Volume 5; Issue 10

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ChemMedChem
Volume 5; Issue 10

ChemMedChem

Volume 5; Issue 10

1

Synthesis of Fatty Acid Amides of Catechol Metabolites that Exhibit Antiobesity Properties

Bruno Almeida, Dr. Jesús Joglar, María Jesús Luque Rojas, Juan Manuel Decara, Francisco Javier Bermúdez-Silva, Dr. Manuel Macias-González, Dr. Montserrat Fitó, Miguel Romero-Cuevas, Dr. Magí Farré, Dr

Journal:

Year:

2010

Language:

english

File:

PDF, 325 KB

english, 2010

2

NOC Chemistry for Tuberculosis—Further Investigations on the Structure–Activity Relationships of Antitubercular Isoxazole-3-carboxylic Acid Ester Derivatives

Dr. Marco Pieroni, Dr. Annamaria Lilienkampf, Dr. Yuehong Wang, Dr. Baojie Wan, Dr. Sanghyun Cho, Prof. Dr. Scott G. Franzblau, Prof. Dr. Alan P. Kozikowski

Journal:

Year:

2010

Language:

english

File:

PDF, 238 KB

english, 2010

3

Synthesis and Evaluation of Bombesin Analogues Conjugated to Two Different Triazolyl-Derived Chelators for 99mTc Labeling

Dr. Luc Brans, Dr. Elisa García-Garayoa, Dr. Christian Schweinsberg, Dr. Veronique Maes, Dr. Harriet Struthers, Prof. Roger Schibli, Prof. Dirk Tourwé

Journal:

Year:

2010

Language:

english

File:

PDF, 630 KB

english, 2010

4

Structural Basis for the Improved Potency of Peroxisome Proliferator-Activated Receptor (PPAR) Agonists

Yi-Hui Peng, Dr. Mohane Selvaraj Coumar, Jiun-Shyang Leou, Jian-Sung Wu, Dr. Hui-Yi Shiao, Dr. Chia-Hui Lin, Dr. Wen-Hsing Lin, Tzu Wen Lien, Dr. Xin Chen, Dr. John T.-A. Hsu, Dr. Yu-Sheng Chao, Dr. C

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Year:

2010

Language:

english

File:

PDF, 689 KB

english, 2010

5

Discovery of a Novel Hsp90 Inhibitor by Fragment Linking

Dr. John J. Barker, Dr. Oliver Barker, Dr. Stephen M. Courtney, Dr. Mihaly Gardiner, Dr. Thomas Hesterkamp, Dr. Osamu Ichihara, Dr. Owen Mather, Dr. Christian A. G. N. Montalbetti, Dr. Annett Müller,

Journal:

Year:

2010

Language:

english

File:

PDF, 606 KB

english, 2010

6

New Halogenated Water-Soluble Chlorin and Bacteriochlorin as Photostable PDT Sensitizers: Synthesis, Spectroscopy, Photophysics, and in vitro Photosensitizing Efficacy

Dr. Janusz M. Dąbrowski, Prof. Luis G. Arnaut, Prof. Mariette M. Pereira, Carlos J. P. Monteiro, Prof. Krystyna Urbańska, Prof. Sérgio Simões, Prof. Grażyna Stochel

Journal:

Year:

2010

Language:

english

File:

PDF, 575 KB

english, 2010

7

The DAT Ligand [18F]PR17.MZ Mirrors the in vivo Pharmacokinetic Profile of [11C]Cocaine with Significantly Improved Monoamine Transporter Selectivity

Dr. Patrick J. Riss, Dr. Markus Piel, Vanessa Bockhart, Nicole Bausbacher, Hans-Georg Buchholz, Dr. Hartmut Lueddens, Dr. Frank Roesch

Journal:

Year:

2010

Language:

english

File:

PDF, 285 KB

english, 2010

8

Lead Generation Approaches in Drug Discovery. Edited by Zoran Rankovic and Richard Morphy.

Journal:

Year:

2010

Language:

english

File:

PDF, 107 KB

english, 2010

9

Design and Synthesis of Selective and Potent Orally Active S1P5 Agonists

Dr. Henri Mattes, Prof. Dr. Kumlesh Kumar Dev, Dr. Rochdi Bouhelal, Dr. Carmen Barske, Dr. Fabrizio Gasparini, Dr. Danilo Guerini, Dr. Anis Khusro Mir, Dr. David Orain, Maribel Osinde, Anne Picard, Ce

Journal:

Year:

2010

Language:

english

File:

PDF, 455 KB

english, 2010

10

Developments in Nonsteroidal Antiandrogens Targeting the Androgen Receptor

Bo Liu, Lei Su, Jingkun Geng, Junjie Liu, Prof. Guisen Zhao

Journal:

Year:

2010

Language:

english

File:

PDF, 488 KB

english, 2010

11

High-Resolution Crystal Structure of a Lasso Peptide

Dr. Herbert Nar, Angela Schmid, Dr. Carsten Puder, Dr. Olivier Potterat

Journal:

Year:

2010

Language:

english

File:

PDF, 633 KB

english, 2010

12

α-Ketoheterocycles as Inhibitors of Leishmania mexicana Cysteine Protease CPB

Dr. Koen Steert, Dr. Maya Berg, Prof. Dr. Jeremy C. Mottram, Dr. Gareth D. Westrop, Prof. Dr. Graham H. Coombs, Prof. Dr. Paul Cos, Prof. Dr. Louis Maes, Dr. Jurgen Joossens, Prof. Dr. Pieter Van der

Journal:

Year:

2010

Language:

english

File:

PDF, 392 KB

english, 2010

13

Structural and Potency Relationships between Scaffolds of Compounds Active against Human Targets

