Volume 2; Issue 1

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ChemMedChem
Volume 2; Issue 1

ChemMedChem

Volume 2; Issue 1

1

Benzo[d]isothiazol-3-yl-benzamidines: a Class of Protective Agents on Culture of Human Cartilage and Chondrocytes Stimulated by IL-1β

Paola Vicini, Matteo Incerti, Venera Cardile, Floriana Garufi, Simone Ronsisvalle, Anna Maria Panico

Journal:

Year:

2007

Language:

english

File:

PDF, 115 KB

english, 2007

2

The Importance of the Active Site Histidine for the Activity of Epoxide- or Aziridine-Based Inhibitors of Cysteine Proteases

Milena Mladenovic, Tanja Schirmeister, Stefan Thiel, Walter Thiel, Bernd Engels

Journal:

Year:

2007

Language:

english

File:

PDF, 670 KB

english, 2007

3

Topical Delivery of Silver Nanoparticles Promotes Wound Healing

Jun Tian, Kenneth K. Y. Wong, Chi-Ming Ho, Chun-Nam Lok, Wing-Yiu Yu, Chi-Ming Che, Jen-Fu Chiu, Paul K. H. Tam

Journal:

Year:

2007

Language:

english

File:

PDF, 661 KB

english, 2007

4

Advances towards the Development of ATP-Competitive Small-Molecule Inhibitors of the Insulin-Like Growth Factor Receptor (IGF-IR)

Robert D. Hubbard, Julie L. Wilsbacher

Journal:

Year:

2007

Language:

english

File:

PDF, 319 KB

english, 2007

5

Design, Syntheses, Biological Evaluation, and Docking Studies of 2-Substituted 5-Methylsulfonyl-1-Phenyl-1H-Indoles: Potent and Selective in vitro Cyclooxygenase-2 Inhibitors

Olga Cruz-López, Juan José Díaz-Mochón, Joaquín M. Campos, Antonio Entrena, María T. Núñez, Luis Labeaga, Aurelio Orjales, Miguel A. Gallo, Antonio Espinosa

Journal:

Year:

2007

Language:

english

File:

PDF, 509 KB

english, 2007

6

Ligand-Based Vascular Targeting of Disease

Jascha-N. Rybak, Eveline Trachsel, Jörg Scheuermann, Dario Neri

Journal:

Year:

2007

Language:

english

File:

PDF, 942 KB

english, 2007

7

Nanomolar Inhibition of Type II Dehydroquinase Based on the Enolate Reaction Mechanism

Miguel D. Toscano, Richard J. Payne, Akira Chiba, Olivier Kerbarh, Chris Abell

Journal:

Year:

2007

Language:

english

File:

PDF, 276 KB

english, 2007

8

Macrocyclic Aminopyrimidines as Multitarget CDK and VEGF-R Inhibitors with Potent Antiproliferative Activities

Ulrich Lücking, Gerhard Siemeister, Martina Schäfer, Hans Briem, Martin Krüger, Philip Lienau, Rolf Jautelat

Journal:

Year:

2007

Language:

english

File:

PDF, 422 KB

english, 2007

9

Simulating α/β Selectivity at the Human Thyroid Hormone Receptor: Consensus Scoring Using Multidimensional QSAR

Angelo Vedani, Martin Zumstein, Markus A. Lill, Beat Ernst

Journal:

Year:

2007

Language:

english

File:

PDF, 673 KB

english, 2007

10

Acetylenic Pyridines for Use in PET Imaging of Nicotinic Receptors

Alan P. Kozikowski, Sheela K. Chellappan, David Henderson, Roger Fulton, Nicolas Giboureau, Yingxian Xiao, Zhi-Liang Wei, Denis Guilloteau, Patrick Emond, Frederic Dolle, Kenneth J. Kellar, Michael Ka

Journal:

Year:

2007

Language:

english

File:

PDF, 114 KB

english, 2007

11

Discovery of Selective Irreversible Inhibitors for Bruton’s Tyrosine Kinase

Zhengying Pan, Heleen Scheerens, Shyr-Jiann Li, Brian E. Schultz, Paul A. Sprengeler, L. Chuck Burrill, Rohan V. Mendonca, Michael D. Sweeney, Keana C. K. Scott, Paul G. Grothaus, Douglas A. Jeffery,

Journal:

Year:

2007

Language:

english

File:

PDF, 242 KB

english, 2007

12

A Soluble Amyloid Fibril Segment to Study Aggregate Formation

Journal:

Year:

2007

Language:

english

File:

PDF, 70 KB

english, 2007

13

The Anionic Boron Cluster (B12H11SH)2− as a Means To Trigger Release of Liposome Contents

Detlef Gabel, Doaa Awad, Tanja Schaffran, Diana Radovan, Daniel Dărăban, Luminita Damian, Mathias Winterhalter, Göran Karlsson, Katarina Edwards

Journal:

Year:

2007

Language:

english

File:

PDF, 200 KB

english, 2007

14

Anniversaries Old and New

Scott D. Williams

Journal:

Year:

2007

Language:

english

File:

PDF, 713 KB

english, 2007

15

Cover Picture: Simulating α/β Selectivity at the Human Thyroid Hormone Receptor: Consensus Scoring Using Multidimensional QSAR (ChemMedChem 1/2007)

Angelo Vedani, Martin Zumstein, Markus A. Lill, Beat Ernst

Journal:

Year:

2007

File:

PDF, 35 KB

2007

16

Preview: ChemMedChem 2/2007

Journal:

Year:

2007

Language:

english

File:

PDF, 31 KB

english, 2007

17

From our sister journals: ChemMedChem 1/2007

Journal:

Year:

2007

Language:

english

File:

PDF, 300 KB

english, 2007

18

Graphical Abstract: ChemMedChem 1/2007

Journal:

Year:

2007

Language:

english

File:

PDF, 688 KB

english, 2007