Volume 9; Issue 6

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Bioorganic & Medicinal Chemistry Letters
Volume 9; Issue 6

Bioorganic & Medicinal Chemistry Letters

Volume 9; Issue 6

1

Piperidinyl-3-phosphinic acids as novel uptake inhibitors of the neurotransmitter γ-aminobutyric acid (GABA)

Jan Kehler, Tine B. Stensbøl, Povl Krogsgaard-Larsen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 236 KB

english, 1999

2

Synthesis, in vitro cytotoxicity and in vivo anti-inflammatory activity of long chain 3-amino-1,2-diols

JoséM. Padrón, Victor S. Martin, Dimitra Hadjipavlou-Litina, Caterina Noula, Violetta Constantinou-Kokotou, Godefridus J. Peters, George Kokotos

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 299 KB

english, 1999

3

Ring constrained analogues of the orvinols: The furanomorphides

Stephen M. Husbands, Simon W. Breeden, Konstantinos Grivas, John W. Lewis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 223 KB

english, 1999

4

Enantio- and diastereocontrolled dopamine D1, D2, D3 and D4 receptor binding of N-(3-pyrrolidinylmethyl)benzamides synthesized from aspartic acid

Christoph Thomas, Harald Hübner, Peter Gmeiner

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 380 KB

english, 1999

5

Syntheses of two trimannose analogs each containing C-mannosyl or 5-thio-C-mannosyl residue: their affinities to concanavalin A

Osamu Tsuruta, Hideya Yuasa, Sadamu Kurono, Hironobu Hashimoto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 198 KB

english, 1999

6

Cytotoxic effects of NSL-1406, a new thienopyrimidine derivative, on leukocytes and osteoclasts

Jun Katada, Kiyoko Iijima, Michiko Muramatsu, Masamichi Takami, Emiko Yasuda, Miki Hayashi, Mari Hattori, Yoshio Hayashi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 397 KB

english, 1999

7

A new class of anti-HIV agents: Synthesis and activity of conjugates of HIV protease inhibitors with a reverse transcriptase inhibitor

Tooru Kimura, Hikaru Matsumoto, Takashi Matsuda, Tomonori Hamawaki, Kenichi Akaji, Yoshiaki Kiso

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 195 KB

english, 1999

8

Synthesis of novel 4′-C-methyl-pyrimidine nucleosides and their biological activities

Kenji Kitano, Haruhiko Machida, Shinji Miura, Hiroshi Ohrui

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 203 KB

english, 1999

9

Polymer-bound N-hydroxysuccinimide esters: A column-free fluorescent-labeling method

Miho Katoh, Mikiko Sodeoka

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 224 KB

english, 1999

10

Combined NK1 and NK2 tachykinin receptor antagonists: Synthesis and structure-activity relationships of novel oxazolidine analogues

Takahide Nishi, Tetsuya Fukazawa, Koki Ishibashi, Katsuyoshi Nakajima, Yuki Sugioka, Yukiko Iio, Hitoshi Kurata, Kazuhiro Itoh, Osamu Mukaiyama, Yumiko Satoh, Takeshi Yamaguchi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 340 KB

english, 1999

11

Novel reverse-turn mimics inhibit farnesyl transferase

Ruiping Liu, Dennis L.-Y. Dong, Rosemarie Sherlock, H.Peter Nestler, Cesare Gennari, Antonia Mielgo, Carlo Scolastici

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 285 KB

english, 1999

12

Benzenesulfonamide derivatives of 2-substituted 4H-3,1-benzoxazin-4-ones and benzthiazin-4-ones as inhibitors of complement C1r protease

Janet S. Plummer, Cuiman Cai, Sheryl J. Hays, John L. Gilmore, Mark R. Emmerling, Walter Michael, Lakshmi S. Narasimhan, M.Desiree Watson, Kevin Wang, Rathna Nath, Lori M. Evans, Juan C. Jaen

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 286 KB

english, 1999

13

Potent and selective bicyclic lactam inhibitors of thrombin: Part 3: P1′ modifications

Janet S. Plummer, Kent A. Berryman, Cuiman Cai, Wayne L. Cody, John DiMaio, Annette M. Doherty, Scott Eaton, Jeremy J. Edmunds, Debra R. Holland, D. Lafleur, Sophie Levesque, Lakshmi S. Narasimhan, J.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 301 KB

english, 1999

14

Synthesis and activity of γ-(L-γ-azaglutamyl)-S-(p-bromobenzyl)-L-cysteinylglycine: A metabolically stable inhibitor of glyoxalase I

Robert Vince, Jay Brownell, Lakshmi B. Akella

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 180 KB

english, 1999

15

Bicyclo[3.2.1]octanes: Synthesis and inhibition of binding at the dopamine and serotonin transporters

Peter C. Meltzer, Paul Blundell, Zhengming Chen, Yaw F. Yong, Bertha K. Madras

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 305 KB

english, 1999

16

Phosphorothioate oligodeoxyribonucleotides inhibit ribonuclease L thereby disabling a mechanism of interferon action

Mark R. Player, Paul F. Torrence

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 279 KB

english, 1999

17

N,N-Dialkyl-dipeptidylamines as novel N-type calcium channel blockers

Lain-Yen Hu, Todd R Ryder, Michael F Rafferty, Wayne L Cody, Susan M Lotarski, George P Miljanich, Elizabeth Millerman, David M Rock, Yuntao Song, Sally J Stoehr, Charles P Taylor, Mark L Weber, Balaz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 260 KB

english, 1999

18

Design, synthesis, and structure-activity relationship studies of himbacine derived muscarinic receptor antagonists

Darío Doller, Samuel Chackalamannil, Michael Czarniecki, Robert McQuade, Vilma Ruperto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 307 KB

english, 1999

19

Investigation of the S3 site of thrombin: Design, synthesis and biological activity of 4-substituted 3-amino-2-pyridones incorporating P1-argininals

John E. Reiner, Margeurita S. Lim-Wilby, Terence K. Brunck, Theresa Ha-Uong, Erick A. Goldman, Matthew A. Abelman, Ruth F. Nutt, J.Edward Semple, Susan Y. Tamura

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 350 KB

english, 1999

20

Biophysical and biochemical properties of oligodeoxynucleotides containing 4′-C- and 5′-C-substituted thymidines

Guangyi Wang, Patrick J. Middleton, Catherine Lin, Zbigniew Pietrzkowski

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 330 KB

english, 1999

21

Nonpeptide glycoprotein IIB/IIIA inhibitors. 19. A new design paradigm employing linearly minimized, centrally constrained, exosite inhibitors

George D. Hartman, Mark E. Duggan, William F. Hoffman, Robert J. Meissner, James J. Perkins, Amy E. Zartman, Adel M. Naylor-Olsen, Jacquelynn J. Cook, Joan D. Glass, Robert J. Lynch, Guixiang Zhang, R

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 308 KB

english, 1999

22

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 73 KB

english, 1999

23

Graphical abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 328 KB

english, 1999

24

Synthesis and hypoglycemic effect of chrysin derivatives

Joon-Su Shin, Kyoung-Soon Kim, Myoung-Bohm Kim, Jae-Hoon Jeong, Bak-Kwang Kim

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 350 KB

english, 1999

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