Volume 76

Bioorganic Chemistry

Volume 76

1

Structural modeling of osteoarthritis ADAMTS4 complex with its cognate inhibitory protein TIMP3 and rational derivation of cyclic peptide inhibitors from the complex interface to target ADAMTS4

Zhang, Wei, Zhong, Biao, Zhang, Chi, Wang, Yukai, Guo, Shang, Luo, Congfeng, Zhan, Yulin

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 4.97 MB

english, 2018

2

Synthesis of benzo[ d ]imidazo[2,1- b ]thiazole-chalcone conjugates as microtubule targeting and apoptosis inducing agents

Sultana, Faria, Reddy Bonam, Srinivasa, Reddy, V. Ganga, Nayak, V. Lakshma, Akunuri, Ravikumar, Rani Routhu, Sunitha, Alarifi, Abdullah, Halmuthur, M. Sampath Kumar, Kamal, Ahmed

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 2.94 MB

english, 2018

3

Efficient one-pot enzymatic synthesis of dephospho coenzyme A

Sapkota, Krishna, Huang, Faqing

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 704 KB

english, 2018

4

Chemical characterization of cytotoxic indole acetic acid derivative from mulberry fruit ( Morus alba L.) against human cervical cancer

Yu, Jae Sik, Lee, Dahae, Lee, Seoung Rak, Lee, Jae Wook, Choi, Chang-Ik, Jang, Tae Su, Kang, Ki Sung, Kim, Ki Hyun

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.47 MB

english, 2018

5

Improving the carbonic anhydrase inhibition profile of the sulfamoylphenyl pharmacophore by attachment of carbohydrate moieties

Riafrecha, Leonardo E., Bua, Silvia, Supuran, Claudiu T., Colinas, Pedro A.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 359 KB

english, 2018

6

Design, synthesis, anti-inflammatory antitumor activities, molecular modeling and molecular dynamics simulations of potential naprosyn® analogs as COX-1 and/or COX-2 inhibitors

El Sayed, Mardia T., El-Sharief, Marwa A.M.Sh., Zarie, Eman S., Morsy, Nesrin M., Elsheakh, Ahmed R., Nayel, Mohammed, Voronkov, Andrey, Berishvili, Vladimir, Sabry, Nermien M., Hassan, Ghada S., Abde

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.50 MB

english, 2018

7

Biocatalytic hydrolysis of chlorinated nicotinamides by a superior AS family amidase and its application in enzymatic production of 2-chloronicotinic acid

Zheng, Ren-Chao, Jin, Jian-Qiang, Wu, Zhe-Ming, Tang, Xiao-Ling, Jin, Li-Qun, Zheng, Yu-Guo

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.38 MB

english, 2018

8

Design, synthesis and molecular modeling studies of new series of antitumor 1,2,4-triazines with potential c-Met kinase inhibitory activity

El-Wakil, Marwa H., Ashour, Hayam M., Saudi, Manal N., Hassan, Ahmed M., Labouta, Ibrahim M.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.63 MB

english, 2018

9

Azole-hydrazone derivatives: Design, synthesis, in vitro biological evaluation, dual EGFR/HER2 inhibitory activity, cell cycle analysis and molecular docking study as anticancer agents

Labib, Madlen B., Philoppes, John N., Lamie, Phoebe F., Ahmed, Esam R.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 3.70 MB

english, 2018

10

Modification of Bischler-Möhlau indole derivatives through palladium catalyzed Suzuki reaction as effective cholinesterase inhibitors, their kinetic and molecular docking studies

Parveen, Shaista, Shah, Muhammad Shakil, Zaib, Sumera, Gul, Tayyaba, Khan, Khalid Mohammed, Iqbal, Jamshed, Hassan, Abbas

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.95 MB

english, 2018

11

Design, synthesis of novel Triazolones and bis-Triazolones derivatives under ultrasound irradiation and evaluation as potent angiotensin converting enzyme (ACE) inhibitors

Ben Salah, Bochra, Hamzaoui, Salwa, Krichen, Fatma, Saadaoui, Ikram, Ben Mansour, Riadh, Miled, Nabil, Bougatef, Ali, Kossentini, Mohamed

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.65 MB

english, 2018

12

Amino acids/peptides conjugated heterocycles: A tool for the recent development of novel therapeutic agents

Wang, Meng, Rakesh, K.P., Leng, Jing, Fang, Wan-Yin, Ravindar, L., Channe Gowda, D., Qin, Hua-Li

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.59 MB

english, 2018

13

Sulfonamides containing curcumin scaffold: Synthesis, characterization, carbonic anhydrase inhibition and molecular docking studies

Ahmed, Mahmood, Qadir, Muhammad Abdul, Hameed, Abdul, Arshad, Muhammad Nadeem, Asiri, Abdullah M., Muddassar, Muhammad

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.06 MB

english, 2018

14

Design, synthesis and evaluation of resveratrol-indazole hybrids as novel monoamine oxidases inhibitors with amyloid- β aggregation inhibition

