Volume 85; Issue 5

Chemical Biology & Drug Design

Volume 85; Issue 5

1

Evaluation of Anti-inflammatory and Analgesic Effects of Synthesized Derivatives of Ibuprofen

Wang, Jingjie, Dai, Dongyan, Qiu, Qianqian, Deng, Xin, Lin, Haiyan, Qian, Hai, Huang, Wenlong

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 458 KB

english, 2015

2

Plant-Derived Flavones as Inhibitors of Aurora B Kinase and Their Quantitative Structure-Activity Relationships

Jung, Yearam, Shin, Soon Young, Yong, Yeonjoong, Jung, Hyeryoung, Ahn, Seunghyun, Lee, Young Han, Lim, Yoongho

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 586 KB

english, 2015

3

Design, Synthesis and Pharmacological Evaluation of Novel NO-Releasing Benzimidazole Hybrids as Potential Antihypertensive Candidate

Zhang, Yanchun, Xu, Jinyi, Li, Yunman, Yao, Hequan, Wu, Xiaoming

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 462 KB

english, 2015

4

Carboxylated Hydroxyethyl Starch: A novel Polysaccharide for the Delivery of Doxorubicin

Paleos, Constantinos M., Sideratou, Zili, Theodossiou, Theodossis A., Tsiourvas, Dimitris

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 544 KB

english, 2015

5

Targeting Receptor Tyrosine Kinases and Their Downstream Signaling with Cell-Penetrating Peptides in Human Pulmonary Artery Smooth Muscle and Endothelial Cells

Yu, Jun, Rupasinghe, Chamila, Wilson, Jamie L., Taylor, Linda, Rahimi, Nader, Mierke, Dale, Polgar, Peter

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 1.68 MB

english, 2015

6

Synthesis and Antitumor Activity of Natural Compound Aloe Emodin Derivatives

Thimmegowda, Naraganahalli R., Park, Chanmi, Shwetha, Bettaswamigowda, Sakchaisri, Krisada, Liu, Kangdong, Hwang, Joonsung, Lee, Sangku, Jeong, Sook J., Soung, Nak K., Jang, Jae H., Ryoo, In-Ja, Ahn,

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 1.48 MB

english, 2015

7

4-Substituted-1-phenyl-1 H -pyrazolo[3,4- d ]pyrimidine Derivatives: Design, Synthesis, Antitumor and EGFR Tyrosine Kinase Inhibitory Activity

Abbas, Safinaz E.-S., Aly, Enayat I., Awadallah, Fadi M., Mahmoud, Walaa R.

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 1.26 MB

english, 2015

8

Biofilm Eradication Kinetics of the Ultrashort Lipopeptide C 12 -OOWW-NH 2 Utilizing a Modified MBEC Assay ™

Laverty, Garry, Gorman, Sean P., Gilmore, Brendan F.

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 907 KB

english, 2015

9

Repurposing Human PDE4 Inhibitors for Neglected Tropical Diseases. Evaluation of Analogs of the Human PDE4 Inhibitor GSK-256066 as Inhibitors of PDEB1 of Trypanosoma brucei

Ochiana, Stefan O., Bland, Nicholas D., Settimo, Luca, Campbell, Robert K., Pollastri, Michael P.

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 4.48 MB

english, 2015

10

Design, Synthesis, and Cercaricidal Activity of Novel High-efficient, Low-toxic Self-spreading PEG- N -salicylanilide Derivatives Against Cercariae Larvae of Schistosome Japonicum Floating on the Water Surface

Guo, Wei, Zheng, Lv-Yin, Wu, Ren-Miao, Fan, Xiao-Lin

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 984 KB

english, 2015

11

Hydrogen-Bonded His93 As a Sensitive Probe for Identifying Inhibitors of the Endocannabinoid Transport Protein FABP7

Tyukhtenko, Sergiy, Chan, Karrie, Jiang, Rubin, Zhou, Han, Mercier, Richard W., Yang, De-Ping, Makriyannis, Alexandros, Guo, Jason J.

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 755 KB

english, 2015

12

Development of Peptidyl Lysine Dendrons: 1,3-Dipolar Cycloaddition for Peptide Coupling and Antibody Recognition

Hüttl, Christine, Hettrich, Cornelia, Riedel, Melanie, Henklein, Petra, Rawel, Harshadrai, Bier, Frank F.

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 680 KB

english, 2015

13

Production of an Antimicrobial Peptide AN5-1 in Escherichia coli and its Dual Mechanisms Against Bacteria

Yi, Tonghui, Huang, Yibing, Chen, Yuxin

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 1.15 MB

english, 2015

14

A Cisplatin Derivative that Inhibits Collagen Fibril-Formation in vitro

Zenda, Miyu, Yasui, Hiroyuki, Oishi, Shinya, Masuda, Ryo, Fujii, Nobutaka, Koide, Takaki

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 1.17 MB

english, 2015

15

Functional Non-Nucleoside Adenylyl Cyclase Inhibitors

Lelle, Marco, Hameed, Abdul, Ackermann, Lisa-Maria, Kaloyanova, Stefka, Wagner, Manfred, Berisha, Filip, Nikolaev, Viacheslav O., Peneva, Kalina

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 447 KB

english, 2015

16

Issue Information

Journal:

Chemical Biology & Drug Design

Year:

2015

Language:

english

File:

PDF, 191 KB

english, 2015