Volume 11; Issue 1

Main
ChemMedChem
Volume 11; Issue 1

ChemMedChem

Volume 11; Issue 1

1

Design, Synthesis and Evaluation of Triazole-Pyrimidine Analogues as SecA Inhibitors

Cui, Jianmei, Jin, Jinshan, Chaudhary, Arpana Sagwal, Hsieh, Ying-hsin, Zhang, Hao, Dai, Chaofeng, Damera, Krishna, Chen, Weixuan, Tai, Phang C., Wang, Binghe

Journal:

Year:

2016

Language:

english

File:

PDF, 1.76 MB

english, 2016

2

Optimization of Inhibitors of Mycobacterium tuberculosis Pantothenate Synthetase Based on Group Efficiency Analysis

Hung, Alvin W., Silvestre, H. Leonardo, Wen, Shijun, George, Guillaume P. C., Boland, Jennifer, Blundell, Tom L., Ciulli, Alessio, Abell, Chris

Journal:

Year:

2016

Language:

english

File:

PDF, 2.05 MB

english, 2016

3

N -Alkyl-, 1- C -Alkyl-, and 5- C -Alkyl-1,5-dideoxy-1,5-imino-( l )-ribitols as Galactosidase Inhibitors

Front, Sophie, Gallienne, Estelle, Charollais-Thoenig, Julie, Demotz, Stéphane, Martin, Olivier R.

Journal:

Year:

2016

Language:

english

File:

PDF, 578 KB

english, 2016

4

Discovery of 3-Hydroxy-3-phenacyloxindole Analogues of Isatin as Potential Monoamine Oxidase Inhibitors

Tripathi, Rati K. P., Krishnamurthy, Sairam, Ayyannan, Senthil R.

Journal:

Year:

2016

Language:

english

File:

PDF, 3.41 MB

english, 2016

5

Why Hydroxamates May Not Be the Best Histone Deacetylase Inhibitors-What Some May Have Forgotten or Would Rather Forget?

Shen, Sida, Kozikowski, Alan P.

Journal:

Year:

2016

Language:

english

File:

PDF, 1.78 MB

english, 2016

6

Epigenetics: Current Research and Emerging Trends. Edited by Brian P. Chadwick

Journal:

Year:

2016

Language:

english

File:

PDF, 175 KB

english, 2016

7

Stereoselective Modulation of P-Glycoprotein by Chiral Small Molecules

Carocci, Alessia, Catalano, Alessia, Turi, Francesco, Lovece, Angelo, Cavalluzzi, Maria M., Bruno, Claudio, Colabufo, Nicola A., Contino, Marialessandra, Perrone, Maria G., Franchini, Carlo, Lentini,

Journal:

Year:

2016

Language:

english

File:

PDF, 522 KB

english, 2016

8

11 C- and 18 F-Labeled Radioligands for P-Glycoprotein Imaging by Positron Emission Tomography

Cantore, Mariangela, Benadiba, Marcel, Elsinga, Philip H., Kwizera, Chantal, Dierckx, Rudi A. J. O., Colabufo, Nicola Antonio, Luurtsema, Gert

Journal:

Year:

2016

Language:

english

File:

PDF, 1.33 MB

english, 2016

9

Structure-Activity Relationship Studies of Amino Acid Substitutions in Radiolabeled Neurotensin Conjugates

Mascarin, Alba, Valverde, Ibai E., Mindt, Thomas L.

Journal:

Year:

2016

Language:

english

File:

PDF, 1.14 MB

english, 2016

10

Photoinduced Isomerization and Hepatoxicities of Semaxanib, Sunitinib and Related 3-Substituted Indolin-2-ones

Ngai, Mun Hong, So, Choon Leng, Sullivan, Michael B., Ho, Han Kiat, Chai, Christina L. L.

Journal:

Year:

2016

Language:

english

File:

PDF, 510 KB

english, 2016

11

Inspired by Nature: The 3-Halo-4,5-dihydroisoxazole Moiety as a Novel Molecular Warhead for the Design of Covalent Inhibitors

Pinto, Andrea, Tamborini, Lucia, Cullia, Gregorio, Conti, Paola, De Micheli, Carlo

Journal:

Year:

2016

Language:

english

File:

PDF, 516 KB

english, 2016

12

Synthesis and Biopharmaceutical Evaluation of Imatinib Analogues Featuring Unusual Structural Motifs

Nicolaou, Kyriacos C., Vourloumis, Dionisios, Totokotsopoulos, Sotirios, Papakyriakou, Athanasios, Karsunky, Holger, Fernando, Hanan, Gavrilyuk, Julia, Webb, Damien, Stepan, Antonia F.

Journal:

Year:

2016

Language:

english

File:

PDF, 2.18 MB

english, 2016

13

Drug Discovery for Schizophrenia. Edited by Tatiana V. Lipina and John C. Roder

Cavallaro, Roberto

Journal:

Year:

2016

Language:

english

File:

PDF, 313 KB

english, 2016

14

A Decade of ChemMedChem

Williams, Scott D., Ortúzar, Natalia

Journal:

Year:

2016

Language:

english

File:

PDF, 718 KB

english, 2016

15

Drug Metabolism Prediction . Edited by Johannes Kirchmair

Journal:

Year:

2016

Language:

english

File:

PDF, 355 KB

english, 2016

16

Cover Picture: How Consistent are Publicly Reported Cytotoxicity Data? Large-Scale Statistical Analysis of the Concordance of Public Independent Cytotoxicity Measurements (ChemMedChem 1/2016)

Cortés-Ciriano, Isidro, Bender, Andreas

Journal:

Year:

2016

File:

PDF, 406 KB

2016

17

Inside Cover: Structure-Activity Relationship Studies of Amino Acid Substitutions in Radiolabeled Neurotensin Conjugates (ChemMedChem 1/2016)

Mascarin, Alba, Valverde, Ibai E., Mindt, Thomas L.

Journal:

Year:

2016

File:

PDF, 845 KB

2016

18

Back Cover: Photoinduced Isomerization and Hepatoxicities of Semaxanib, Sunitinib and Related 3-Substituted Indolin-2-ones (ChemMedChem 1/2016)

Ngai, Mun Hong, So, Choon Leng, Sullivan, Michael B., Ho, Han Kiat, Chai, Christina L. L.

Journal:

Year:

2016

File:

PDF, 1.46 MB

2016

19

Spotlights on our sister journals: ChemMedChem 1/2016

Journal:

Year:

2016

Language:

english

File:

PDF, 2.82 MB

english, 2016

20

How Consistent are Publicly Reported Cytotoxicity Data? Large-Scale Statistical Analysis of the Concordance of Public Independent Cytotoxicity Measurements

Cortés-Ciriano, Isidro, Bender, Andreas

Journal:

Year:

2016

Language:

english

File:

PDF, 5.33 MB

english, 2016

21

Identification of HDAC6-Selective Inhibitors of Low Cancer Cell Cytotoxicity

Gaisina, Irina N., Tueckmantel, Werner, Ugolkov, Andrey, Shen, Sida, Hoffen, Jessica, Dubrovskyi, Oleksii, Mazar, Andrew, Schoon, Renee A., Billadeau, Daniel, Kozikowski, Alan P.

Journal:

Year:

2016

Language:

english

File:

PDF, 1.31 MB

english, 2016

22

Designing Irreversible Inhibitors-Worth the Effort?

González-Bello, Concepción

Journal:

Year:

2016

Language:

english

File:

PDF, 3.85 MB

english, 2016