Volume 9; Issue 17

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Bioorganic & Medicinal Chemistry Letters
Volume 9; Issue 17

Bioorganic & Medicinal Chemistry Letters

Volume 9; Issue 17

1

Human telomerase inhibition by substituted acridine derivatives

R. John Harrison, Sharon M. Gowan, Lloyd R. Kelland, Stephen Neidle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 348 KB

english, 1999

2

2,7-Diazabicyclo[3.3.0]octanes as novel h5-HT1D receptor agonists

Michael G.N. Russell, Margaret S. Beer, Josephine A. Stanton, Bindi Sohal, Russell J. Mortishire-Smith, José L. Castro

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 301 KB

english, 1999

3

Structure-related enhancing activity of escins Ia, Ib, IIa and IIb on magnesium absorption in mice

Li Yuhao, Hisashi Matsuda, Suping Wen, Johji Yamahara, Masayuki Yoshikawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 347 KB

english, 1999

4

6-Arylamino-5,8-quinolinediones and 7-arylamino-5,8-isoquinolinediones as inhibitors of endothelium-dependent vasorelaxation

Chung-Kyu Ryu, Sung-Hee Jung, Joung-Ah Lee, Hwa-Jung Kim, Soo-Hwan Lee, Jin-Ho Chung

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 209 KB

english, 1999

5

Fluorobenzamidrazone thrombin inhibitors: Influence of fluorine on enhancing oral absorption

Koo Lee, Won-Hyuk Jung, Sang Yeul Hwang, Sung-Hack Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 231 KB

english, 1999

6

Synthesis and phorbol ester-binding studies of the individual cysteine-rich motifs of protein Kinase D

Kazuhiro Irie, Akifumi Nakahara, Hajime Ohigashi, Hiroyuki Fukuda, Paul A. Wender, Hiroaki Konishi, Ushio Kikkawa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 276 KB

english, 1999

7

Properties of mixed backbone oligonucleotides containing 3′-O-methyl ribonucleosides

Prabhat Kumar, Hiroshi Takaku

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 321 KB

english, 1999

8

Sodium channel activity and sigma binding of 2-aminopropanamide anticonvulsants

Paolo Pevarello, Alberto Bonsignori, Carla Caccia, Raffaella Amici, Robert A. McArthur, Ruggero G. Fariello, Patricia Salvati, Mario Varasi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 263 KB

english, 1999

9

Simple mono-derivatisation of the aryl moiety of D4A and DDA-based phosphoramidate prodrugs significantly enhances their anti-HIV potency in cell culture

Adam Q. Siddiqui, Christopher McGuigan, Carlo Ballatore, Orson Wedgwood, Erik De Clercq, Jan Balzarini

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 338 KB

english, 1999

10

Novel benzo-fused lactam scaffolds as factor Xa inhibitors

Susan Y. Tamura, Erick A. Goldman, Peter W. Bergum, J. Edward Semple

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 356 KB

english, 1999

11

The design of potent and selective inhibitors of thrombin utilizing a piperazinedione template: Part 1

Wayne L. Cody, Cuiman Cai, Annette M. Doherty, Jeremy J. Edmunds, John X. He, Lakshmi S. Narasimhan, Janet S. Plummer, Stephen T. Rapundalo, J. Ronald Rubin, Chad A. Van Huis, Yves St-Denis, Peter D.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 280 KB

english, 1999

12

The design of potent and selective inhibitors of thrombin utilizing a piperazinedione template: Part 2

Wayne L. Cody, Corinne E. Augelli-Szafran, Kent A. Berryman, Cuiman Cai, Annette M. Doherty, Jeremy J. Edmunds, John X. He, Lakshmi S. Narasimhan, Jan Penvose-Yi, Janet S. Plummer, Stephen T. Rapundal

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 257 KB

english, 1999

13

Preparation and receptor binding affinities of cyclic C-terminal neurotensin (8–13) and (9–13) analogues

Joseph T. Lundquist IV, Thomas A. Dix

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 227 KB

english, 1999

14

Aminoisoquinolines: Design and synthesis of an orally active benzamidine isostere for the inhibition of factor XA

Y.M. Choi-Sledeski, M.R. Becker, D.M. Green, R. Davis, W.R. Ewing, H.J. Mason, C. Ly, A. Spada, G. Liang, D. Cheney, J. Barton, V. Chu, K. Brown, D. Colussi, R. Bentley, R. Leadley, C. Dunwiddie, H.W.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 323 KB

english, 1999

15

Versatile fluorescence labeling method using activated esters on solid support

Young-Tae Chang, Peter G. Schultz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 212 KB

english, 1999

16

Acylcarnitine analogues as topical, microbicidal spermicides.

