Volume 4; Issue 9

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ChemMedChem
Volume 4; Issue 9

ChemMedChem

Volume 4; Issue 9

1

Pyrrole-Based Hydroxamates and 2-Aminoanilides: Histone Deacetylase Inhibition and Cellular Activities

Sergio Valente, Mariarosaria Conte, Maria Tardugno, Silvio Massa, Angela Nebbioso, Lucia Altucci, Antonello Mai

Journal:

Year:

2009

Language:

english

File:

PDF, 290 KB

english, 2009

2

Structure–Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability

Federica Vacondio, Claudia Silva, Alessio Lodola, Alessandro Fioni, Silvia Rivara, Andrea Duranti, Andrea Tontini, Silvano Sanchini, Jason R. Clapper, Daniele Piomelli, Marco Mor, Giorgio Tarzia

Journal:

Year:

2009

Language:

english

File:

PDF, 271 KB

english, 2009

3

Inhibition of Human Leukocyte Elastase by Brunsvicamides A–C: Cyanobacterial Cyclic Peptides

Mihiret T. Sisay, Stephanie Hautmann, Christian Mehner, Gabriele M. König, Jürgen Bajorath, Michael Gütschow

Journal:

Year:

2009

Language:

english

File:

PDF, 341 KB

english, 2009

4

Discovery of Ligands for the Human Intestinal Di-/Tripeptide Transporter (hPEPT1) Using a QSAR-Assisted Virtual Screening Strategy

Simon Birksø Larsen, Diana Højmark Omkvist, Birger Brodin, Carsten Uhd Nielsen, Bente Steffansen, Lars Olsen, Flemming Steen Jørgensen

Journal:

Year:

2009

Language:

english

File:

PDF, 494 KB

english, 2009

5

Indoloquinolizidine–Peptide Hybrids as Multiple Agonists for D1 and D2 Dopamine Receptors

Marc Vendrell, Aroa Soriano, Vicent Casadó, José Luis Díaz, Rodolfo Lavilla, Enric I. Canela, Carme Lluís, Rafael Franco, Fernando Albericio, Miriam Royo

Journal:

Year:

2009

Language:

english

File:

PDF, 287 KB

english, 2009

6

Synthesis and in vitro Evaluation of Trifluoroethylamine Analogues of Enkephalins

Roberta Sinisi, Alessandra Ghilardi, Stefania Ruiu, Paolo Lazzari, Luciana Malpezzi, Monica Sani, Luca Pani, Matteo Zanda

Journal:

Year:

2009

Language:

english

File:

PDF, 222 KB

english, 2009

7

Induced-Fit Docking Approach Provides Insight into the Binding Mode and Mechanism of Action of HIV-1 Integrase Inhibitors

Maria Letizia Barreca, Nunzio Iraci, Laura De Luca, Alba Chimirri

Journal:

Year:

2009

Language:

english

File:

PDF, 891 KB

english, 2009

8

Synthesis, Crystal Structure and Immunosuppressive Activity of Acylamide Derivatives Containing 1,4-Benzodioxan

Peng-Cheng Lv, Kai-Rui Wang, Wen-Jun Mao, Jing Xiong, Huan-Qiu Li, Ying Yang, Lei Shi, Hai-Liang Zhu

Journal:

Year:

2009

Language:

english

File:

PDF, 231 KB

english, 2009

9

Ex vivo and in vivo Evaluation of [18F]PR04.MZ in Rodents: A Selective Dopamine Transporter Imaging Agent

Patrick J. Riss, Fabian Debus, René Hummerich, Ulrich Schmidt, Patrick Schloss, Hartmut Lueddens, Frank Roesch

Journal:

Year:

2009

Language:

english

File:

PDF, 449 KB

english, 2009

10

Synthesis and Evaluation of New Antagonists of Bacterial Quorum Sensing in Vibrio harveyi

Hanjing Peng, Yunfeng Cheng, Nanting Ni, Minyong Li, Gaurav Choudhary, Han Ting Chou, Chung-Dar Lu, Phang C. Tai, Binghe Wang

Journal:

Year:

2009

Language:

english

File:

PDF, 478 KB

english, 2009

11

Retro-Enantio N-Methylated Peptides as β-Amyloid Aggregation Inhibitors

Dolors Grillo-Bosch, Natàlia Carulla, Montse Cruz, Laia Sánchez, Rosa Pujol-Pina, Sergio Madurga, Francesc Rabanal, Ernest Giralt

Journal:

Year:

2009

Language:

english

File:

PDF, 588 KB

english, 2009

12

Docking Studies of Structurally Diverse Antimalarial Drugs Targeting PfATP6: No Correlation between in silico Binding Affinity and in vitro Antimalarial Activity.

