Volume 85; Issue 3

Chemical Biology & Drug Design

Volume 85; Issue 3

1

Synthesis and Evaluation of Salicylanilide Derivatives as Potential Epidermal Growth Factor Receptor Inhibitors

Hu, Minhua, Ye, Wenfeng, Li, Jiaming, Zhong, Guochen, He, Guangwei, Xu, Qinlong, Zhang, Yanchun

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 480 KB

english, 2015

2

The Evaluation of Statins as Potential Inhibitors of the LEDGF/p75-HIV-1 Integrase interaction

Harrison, Angela T., Kriel, Frederik H., Papathanasopoulos, Maria A., Mosebi, Salerwe, Abrahams, Shaakira, Hewer, Raymond

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 162 KB

english, 2015

3

Molecular Modeling, Synthesis and Biological Evaluation of N -Heteroaryl Compounds as Reverse Transcriptase Inhibitors Against HIV-1

Singh, Anuradha, Yadav, Dipti, Yadav, Madhu, Dhamanage, Ashwini, Kulkarni, Smita, Singh, Ramendra K.

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 593 KB

english, 2015

4

Structure-activity Relationship Studies of Microbiologically Active Thiosemicarbazides Derived from Hydroxybenzoic Acid Hydrazides

Plech, Tomasz, Paneth, Agata, Kaproń, Barbara, Kosikowska, Urszula, Malm, Anna, Strzelczyk, Aleksandra, Stączek, Paweł

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 1.22 MB

english, 2015

5

Structural and Binding Studies of SAP-1 Protein With Heparin

Yadav, Vikash K., Mandal, Rahul S., Puniya, Bhanwar L., Kumar, Rahul, Dey, Sharmistha, Singh, Sarman, Yadav, Savita

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 1.28 MB

english, 2015

6

Synthesis and Biological Evaluation of Bisphosphonate Compound Labeled with 99m Tc(CO) 3+

Şenocak, Kamile, Teksöz, Serap, İçhedef, Çiğdem, Uçar, Eser

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 236 KB

english, 2015

7

Anticancer Activity and DNA-Binding Investigations of the Cu(II) and Ni(II) Complexes with Coumarin Derivative

Zhu, Taofeng, Wang, Yuan, Ding, Weiliang, Xu, Jun, Chen, Ruhua, Xie, Jing, Zhu, Wenjiao, Jia, Lei, Ma, Tieliang

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 590 KB

english, 2015

8

PEG Mediated Synthesis and Biological Evaluation of Asymmetrical Pyrazole Curcumin Analogues as Potential Analgesic, Anti-Inflammatory and Antioxidant Agents

Jadhav, Shravan Y., Bhosale, Raghunath B., Shirame, Sachin P., Patil, Sandeep B., Kulkarni, Suresh D.

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 185 KB

english, 2015

9

Design, Synthesis, and Preliminary Activity Evaluation of Novel Pyrimidine Derivatives as Acid Pump Antagonists

Song, Weiguo, Zhang, Xiaopan, Li, Shutao, Xu, Wenfang

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 750 KB

english, 2015

10

Synthesis, Biological Evaluation, and Molecular Docking Studies of Xanthone Sulfonamides as ACAT Inhibitors

Li, Xiang, Zou, Yan, Zhao, Qingjie, Yang, Yan, Wu, Maocheng, Huang, Ting, Hu, Honggang, Wu, Qiuye

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 950 KB

english, 2015

11

Up Regulation of Liver-enriched Transcription Factors HNF4a and HNF6 and Liver-Specific MicroRNA (miR-122) by Inhibition of Let-7b in Mesenchymal Stem Cells

Alizadeh, Effat, Akbarzadeh, Abolfazl, Eslaminejad, Mohamadreza Baghaban, Barzegar, Abolfazl, Hashemzadeh, Shahryar, Nejati-Koshki, Kazem, Zarghami, Nosratollah

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 2.51 MB

english, 2015

12

Zebrafish as a New Model for Phenotype-based Screening of Positive Inotropic Agents

Tang, Chunlei, Xie, Desheng, Feng, Bainian

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 900 KB

english, 2015

13

Feleucin-BO1: A Novel Antimicrobial Non-Apeptide Amide from the Skin Secretion of the Toad, Bombina orientalis, and Design of a Potent Broad-Spectrum Synthetic Analogue, Feleucin-K3

Hou, Xiaojuan, Du, Qiang, Li, Renjie, Zhou, Mei, Wang, Hui, Wang, Lei, Guo, Can, Chen, Tianbao, Shaw, Chris

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 779 KB

english, 2015

14

Strong Inhibition of Beta-Amyloid Peptide Aggregation Realized by Two-Steps Evolved Peptides

Ghimire Gautam, Sunita, Komatsu, Masayuki, Nishigaki, Koichi

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 1.71 MB

english, 2015

15

Synthesis and Biological Evaluation of 2-oxo-pyrazine-3-carboxamide-yl Nucleoside Analogues and Their Epimers as Inhibitors of Influenza A Viruses

Gao, Jingjing, Luo, Xianjin, Li, Yuhuan, Gao, Rongmei, Chen, Haifeng, Ji, Dingjue

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 751 KB

english, 2015

16

Synthesis and Evaluation of Antidepressant-like Activity of Some 4-Substituted 1-(2-methoxyphenyl)Piperazine Derivatives

Waszkielewicz, Anna M., Pytka, Karolina, Rapacz, Anna, Wełna, Elżbieta, Jarzyna, Monika, Satała, Grzegorz, Bojarski, Andrzej, Sapa, Jacek, Żmudzki, Paweł, Filipek, Barbara, Marona, Henryk

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 660 KB

english, 2015

17

Synthesis and Biological Evaluation of 5-Nitropyrimidine-2,4-dione Analogues as Inhibitors of Nitric Oxide and iNOS Activity

Ma, Liang, He, Linhong, Lei, Lei, Liang, Xiaolin, Lei, Kai, Zhang, Ronghong, Yang, Zhuang, Chen, Lijuan

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 447 KB

english, 2015

18

Highly Stable, Fluorescence-Labeled Heptapeptides Substituted with a D-Amino Acid for the Specific Detection of Oxidized Low-Density Lipoprotein in Plasma

Sato, Akira, Yamanaka, Hikaru, Oe, Keitaro, Yokoyama, Izumi, Yamazaki, Yoji, Ebina, Keiichi

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 767 KB

english, 2015

19

Issue Information

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 998 KB

english, 2015

20

Microwave-assisted Synthesis of Cyclic Phosphopeptide on Solid Support

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 561 KB

english, 2015