Volume 2; Issue 8

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ChemMedChem
Volume 2; Issue 8

ChemMedChem

Volume 2; Issue 8

1

Are MAP Kinases Drug Targets? Yes, but Difficult Ones

Simona Margutti, Stefan A. Laufer

Journal:

Year:

2007

Language:

english

File:

PDF, 1.17 MB

english, 2007

2

Tuning Sensitivity in Paramagnetic NMR Detection of Ligand–DNA Interactions

Emanuele Chirivino, Cesare Giordano, Sara Faini, Luciano Cellai, Marco Fragai

Journal:

Year:

2007

Language:

english

File:

PDF, 148 KB

english, 2007

3

Synthesis and Biological Evaluation of Phosphate Prodrugs of 4-Phospho-D -erythronohydroxamic Acid, an Inhibitor of 6-Phosphogluconate Dehydrogenase

Gian Filippo Ruda, Vincent P. Alibu, Christos Mitsos, Olivier Bidet, Marcel Kaiser, Reto Brun, Michael P. Barrett, Ian H. Gilbert

Journal:

Year:

2007

Language:

english

File:

PDF, 354 KB

english, 2007

4

Characterisation of a Novel Growth Hormone Variant Comprising a Thioether Link between Cys182 and Cys189

Antonio Datola, Sophie Richert, Horst Bierau, David Agugiaro, Anna Izzo, Mara Rossi, David Cregut, Hélène Diemer, Christine Schaeffer, Alain Van Dorsselaer, Carlo Emanuele Giartosio, Carl Jone

Journal:

Year:

2007

Language:

english

File:

PDF, 787 KB

english, 2007

5

Pyridin-2(1H)-ones: A Promising Class of HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors

José Luis Medina-Franco, Karina Martínez-Mayorga, Cecilia Juárez-Gordiano, Rafael Castillo

Journal:

Year:

2007

Language:

english

File:

PDF, 298 KB

english, 2007

6

Predicting and Tuning Physicochemical Properties in Lead Optimization: Amine Basicities

Martin Morgenthaler, Eliane Schweizer, Anja Hoffmann-Röder, Fausta Benini, Rainer E. Martin, Georg Jaeschke, Björn Wagner, Holger Fischer, Stefanie Bendels, Daniel Zimmerli, Josef Schneider, François

Journal:

Year:

2007

Language:

english

File:

PDF, 529 KB

english, 2007

7

Mannosylated G(0) Dendrimers with Nanomolar Affinities to Escherichia coli FimH

Mohamed Touaibia, Adinda Wellens, Tze Chieh Shiao, Qingan Wang, Suzanne Sirois, Julie Bouckaert, René Roy

Journal:

Year:

2007

Language:

english

File:

PDF, 360 KB

english, 2007

8

Oxime and Oxime Ether Derivatives of 1,4-Benzothiazine Related to Oxiconazole

Lara Milanese, Nicola Giacchè, Fausto Schiaffella, Anna Vecchiarelli, Antonio Macchiarulo, Renata Fringuelli

Journal:

Year:

2007

Language:

english

File:

PDF, 222 KB

english, 2007

9

Amphiphilic Poly[(propylene glycol)-block-(2-methyl-2-oxazoline)] Copolymers for Gene Transfer in Skeletal Muscle

Blandine Brissault, Antoine Kichler, Christian Leborgne, Nathalie Jarroux, Hervé Cheradame, Christine Guis

Journal:

Year:

2007

Language:

english

File:

PDF, 139 KB

english, 2007

10

Screening of Protease Inhibitors as Antiplasmodial Agents. Part I: Aziridines and Epoxides

Franziska Schulz, Christoph Gelhaus, Björn Degel, Radim Vicik, Saskia Heppner, Alexander Breuning, Matthias Leippe, Jiri Gut, Philip J. Rosenthal, Tanja Schirmeister

Journal:

Year:

2007

Language:

english

File:

PDF, 220 KB

english, 2007

11

Chemical Medicine: Novel 10-Substituted Cytisine Derivatives with Increased Selectivity for α4β2 Nicotinic Acetylcholine Receptors

Alan P. Kozikowski, Sheela K. Chellappan, Yingxian Xiao, Krishna Mohan Bajjuri, Hongbin Yuan, Kenneth J. Kellar, Pavel A. Petukhov

Journal:

Year:

2007

Language:

english

File:

PDF, 169 KB

english, 2007

12

The Construction of a Functional Photoactivatable Cancer Targeting Bispecific Antibody Conjugate

Stephen Thompson, Marie-Claude Fawcett, Colin H Self

Journal:

Year:

2007

Language:

english

File:

PDF, 198 KB

english, 2007

13

SERS Classification of Highly Related Performance Enhancers

Ramon A. Alvarez-Puebla, Juan P. Bravo-Vasquez, Bo Cui, Teodor Veres, Hicham Fenniri

Journal:

Year:

2007

Language:

english

File:

PDF, 384 KB

english, 2007

14

Hydrocarbon-Stapled Helices: A Novel Approach for Blocking Protein-Protein Interactions

Paul T. Wilder, Thomas H. Charpentier, David J. Weber

Journal:

Year:

2007

Language:

english

File:

PDF, 82 KB

english, 2007

15

Cover Picture: Mannosylated G(0) Dendrimers with Nanomolar Affinities to Escherichia coli FimH (ChemMedChem 8/2007)

Mohamed Touaibia, Adinda Wellens, Tze Chieh Shiao, Qingan Wang, Suzanne Sirois, Julie Bouckaert, René Roy

Journal:

Year:

2007

File:

PDF, 40 KB

2007

16

Graphical Abstract: ChemMedChem 8/2007

Journal:

Year:

2007

Language:

english

File:

PDF, 618 KB

english, 2007

17

Spotlights on our sister journals: ChemMedChem 8/2007

Journal:

Year:

2007

Language:

english

File:

PDF, 249 KB

english, 2007

18

Preview: ChemMedChem 9/2007

Journal:

Year:

2007

Language:

english

File:

PDF, 32 KB

english, 2007