Prashant S. Savle, Gustavo F. Doncel, Stephen D. Bryant, M. Patricia Hubieki, R. Graham Robinette, Richard D. Gandour

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 291 KB

english, 1999

17

A new potent inhibitor of fungal melanin biosynthesis identified through combinatorial chemistry

Lee D. Jennings, Zdzislaw Wawrzak, Denise Amorose, Rand S. Schwartz, Douglas B. Jordan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 298 KB

english, 1999

18

Synthesis and SAR of thioester and thiol inhibitors of IMP-1 Metallo-β-Lactamase

Mark L. Greenlee, Joanne B. Laub, James M. Balkovec, Milton L. Hammond, Gail G. Hammond, David L. Pompliano, Jeffrey H. Epstein-Toney

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 408 KB

english, 1999

19

BN 80927: A novel homocamptothecin with inhibitory activities on both topoisomerase I and topoisomerase II

Olivier Lavergne, Jeremiah Harnett, Alain Rolland, Christophe Lanco, Laurence Lesueur-Ginot, Danièle Demarquay, Marion Huchet, Hélène Coulomb, Dennis C.H. Bigg

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 204 KB

english, 1999

20

Synthesis and antiviral activity of some N-benzenesulphonylbenzimidazoles

Laura Garuti, Marinella Roberti, Claudio Cermelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 268 KB

english, 1999

21

On topography and functionality in the B-D rings of cephalostatin cytotoxins

Thomas G. LaCour, Chuangxing Guo, Sunghoon Ma, Jae Uk Jeong, Michael R. Boyd, Shikegi Matsunaga, Nobuhiro Fusetani, P.L. Fuchs

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 511 KB

english, 1999

22

Dysidiolide and related γ-hydroxy butenolide compounds as inhibitors of the protein tyrosine phosphatase, CDC25

Jill L. Blanchard, David M. Epstein, Michael D. Boisclair, Johannes Rudolph, Kollol Pal

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 118 KB

english, 1999

23

A new class of selective and potent inhibitors of neuronal nitric oxide synthase

John A. Lowe III, Weimin Qian, Robert A. Volkmann, Steven Heck, Jolanta Nowakowski, Robert Nelson, Charles Nolan, Dane Liston, Karen Ward, Stevin Zorn, Celeste Johnson, Michelle Vanase, W. Stephen Far

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 171 KB

english, 1999

24

Synthesis and structure activity relationships of novel small molecule cathepsin D inhibitors

Jacques Dumas, David Brittelli, Jinshan Chen, Brian Dixon, Holia Hatoum-Mokdad, Gerhard König, Robert Sibley, James Witowsky, Stephen Wong

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 327 KB

english, 1999

25

New generation dopaminergic agents. 7. Heterocyclic bioisosteres that exploit the 3-OH-phenoxyethylamine D2 template

Richard E. Mewshaw, James A. Nelson, Uresh S. Shah, Xiaojie Shi, Hossein Mazandarani, Joseph Coupet, Karen Marquis, Julie A. Brennan, Terrance H. Andree

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 248 KB

english, 1999

26

Isoquinoline-6-carboxamides as potent and selective anti-human cytomegalovirus (HCMV) inhibitors

Laval Chan, Haolun Jin, Tomislav Stefanac, Wei Wang, Jean-François Lavallée, Jean Bédard, Suzanne May

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 169 KB

english, 1999

27

Protein kinase C modulators bearing dicarba-closo-dodecaborane as a hydrophobic pharmacophore

Yasuyuki Endo, Tomohiro Yoshimi, Kaname Kimura, Akiko Itai

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 269 KB

english, 1999

28

First synthesis of optically active benzocyclobutene and biphenylene-based unusual α-amino acid derivatives

Sambasivarao Kotha, Nampally Sreenivasachary, Somnath Halder

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 200 KB

english, 1999

29

Fecal excretion pattern of bile acids in rats fed high fat diets and neomycin in induced colon tumorigenesis

Shyamal K. Panda, Selwyn A. Broitman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 266 KB

english, 1999

30

P′-extended α-ketoamide inhibitors of proteasome

Sankar Chatterjee, Derek Dunn, Satish Mallya, Mark A. Ator

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 184 KB

english, 1999

31

Quinoline-2,4-dicarboxylic acids: Synthesis and evaluation as inhibitors of the glutamate vesicular transport system

Christina N. Carrigan, C. Sean Esslinger, Richard D. Bartlett, Richard J. Bridges, Charles M. Thompson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 337 KB

english, 1999

32

The design of (−)-(S)-2-nitrooxyethyl 1,4-dihydro-2,6-dimethyl-3-nitro-4-(2-trifluoromethylphenyl)Pyridine-5-carboxylate: A cardioselective positive inotropic derivative of bay K 8644

Rudong Shan, Edward E. Knaus

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 121 KB

english, 1999

33

Identification and initial structure-activity relationships of a novel non-peptide quinolone GnRH receptor antagonist

Robert J. DeVita, Darius D. Hollings, Mark T. Goulet, Matthew J. Wyvratt, Michael H. Fisher, Jane-L. Lo, Yi Tien Yang, Kang Cheng, Roy G. Smith

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 339 KB

english, 1999

34

Investigation of the 4-O-alkylamine substituent of non-peptide quinolone GnRH receptor antagonists

Robert J. DeVita, Mark T. Goulet, Matthew J. Wyvratt, Michael H. Fisher, Jane-L. Lo, Yi Tien Yang, Kang Cheng, Roy G. Smith

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 233 KB

english, 1999

35

Asymmetric synthesis of novel quaternary α-Hydroxy-δ-lactam dipeptide surrogates

Nathaniel K. Minami, John E. Reiner, J. Edward Semple

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 292 KB

english, 1999

36

Facile synthesis of N-protected γ and δ-Amino-β-Keto-esters

Li Baoqing, Richard W. Franck

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 274 KB

english, 1999

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