Volume 2; Issue 5

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ChemMedChem
Volume 2; Issue 5

ChemMedChem

Volume 2; Issue 5

1

Fluoroartemisinins: Metabolically More Stable Antimalarial Artemisinin Derivatives

Jean-Pierre Bégué, Danièle Bonnet-Delpon

Journal:

Year:

2007

Language:

english

File:

PDF, 819 KB

english, 2007

2

Chemical Tools to Investigate Sphingolipid Metabolism and Functions

Antonio Delgado, Josefina Casas, Amadeu Llebaria, José Luis Abad, Gemma Fabriás

Journal:

Year:

2007

Language:

english

File:

PDF, 917 KB

english, 2007

3

ESI–MS Characterisation of Protein Adducts of Anticancer Ruthenium(II)-Arene PTA (RAPTA) Complexes

Angela Casini, Guido Mastrobuoni, Wee Han Ang, Chiara Gabbiani, Giuseppe Pieraccini, Gloriano Moneti, Paul J. Dyson, Luigi Messori

Journal:

Year:

2007

Language:

english

File:

PDF, 163 KB

english, 2007

4

Highly Potent Fluorescence-Tagged Nonimidazole Histamine H3 Receptor Ligands

Michael Amon, Xavier Ligneau, Jean-Claude Camelin, Isabelle Berrebi-Bertrand, Jean-Charles Schwartz, Holger Stark

Journal:

Year:

2007

Language:

english

File:

PDF, 178 KB

english, 2007

5

Development of a Method for the Quantification of the Molar Gold Concentration in Tumour Cells Exposed to Gold-Containing Drugs

Ingo Ott, Heike Scheffler, Ronald Gust

Journal:

Year:

2007

Language:

english

File:

PDF, 165 KB

english, 2007

6

α-Substituted Phosphonate Analogues of Lysophosphatidic Acid (LPA) Selectively Inhibit Production and Action of LPA

Guowei Jiang, Yong Xu, Yuko Fujiwara, Tamotsu Tsukahara, Ryoko Tsukahara, Joanna Gajewiak, Gabor Tigyi, Glenn D. Prestwich

Journal:

Year:

2007

Language:

english

File:

PDF, 233 KB

english, 2007

7

G-Quadruplex Recognition by Quinacridines: a SAR, NMR, and Biological Study

Candide Hounsou, Lionel Guittat, David Monchaud, Muriel Jourdan, Nicolas Saettel, Jean-Louis Mergny, Marie-Paule Teulade-Fichou

Journal:

Year:

2007

Language:

english

File:

PDF, 516 KB

english, 2007

8

Selective Inhibition of c-Myc/Max Dimerization by a Pyrazolo[1,5-a]pyrimidine

Anke Kiessling, Rita Wiesinger, Bianca Sperl, Thorsten Berg

Journal:

Year:

2007

Language:

english

File:

PDF, 257 KB

english, 2007

9

Fluorescent Probes for Rapid Screening of Potential Drug–Drug Interactions at the CYP3A4 Level

Antoinette Chougnet, Yelena Grinkova, David Ricard, Stephen Sligar, Wolf-D. Woggon

Journal:

Year:

2007

Language:

english

File:

PDF, 250 KB

english, 2007

10

Synthesis, Biological Evaluation, and Molecular Modeling Investigation of Chiral Phenoxyacetic Acid Analogues with PPARα and PPARγ Agonist Activity

Giuseppe Fracchiolla, Antonio Laghezza, Luca Piemontese, Giuseppe Carbonara, Antonio Lavecchia, Paolo Tortorella, Maurizio Crestani, Ettore Novellino, Fulvio Loiodice

Journal:

Year:

2007

Language:

english

File:

PDF, 705 KB

english, 2007

11

Opening Ion Channels: Enzyme at the Gate

Jun Chen, Murali Gopalakrishnan

Journal:

Year:

2007

Language:

english

File:

PDF, 98 KB

english, 2007

12

Ensemble-Docking Approach on BACE-1: Pharmacophore Perception and Guidelines for Drug Design

Vittorio Limongelli, Luciana Marinelli, Sandro Cosconati, Hannes A. Braun, Boris Schmidt, Ettore Novellino

Journal:

Year:

2007

Language:

english

File:

PDF, 803 KB

english, 2007

13

Overcoming Tumor Drug Resistance with High-Affinity Taxanes: A SAR Study of C2-Modified 7-Acyl-10-Deacetyl Cephalomannines

Chun-Gang Yang, Isabel Barasoain, Xuan Li, Ruth Matesanz, Ronghua Liu, Frances J. Sharom, Da-Li Yin, J. Fernando Díaz, Wei-Shuo Fang

Journal:

Year:

2007

Language:

english

File:

PDF, 229 KB

english, 2007

14

Chemical Space Travel

Ruud van Deursen, Jean-Louis Reymond

Journal:

Year:

2007

Language:

english

File:

PDF, 383 KB

english, 2007

15

Pathogenomics: Genome Analysis of Pathogenic Microbes. Edited by Jörg Hacker and Ulrich Dobrindt.

Journal:

Year:

2007

Language:

english

File:

PDF, 67 KB

english, 2007

16

Bioorganometallics: Biomolecules, Labeling, Medicine. Edited by Gérard Jaouen.

Journal:

Year:

2007

Language:

english

File:

PDF, 41 KB

english, 2007

17

Chirality in Drug Research. Edited by Eric Francotte and Wolfgang Lindner.

Journal:

Year:

2007

Language:

english

File:

PDF, 50 KB

english, 2007

18

Cover Picture: Ensemble-Docking Approach on BACE-1: Pharmacophore Perception and Guidelines for Drug Design (ChemMedChem 5/2007)

Vittorio Limongelli, Luciana Marinelli, Sandro Cosconati, Hannes A. Braun, Boris Schmidt, Ettore Novellino

Journal:

Year:

2007

File:

PDF, 36 KB

2007

19

Graphical Abstract: ChemMedChem 5/2007

Journal:

Year:

2007

Language:

english

File:

PDF, 444 KB

english, 2007

20

Spotlights on our sister journals: ChemMedChem 5/2007

Journal:

Year:

2007

Language:

english

File:

PDF, 328 KB

english, 2007

21

Preview: ChemMedChem 6/2007

Journal:

Year:

2007

Language:

english

File:

PDF, 30 KB

english, 2007