Ye Hu, Prof. Dr. Jürgen Bajorath

Journal:

Year:

2010

Language:

english

File:

PDF, 491 KB

english, 2010

14

Synthesis and Antiplasmodial Activity of Highly Active Reverse Analogues of the Antimalarial Drug Candidate Fosmidomycin

Christoph T. Behrendt, Andrea Kunfermann, Dr. Victoria Illarionova, An Matheeussen, Dr. Tobias Gräwert, Prof. Michael Groll, Dr. Felix Rohdich, Prof. Adelbert Bacher, Dr. Wolfgang Eisenreich, Prof. Dr

Journal:

Year:

2010

Language:

english

File:

PDF, 232 KB

english, 2010

15

Understanding the Key Factors that Control the Inhibition of Type II Dehydroquinase by (2R)-2-Benzyl-3-dehydroquinic Acids

Antonio Peón, Dr. José M. Otero, Lorena Tizón, Verónica F. V. Prazeres, Dr. Antonio L. Llamas-Saiz, Dr. Gavin C. Fox, Dr. Mark J. van Raaij, Dr. Heather Lamb, Prof. Dr. Alastair R. Hawkins, Prof. Dr.

Journal:

Year:

2010

Language:

english

File:

PDF, 1.29 MB

english, 2010

16

Dansyl C-Glucoside as a Novel Agent Against Endotoxic Shock

Dr. Barbara La Ferla, Valerio Spinosa, Giuseppe D'Orazio, Dr. Marco Palazzo, Prof. Andrea Balsari, Dr. Anastasia A. Foppoli, Prof. Cristiano Rumio, Prof. Francesco Nicotra

Journal:

Year:

2010

Language:

english

File:

PDF, 404 KB

english, 2010

17

20S Proteasome Inhibition: Designing Noncovalent Linear Peptide Mimics of the Natural Product TMC-95A

Prof. Dr. Michael Groll, Nerea Gallastegui, Xavier Maréchal, Dr. Virginie Le Ravalec, Dr. Nicolas Basse, Dr. Nicolas Richy, Dr. Emilie Genin, Prof. Dr. Robert Huber, Prof. Dr. Luis Moroder, Prof. Dr.

Journal:

Year:

2010

Language:

english

File:

PDF, 548 KB

english, 2010

18

Synthesis of Benzofuran, Benzothiophene, and Benzothiazole-Based Thioamides and their Evaluation as KATP Channel Openers

Andreas Fischer , Claas Schmidt , Dr. Stefan Lachenicht, Dagmar Grittner, Dr. Marcus Winkler, Thomas Wrobel, Achim Rood, Prof. Dr. Horst Lemoine, Prof. Dr. Walter Frank, Prof. Dr. Manfred Braun

Journal:

Year:

2010

Language:

english

File:

PDF, 360 KB

english, 2010

19

Handbook of Pharmaceutical Natural Products. By Goutam Brahmachari.

Prof. Dr. Karl-Heinz Altmann

Journal:

Year:

2010

Language:

english

File:

PDF, 121 KB

english, 2010

20

Drugs for Hepatitis C: Unlocking a New Mechanism of Action

Prof. Thomas W. Bell

Journal:

Year:

2010

Language:

english

File:

PDF, 174 KB

english, 2010

21

Cover Picture: High-Resolution Crystal Structure of a Lasso Peptide (ChemMedChem 10/2010)

Dr. Herbert Nar, Angela Schmid, Dr. Carsten Puder, Dr. Olivier Potterat

Journal:

Year:

2010

File:

PDF, 797 KB

2010

22

Inside Cover: Design and Synthesis of Selective and Potent Orally Active S1P5 Agonists (ChemMedChem 10/2010)

Dr. Henri Mattes, Prof. Dr. Kumlesh Kumar Dev, Dr. Rochdi Bouhelal, Dr. Carmen Barske, Dr. Fabrizio Gasparini, Dr. Danilo Guerini, Dr. Anis Khusro Mir, Dr. David Orain, Maribel Osinde, Anne Picard, Ce

Journal:

Year:

2010

Language:

english

File:

PDF, 518 KB

english, 2010

23

Graphical Abstract: ChemMedChem 10/2010

Journal:

Year:

2010

Language:

english

File:

PDF, 978 KB

english, 2010

24

Corrigendum: Design and Synthesis of Selective and Potent Orally Active S1P5 Agonists

Dr. Henri Mattes, Prof. Dr. Kumlesh Kumar Dev, Dr. Rochdi Bouhelal, Dr. Carmen Barske, Dr. Fabrizio Gasparini, Dr. Danilo Guerini, Dr. Anis Khusro Mir, Dr. David Orain, Maribel Osinde, Anne Picard, Ce

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2010

File:

PDF, 57 KB

2010

25

Spotlights on our sister journals: ChemMedChem 10/2010

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Year:

2010

Language:

english

File:

PDF, 823 KB

english, 2010

26

Preview: ChemMedChem 11/2010

Journal:

Year:

2010

Language:

english

File:

PDF, 80 KB

english, 2010

27

Structure–Activity Relationships and Molecular Docking of Novel Dihydropyrimidine-Based Mitotic Eg5 Inhibitors

Dr. Hana Prokopcová, Dr. Doris Dallinger, Prof. Dr. Georg Uray, Hung Yi Kristal Kaan, Dr. Venkatasubramanian Ulaganathan, Prof. Dr. Frank Kozielski, Dr. Christian Laggner, Prof. Dr. C. Oliver Kappe

Journal:

Year:

2010

Language:

english

File:

PDF, 455 KB

english, 2010

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