Fatima Bousejra-El Garah, Jean-Luc Stigliani, Frédéric Coslédan, Bernard Meunier, Anne Robert

Journal:

Year:

2009

Language:

english

File:

PDF, 1.02 MB

english, 2009

13

MS Binding Assays—with MALDI toward High Throughput

Georg Höfner, Dietrich Merkel, Klaus Theodor Wanner

Journal:

Year:

2009

Language:

english

File:

PDF, 258 KB

english, 2009

14

A Consistent Dataset of Kinetic Solubilities for Early-Phase Drug Discovery

Christian Kramer, Tilmann Heinisch, Thilo Fligge, Bernd Beck, Timothy Clark

Journal:

Year:

2009

Language:

english

File:

PDF, 446 KB

english, 2009

15

A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo

Jason R. Clapper, Federica Vacondio, Alvin R. King, Andrea Duranti, Andrea Tontini, Claudia Silva, Silvano Sanchini, Giorgio Tarzia, Marco Mor, Daniele Piomelli

Journal:

Year:

2009

Language:

english

File:

PDF, 302 KB

english, 2009

16

Design, Synthesis, and SAR of Naphthyl-Substituted Diarylpyrimidines as Non-Nucleoside Inhibitors of HIV-1 Reverse Transcriptase

Yong-Hong Liang, Xiao-Qing Feng, Zhao-Sen Zeng, Fen-Er Chen, Jan Balzarini, Christophe Pannecouque, Erik De Clercq

Journal:

Year:

2009

Language:

english

File:

PDF, 314 KB

english, 2009

17

Systematic Extraction of Structure–Activity Relationship Information from Biological Screening Data

Mathias Wawer, Jürgen Bajorath

Journal:

Year:

2009

Language:

english

File:

PDF, 552 KB

english, 2009

18

Chemoinformatics Approaches to Virtual Screening. Edited by Alexandre Varnek and Alexander Tropsha.

Christof Wegscheid-Gerlach

Journal:

Year:

2009

Language:

english

File:

PDF, 100 KB

english, 2009

19

Drugs: From Discovery to Approval (2nd ed.). By Rick Ng.

Journal:

Year:

2009

Language:

english

File:

PDF, 133 KB

english, 2009

20

Structure-Based and in silico Design of Hsp90 Inhibitors

Miriam Sgobba, Giulio Rastelli

Journal:

Year:

2009

Language:

english

File:

PDF, 727 KB

english, 2009

21

Cover Picture: Structure–Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability / A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo (ChemMedChem 9/2009)

Federica Vacondio, Claudia Silva, Alessio Lodola, Alessandro Fioni, Silvia Rivara, Andrea Duranti, Andrea Tontini, Silvano Sanchini, Jason R. Clapper, Daniele Piomelli, Marco Mor, Giorgio Tarzia, Alvi

Journal:

Year:

2009

Language:

english

File:

PDF, 792 KB

english, 2009

22

Inside Cover: Docking Studies of Structurally Diverse Antimalarial Drugs Targeting PfATP6: No Correlation between in silico Binding Affinity and in vitro Antimalarial Activity. (ChemMedChem 9/2009)

Fatima Bousejra-El Garah, Jean-Luc Stigliani, Frédéric Coslédan, Bernard Meunier, Anne Robert

Journal:

Year:

2009

Language:

english

File:

PDF, 547 KB

english, 2009

23

Graphical Abstract: ChemMedChem 9/2009

Journal:

Year:

2009

Language:

english

File:

PDF, 1.00 MB

english, 2009

24

Spotlights on our sister journals: ChemMedChem 9/2009

Journal:

Year:

2009

Language:

english

File:

PDF, 571 KB

english, 2009

25

Preview: ChemMedChem 10/2009

Journal:

Year:

2009

Language:

english

File:

PDF, 109 KB

english, 2009

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