Volume 11; Issue 4

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ChemMedChem
Volume 11; Issue 4

ChemMedChem

Volume 11; Issue 4

1

New Insight into the Structure-Activity Relationships of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitors UCPH-101 and UCPH-102

Hansen, Stinne W., Erichsen, Mette N., Huynh, Tri H. V., Ruiz, Josep A., Haym, Isabell, Bjørn-Yoshimoto, Walden E., Abrahamsen, Bjarke, Hansen, Jeanette, Storgaard, Morten, Eriksen, Anette L., Jensen,

Journal:

Year:

2016

Language:

english

File:

PDF, 1.66 MB

english, 2016

2

Application of Site-Specific Spin Labeling for NMR Detecting Inhibitor-Induced Conformational Change of HIV-1 Reverse Transcriptase

Seetaha, Supaporn, Yagi-Utsumi, Maho, Yamaguchi, Takumi, Ishii, Kentaro, Hannongbua, Supa, Choowongkomon, Kiattawee, Kato, Koichi

Journal:

Year:

2016

Language:

english

File:

PDF, 907 KB

english, 2016

3

Bioavailability Studies and in vitro Profiling of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitor UCPH-102

Haym, Isabell, Huynh, Tri H. V., Hansen, Stinne W., Pedersen, Martin H. F., Ruiz, Josep A., Erichsen, Mette N., Gynther, Mikko, Bjørn-Yoshimoto, Walden E., Abrahamsen, Bjarke, Bastlund, Jesper F., Bun

Journal:

Year:

2016

Language:

english

File:

PDF, 834 KB

english, 2016

4

Broadly Neutralizing Antibody-Guided Carbohydrate-Based HIV Vaccine Design: Challenges and Opportunities

Liu, Chang-Cheng, Zheng, Xiu-Jing, Ye, Xin-Shan

Journal:

Year:

2016

Language:

english

File:

PDF, 511 KB

english, 2016

5

EPR Studies of V-ATPase with Spin-Labeled Inhibitors DCC and Archazolid: Interaction Dynamics with Proton Translocating Subunit c

Gölz, Jan Philipp, Bockelmann, Svenja, Mayer, Kerstin, Steinhoff, Heinz-Jürgen, Wieczorek, Helmut, Huss, Markus, Klare, Johann P., Menche, Dirk

Journal:

Year:

2016

Language:

english

File:

PDF, 2.33 MB

english, 2016

6

A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression

Guglielmo, Stefano, Contino, Marialessandra, Lazzarato, Loretta, Perrone, Maria Grazia, Blangetti, Marco, Fruttero, Roberta, Colabufo, Nicola Antonio

Journal:

Year:

2016

Language:

english

File:

PDF, 563 KB

english, 2016

7

Screening, Synthesis, and In Vitro Evaluation of Vinyl Sulfones as Inhibitors of Complement-Dependent Cytotoxicity in Neuromyelitis Optica

Ju, Eun Ji, Yeon, Seul Ki, Park, Jong-Hyun, Cheon, So Young, Choi, Ji Won, Ha, Taehwan, Jang, Bo Ko, Kim, Siwon, Kang, Yong Gu, Hwang, Hayoung, Cho, Sung Jin, Cheong, Eunji, Bahn, Yong Sun, Pae, Ae Ni

Journal:

Year:

2016

Language:

english

File:

PDF, 913 KB

english, 2016

8

Spotlights on our sister journals: ChemMedChem 4/2016

Journal:

Year:

2016

Language:

english

File:

PDF, 2.83 MB

english, 2016

9

ω-Imidazolyl- and ω-Tetrazolylalkylcarbamates as Inhibitors of Fatty Acid Amide Hydrolase: Biological Activity and in vitro Metabolic Stability

Terwege, Tobias, Hanekamp, Walburga, Garzinsky, David, König, Simone, Koch, Oliver, Lehr, Matthias

Journal:

Year:

2016

Language:

english

File:

PDF, 2.13 MB

english, 2016

10

Antivirulence Isoquinolone Mannosides: Optimization of the Biaryl Aglycone for FimH Lectin Binding Affinity and Efficacy in the Treatment of Chronic UTI

Jarvis, Cassie, Han, Zhenfu, Kalas, Vasilios, Klein, Roger, Pinkner, Jerome S., Ford, Bradley, Binkley, Jana, Cusumano, Corinne K., Cusumano, Zachary, Mydock-McGrane, Laurel, Hultgren, Scott J., Janet

Journal:

Year:

2016

Language:

english

File:

PDF, 1.16 MB

english, 2016

11

Cover Picture: Antivirulence Isoquinolone Mannosides: Optimization of the Biaryl Aglycone for FimH Lectin Binding Affinity and Efficacy in the Treatment of Chronic UTI (ChemMedChem 4/2016)

Jarvis, Cassie, Han, Zhenfu, Kalas, Vasilios, Klein, Roger, Pinkner, Jerome S., Ford, Bradley, Binkley, Jana, Cusumano, Corinne K., Cusumano, Zachary, Mydock-McGrane, Laurel, Hultgren, Scott J., Janet

Journal:

Year:

2016

File:

PDF, 375 KB

2016

12

Inside Cover: Screening, Synthesis, and In Vitro Evaluation of Vinyl Sulfones as Inhibitors of Complement-Dependent Cytotoxicity in Neuromyelitis Optica (ChemMedChem 4/2016)

Ju, Eun Ji, Yeon, Seul Ki, Park, Jong-Hyun, Cheon, So Young, Choi, Ji Won, Ha, Taehwan, Jang, Bo Ko, Kim, Siwon, Kang, Yong Gu, Hwang, Hayoung, Cho, Sung Jin, Cheong, Eunji, Bahn, Yong Sun, Pae, Ae Ni

Journal:

Year:

2016

File:

PDF, 1014 KB

2016

13

Back Cover: EPR Studies of V-ATPase with Spin-Labeled Inhibitors DCC and Archazolid: Interaction Dynamics with Proton Translocating Subunit c (ChemMedChem 4/2016)

Gölz, Jan Philipp, Bockelmann, Svenja, Mayer, Kerstin, Steinhoff, Heinz-Jürgen, Wieczorek, Helmut, Huss, Markus, Klare, Johann P., Menche, Dirk

Journal:

Year:

2016

File:

PDF, 1.52 MB

2016