Lan, Jin-Shuai, Liu, Yun, Hou, Jian-wei, Yang, Jing, Zhang, Xin-Yu, Zhao, Yuan, Xie, Sai-Sai, Ding, Yue, Zhang, Tong

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.57 MB

english, 2018

15

Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1,4]oxazepine-based carbonic anhydrase inhibitors

Sapegin, Alexander, Kalinin, Stanislav, Angeli, Andrea, Supuran, Claudiu T., Krasavin, Mikhail

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 981 KB

english, 2018

16

Design, synthesis, monoamine oxidase inhibition and docking studies of new dithiocarbamate derivatives bearing benzylamine moiety

Kaya Çavuşoğlu, Betül, Sağlık, Begüm Nurpelin, Özkay, Yusuf, İnci, Beril, Kaplancıklı, Zafer Asım

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.83 MB

english, 2018

17

Synthesis and biological evaluation of new oxopyrrolidine derivatives as inhibitors of acetyl cholinesterase and β amyloid protein as anti – Alzheimer’s agents

Mohamed, Lamia W., Abuel-Maaty, Suzan M., Mohammed, Waleed A., Galal, May A.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 699 KB

english, 2018

18

First evaluation of organotellurium derivatives as carbonic anhydrase I, II, IV, VII and IX inhibitors

Angeli, Andrea, Tanini, Damiano, Capperucci, Antonella, Supuran, Claudiu T.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 517 KB

english, 2018

19

Design, synthesis and evaluation of novel N -hydroxybenzamides/ N -hydroxypropenamides incorporating quinazolin-4(3 H )-ones as histone deacetylase inhibitors and antitumor agents

Hieu, Doan Thanh, Anh, Duong Tien, Tuan, Nguyen Minh, Hai, Pham-The, Huong, Le-Thi-Thu, Kim, Jisung, Kang, Jong Soon, Vu, Tran Khac, Dung, Phan Thi Phuong, Han, Sang-Bae, Nam, Nguyen-Hai, Hoa, Nguyen-

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.43 MB

english, 2018

20

NO inhibitory constituents as potential anti-neuroinflammatory agents for AD from Blumea balsamifera

Ma, Jun, Ren, Quanhui, Dong, Bangjian, Shi, Zhaoyu, Zhang, Jie, Jin, Da-Qing, Xu, Jing, Ohizumi, Yasushi, Lee, Dongho, Guo, Yuanqiang

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.22 MB

english, 2018

21

Aminoadamantanes containing monoterpene-derived fragments as potent tyrosyl-DNA phosphodiesterase 1 inhibitors

Ponomarev, Konstantin Yu., Suslov, Evgeniy V., Zakharenko, Alexandra L., Zakharova, Olga D., Rogachev, Artem D., Korchagina, Dina V., Zafar, Ayesha, Reynisson, Jóhannes, Nefedov, Andrey A., Volcho, Ko

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.24 MB

english, 2018

22

Bioactivity evaluation of natural product α-mangostin as a novel xanthone-based lysine-specific demethylase 1 inhibitor to against tumor metastasis

Han, Chao, Li, Zhongrui, Hou, Jiqin, Wang, Zhen, Xu, Dingqiao, Xue, Guimin, Kong, Lingyi

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.38 MB

english, 2018

23

Synthesis, molecular docking and biological evaluation of some benzimidazole derivatives as potent pancreatic lipase inhibitors

Menteşe, Emre, Yılmaz, Fatih, Emirik, Mustafa, Ülker, Serdar, Kahveci, Bahittin

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 611 KB

english, 2018

24

Bovine Serum Albumin (BSA) coated iron oxide magnetic nanoparticles as biocompatible carriers for curcumin-anticancer drug

Nosrati, Hamed, Sefidi, Naser, Sharafi, Ali, Danafar, Hossein, Kheiri Manjili, Hamidreza

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 2.10 MB

english, 2018

25

Design, synthesis, and biological evaluation of novel substituted benzamide derivatives bearing a 1,2,3-triazole moiety as potent human dihydroorotate dehydrogenase inhibitors

Lu, Kuan, Cai, Lude, Zhang, Xue, Wu, Guodong, Xu, Congjun, Zhao, Yanfang, Gong, Ping

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.36 MB

english, 2018

26

Protonography and anion inhibition profile of the α-carbonic anhydrase (CruCA4) identified in the Mediterranean red coral Corallium rubrum

Del Prete, Sonia, Vullo, Daniela, Caminiti-Segonds, Natacha, Zoccola, Didier, Tambutté, Sylvie, Supuran, Claudiu T., Capasso, Clemente

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.65 MB

english, 2018

27

Synthesis, biological evaluation and molecular docking studies of a new series of chalcones containing naphthalene moiety as anticancer agents

Wang, Guangcheng, Qiu, Jie, Xiao, Xiangwei, Cao, Anbai, Zhou, Fengjiao

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.58 MB

english, 2018

28

Issue TOC

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 4.65 MB

english, 2018

29

Editorial Board

Journal:

Bioorganic Chemistry

Year:

2018

File:

PDF, 39 KB

2018

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