Volume 79

Bioorganic Chemistry

Volume 79

1

Functional group and stereochemical requirements for substrate binding by ghrelin O -acyltransferase revealed by unnatural amino acid incorporation

Cleverdon, Elizabeth R., Davis, Tasha R., Hougland, James L.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.25 MB

english, 2018

2

A novel derivatives of thiazol-4(5 H )-one and their activity in the inhibition of 11β-hydroxysteroid dehydrogenase type 1

Studzińska, Renata, Kołodziejska, Renata, Kupczyk, Daria, Płaziński, Wojciech, Kosmalski, Tomasz

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 855 KB

english, 2018

3

New α-Glucosidase inhibitors from the resins of Boswellia species with structure–glucosidase activity and molecular docking studies

Ur. Rehman, Najeeb, Khan, Ajmal, Al-Harrasi, Ahmed, Hussain, Hidayat, Wadood, Abdul, Riaz, Muhammad, Al-Abri, Zahra

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.31 MB

english, 2018

4

Spiropyrrolidine/spiroindolizino[6,7- b ]indole heterocyclic hybrids: Stereoselective synthesis, cholinesterase inhibitory activity and their molecular docking study

Arumugam, Natarajan, Almansour, Abdulrahman I., Suresh Kumar, Raju, Altaf, Mohammad, Padmanaban, R., Sureshbabu, Popuri, Angamuthu, Gnanavel, Kotresha, D., Manohar, Thota Sai, Venketesh, S.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.66 MB

english, 2018

5

Identification of novel indole based heterocycles as selective estrogen receptor modulator

Singla, Ramit, Prakash, Kunal, Bihari Gupta, Kunj, Upadhyay, Shishir, Dhiman, Monisha, Jaitak, Vikas

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 3.48 MB

english, 2018

6

Steroids from Ganoderma sinense as new natural inhibitors of cancer-associated mutant IDH1

Zheng, Mengzhu, Tang, Ruotian, Deng, Yue, Yang, Kaiyin, Chen, Lixia, Li, Hua

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.84 MB

english, 2018

7

Molecular modelling and synthesis of spiroimidazolidine-2,4-diones with dual activities as hypoglycemic agents and selective inhibitors of aldose reductase

Salem, Manar G., Abdel Aziz, Yasmine M., Elewa, Marwa, Elshihawy, Hosam A., Said, Mohamed M.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 2.04 MB

english, 2018

8

Sophoflavanones A and B, two novel prenylated flavanones from the roots of Sophora flavescens

Zhu, Hui, Yang, Ya-nan, Feng, Zi-ming, Jiang, Jian-shuang, Zhang, Pei-cheng

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 376 KB

english, 2018

9

Novel tetrahydrofuran derivatives from Trigonostemon howii with their potential anti-HIV-1 activities

Liu, Yan-Ping, Zhao, Wan-Hui, Feng, Xing-Yang, Zhang, Zhi-Jie, Zong, Kang, Sun, Zhi-Guo, Zheng, Yong-Tang, Fu, Yan-Hui

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 280 KB

english, 2018

10

Synthesis, biological evaluation and molecular modeling of 2-amino-2-phenylethanol derivatives as novel β 2 -adrenoceptor agonists

Ge, Xinyue, Mo, Yongmei, Xing, Gang, Ji, Lei, Zhao, Haiyan, Chen, Jianfang, He, Bin, Chen, Xuyao, Xing, Ruijuan, Li, Xiaoqiang, Zhao, Ying, Li, Jinyan, Yan, Haining, Woo, Anthony Yiu-Ho, Zhang, Yuyang

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.35 MB

english, 2018

11

Design and synthesis of some new carboxamide and propanamide derivatives bearing phenylpyridazine as a core ring and the investigation of their inhibitory potential on in-vitro acetylcholinesterase and butyrylcholinesterase

Kilic, Burcu, Gulcan, Hayrettin O., Aksakal, Fatma, Ercetin, Tugba, Oruklu, Nihan, Umit Bagriacik, E., Dogruer, Deniz S.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.39 MB

english, 2018

12

Catalytic asymmetric synthesis of indole derivatives as novel α -glucosidase inhibitors in vitro

Islam, Mohammad Shahidul, Barakat, Assem, Al-Majid, Abdullah Mohammed, Ali, M., Yousuf, Sammer, Iqbal Choudhary, M., Khalil, Ruqaiya, Ul-Haq, Zaheer

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.04 MB

english, 2018

13

Fructose furoic acid ester: An effective quorum sensing inhibitor against uropathogenic Escherichia coli

Vinothkannan, Ravichandran, Muthu Tamizh, Manoharan, David Raj, Chellappan, Adline Princy, S.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 2.47 MB

english, 2018

14

Oxidation at C-16 enhances butyrylcholinesterase inhibition in lupane triterpenoids

