Volume 77; Issue 4

Chemical Biology & Drug Design

Volume 77; Issue 4

1

Structural Requirements of Isoquinolones as Novel Selective c-Jun N-terminal Kinase 1 Inhibitors: 2D and 3D QSAR Analyses

Juan Du, Lili Xi, Beilei Lei, Huanxiang Liu, Xiaojun Yao

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 519 KB

english, 2011

2

Issue Information

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 279 KB

english, 2011

3

In Vitro Antifungal and Antibacterial Activities of Pentacycloundecane Tetra-Amines

Oluseye K. Onajole, Yacoob Coovadia, Thavendran Govender, Hendrik G. Kruger, Glenn E. M. Maguire, Dianithi Naidu, Nisha Singh, Patrick Govender

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 103 KB

english, 2011

4

Synthesis and Biological Evaluation of New Quinoxaline Derivatives as Antioxidant and Anti-Inflammatory Agents

Asunción Burguete, Eleni Pontiki, Dimitra Hadjipavlou-Litina, Saioa Ancizu, Raquel Villar, Beatriz Solano, Elsa Moreno, Enrique Torres, Silvia Pérez, Ignacio Aldana, Antonio Monge

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 216 KB

english, 2011

5

Calendar of Events – April 2011

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 16 KB

english, 2011

6

Interaction of a Curcumin Analogue Dimethoxycurcumin with DNA

Amit Kunwar, Emmanuel Simon, Umang Singh, Rajnikant K. Chittela, Deepak Sharma, Santosh K. Sandur, Indira K. Priyadarsini

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 353 KB

english, 2011

7

Ligand-Based 3D-QSAR Studies of Diaryl Acyl-sulfonamide Analogues as Human Umbilical Vein Endothelial Cells Inhibitors Stimulated by VEGF

Zaheer Ul-Haq, Uzma Mahmood, Sualeha Reza, Reaz Uddin, Mehwish Aleem

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 260 KB

english, 2011

8

N-Substituted Glutamyl Sulfonamides as Inhibitors of Glutamate Carboxypeptidase II (GCP2)

Brian R. Blank, Pinar Alayoglu, William Engen, Joseph K. Choi, Clifford E. Berkman, Marc O. Anderson

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 186 KB

english, 2011

9

Rational Design of α-Helical Antimicrobial Peptides to Target Gram-negative Pathogens, Acinetobacter baumannii and Pseudomonas aeruginosa: Utilization of Charge, ‘Specificity Determinants,’ Total Hydrophobicity, Hydrophobe Type and Location as Design Parameters to Improve the Therapeutic Ratio

Ziqing Jiang, Adriana I. Vasil, Lajos Gera, Michael L. Vasil, Robert S. Hodges

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 497 KB

english, 2011

10

Sequential Virtual Screening Approach to the Identification of Small Organic Molecules as Potential BACE-1 Inhibitors

Gianpaolo Chiriano, Andrea Sartini, Francesca Mancini, Vincenza Andrisano, Maria L. Bolognesi, Marinella Roberti, Maurizio Recanatini, Paolo Carloni, Andrea Cavalli

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 316 KB

english, 2011

11

Site-Specific Free Energy Changes in Proteins upon Ligand Binding by Nuclear Magnetic Resonance: Ca2+-Displacement by Ln3+ in a Ca2+-Binding Protein from Entamoeba histolytica

Kousik Chandra, Sourajit M. Mustafi, Subramanian Muthukumar, Kandala V. R. Chary

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 292 KB

english, 2011