Ye, Hui Li, Kathleen F. Kadow, Raouf A. Hussain, Stella Huang, Donald R. Gustavson, Susan E. Lowe, Li-Ping Chang, Dolores M. Pirnik, Krishna Kodukula

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 217 KB

english, 1997

23

Serotonin 5-HT4 agonist activity of a series of meso-azanoradamantane benzamides

Daniel P. Becker, Roger Nosal, Clara I. Villamil, Gary Gullikson, Chafiq Moummi, Dai-Chang Yang, Daniel L. Flynn

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 255 KB

english, 1997

24

C32-amino derivatives of the immunosuppressant ascomycin

Hyun O. Ok, John L. Szumiloski, Thomas R. Beattie, Mark T. Goulet, Mary Jo Staruch, Francis J. Dumont, Matthew J. Wyvratt

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 261 KB

english, 1997

25

The efficient synthesis of a bis-glycosylated steroid drug transport reagent: Methyl 3-β-amino-7α, 12α-di(1′α-glucosyl)-5β-cholate (TC002)

Michael J. Sofia, Ramesh Kakarla, Natan Kogan, Richard Dulina, Y.W. Hui, Nicole T. Hatzenbuhler, Dashan Liu, Anna Chen, Thomas Wagler

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 182 KB

english, 1997

26

Unprecedented detoxification of the cruciferous phytoalexin camalexin by a root phytopathogen

M. Soledade, C. Pedras, Abdul Q. Khan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 375 KB

english, 1997

27

Synthesis of new 3-thiosubstituted carbacephem antibiotics and their activity against penicillin resistant Streptococcus pneumoniae

Larry C. Blaszczak, Clark N. Eid, Jane Flokowitsch, G.Stuart Gregory, Stephen A. Hitchcock, George W. Huffman, Daniel R. Mayhugh, Michael J. Nesler, David A. Preston, Mohammad Zia-Ebrahimi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 208 KB

english, 1997

28

The inhibition of glutamate racemase by d-N-hydroxyglutamate

Suzana Glavas, Martin E. Tanner

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 406 KB

english, 1997

29

3-Substituted-4-hydroxy-7-chromanylacetic acid derivatives as antagonists of the leukotriene B4 (LTB4) receptor

Lawrence A. Reiter, Lawrence S. Melvin Jr., Geraldine L. Crean, Henry J. Showell, Kevin Koch, Michael S. Biggers, John B. Cheng, Robbin Breslow, Maryrose J. Conklyn, Cathy A. Farrell, William A. Hada,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 384 KB

english, 1997

30

Anti-histaminic activity of bromopyrrole alkaloids isolated from Caribbean Agelas sponges

Francesco Cafieri, Rosa Carnuccio, Ernesto Fattorusso, Orazio Taglialatela-Scafati, Teresa Vallefuoco

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 360 KB

english, 1997

31

Design and synthesis of the cartilage protective agent (CPA, Ro32-3555)

M.J. Broadhurst, P.A. Brown, G. Lawton, N. Ballantyne, N. Borkakoti, K.M.K. Bottomley, M.I. Cooper, A.J. Eatherton, I.R. Kilford, P.J. Malsher, J.S. Nixon, E.J. Lewis, B.M. Sutton, W.H. Johnson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 219 KB

english, 1997

32

An aromatic moiety is not essential for pharmacophore binding to sigma binding sites: Synthesis of N-alkylazacycloheptane derivatives as potent sigma ligands

Akitake Yamashita, Nobuyuki Takahashi, Daisuke Mochizuki, Ryuichi Tsujita, Shinji Yamada, Hiromu Kawakubo, Yukio Suzuki, Hideyuki Watanabe

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 178 KB

english, 1997

33

New hepatoprotective saponins, bupleurosides III, VI, IX, and XIII, from Chinese Bupleuri Radix: Structure-requirements for the cytoprotective activity in primary cultured rat hepatocytes

Hisashi Matsuda, Toshiyuki Murakami, Kiyofumi Ninomiya, Masahiro Inadzuki, Masayuki Yoshikawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 333 KB

english, 1997

34

Additions and corrections

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

File:

PDF, 15 KB

1997

35

Synthesis and receptor binding affinity of conformationally restricted retinoic acid analogues

Man Fai Wong, Joyce J Repa, Margaret Clagett-Dame, Robert W Curley Jr.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 292 KB

english, 1997

36

The design and synthesis of orally active short duration spiroindane growth hormone secretagogues

James R. Tata, Zhijian Lu, Thomas M. Jacks, Klaus D. Schleim, Kang Cheng, Liente Wei, Wanda W.-S. Chan, Bridget Butler, Nancy Tsou, Kwan Leung, S.-H.L. Chiu, Gerard Hickey, Roy G. Smith, Arthur A. Pat

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 264 KB

english, 1997

37

Robustaflavone, a naturally occurring biflavanoid, is a potent non-nucleoside inhibitor of hepatitis B virus replication in vitro

Yuh-Meei Lin, David E Zembower, Michael T Flavin, Ralph M Schure, Herbert M Anderson, Brent E Korba, Fa-Ching Chen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 228 KB

english, 1997

38

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 108 KB

english, 1997

39

Graphical abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 532 KB

english, 1997

To build up a library is to create a life. It’s never just a random collection of books.

— Carlos María Domínguez

Official channel

Z-Library Desktop Launcher

Tor version

Z-Library

Z-Library Since 2009 support@z-lib.do

EnglishРусскийEspañolItalianoελληνικάاللغة العربيةBahasa IndonesiaBahasa Malaysiaहिन्दीDeutschFrançaisPortuguêsУкраїнськаPolski中文繁體中文日本語Tiếng ViệtAzərbaycan DiliՀայոց լեզուภาษาไทยTürk Diliქართველიবাংলাپښتوతెలుగుاردو한국어SrpskiБългарски