Castro, María Julia, Richmond, Victoria, Faraoni, María Belén, Murray, Ana Paula

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.29 MB

english, 2018

15

Selenides bearing benzenesulfonamide show potent inhibition activity against carbonic anhydrases from pathogenic bacteria Vibrio cholerae and Burkholderia pseudomallei

Angeli, Andrea, Abbas, Ghulam, del Prete, Sonia, Capasso, Clemente, Supuran, Claudiu T.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 636 KB

english, 2018

16

Drechmerin H, a novel 1(2), 2(18)-di seco indole diterpenoid from the fungus Drechmeria sp. as a natural agonist of human pregnane X receptor

Zhao, Jian-Chao, Luan, Zhi-Lin, Liang, Jia-Hao, Cheng, Zhong-Bin, Sun, Cheng-Peng, Wang, Ya-Li, Zhang, Meng-Yue, Zhang, Tian-Yuan, Wang, Yong, Yang, Tian-Mei, Wu, Ying-Ying, Zhang, Yi-Xuan, Zhao, Xin-

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.03 MB

english, 2018

17

Synthesis, SAR elucidations and molecular docking study of newly designed isatin based oxadiazole analogs as potent inhibitors of thymidine phosphorylase

Javid, Muhammad Tariq, Rahim, Fazal, Taha, Muhammad, Nawaz, Mohsan, Wadood, Abdul, Ali, Muhammad, Mosaddik, Ashik, Shah, Syed Adnan Ali, Farooq, Rai Khalid

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.30 MB

english, 2018

18

Novel γ -lactone derivatives from Trigonostemon heterophyllus with their potential antiproliferative activities

Liu, Yan-Ping, Hu, Shi, Wen, Qing, Ma, Yan-Lei, Jiang, Zhi-Hua, Tang, Jin-Ying, Fu, Yan-Hui

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 319 KB

english, 2018

19

Discovery of potent α-glucosidase inhibitor flavonols: Insights into mechanism of action through inhibition kinetics and docking simulations

Şöhretoğlu, Didem, Sari, Suat, Barut, Burak, Özel, Arzu

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.70 MB

english, 2018

20

Synthesis of aryl pyrazole via Suzuki coupling reaction, in vitro mushroom tyrosinase enzyme inhibition assay and in silico comparative molecular docking analysis with Kojic acid

Channar, Pervaiz Ali, Saeed, Aamer, Larik, Fayaz Ali, Batool, Bakhtawar, Kalsoom, Saima, Hasan, M.M, Erben, Mauricio F., El-Seedi, Hesham R., Ali, Musrat, Ashraf, Zaman

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.15 MB

english, 2018

21

Hit optimization studies of 3-hydroxy-indolin-2-one analogs as potential anti-HIV-1 agents

Chander, Subhash, Tang, Cheng-Run, Penta, Ashok, Wang, Ping, Bhagwat, Deepak P., Vanthuyne, Nicolas, Albalat, Muriel, Patel, Payal, Sankpal, Sanskruti, Zheng, Yong-Tang, Sankaranarayanan, Murugesan

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.31 MB

english, 2018

22

Design and synthesis of aminocoumarin derivatives as DPP-IV inhibitors and anticancer agents

Soni, Rina, Soman, Shubhangi S.

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 876 KB

english, 2018

23

Pyran-2-one derivatives from Croton crassifolius as potent apoptosis inducers in HepG2 cells via p53-mediated Ras/Raf/ERK pathway

Tian, Jin-Long, Yao, Guo-Dong, Zhang, Ying-Ying, Lin, Bin, Zhang, Yan, Li, Ling-Zhi, Huang, Xiao-Xiao, Song, Shao-Jiang

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 2.08 MB

english, 2018

24

New fluorescent rosamine chelator showing promising antibacterial activity against Gram-positive bacteria

Novais, Ângela, Moniz, Tânia, Rebelo, Ana Rita, Silva, Ana M.G., Rangel, Maria, Peixe, Luísa

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 682 KB

english, 2018

25

1-[(4′-Chlorophenyl) carbonyl-4-(aryl) thiosemicarbazide derivatives as potent urease inhibitors: Synthesis, in vitro and in silico studies

Ali, Basharat, Khan, Khalid Mohammed, Salar, Uzma, Kanwal,, Hussain, Safdar, Ashraf, Muhammad, Riaz, Muhammad, Wadood, Abdul, Taha, Muhammad, Perveen, Shahnaz

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 1.29 MB

english, 2018

26

Editorial Board

Journal:

Bioorganic Chemistry

Year:

2018

Language:

english

File:

PDF, 49 KB

english, 2018

27

Issue TOC

Journal:

Bioorganic Chemistry

Year:

2018

File:

PDF, 2.26 MB

2018