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Volume 5; Issue 8
Main
ChemMedChem
Volume 5; Issue 8
ChemMedChem
Volume 5; Issue 8
1
Modelling Inhalational Anaesthetics Using Bayesian Feature Selection and QSAR Modelling Methods
David T. Manallack
,
Frank R. Burden
,
David A. Winkler
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 171 KB
Your tags:
english, 2010
2
Exploring the ‘RPRL’ Motif of Apelin-13 through Molecular Simulation and Biological Evaluation of Cyclic Peptide Analogues
N. J. Maximilian Macaluso
,
Robert C. Glen
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 577 KB
Your tags:
english, 2010
3
Design and Synthesis of Thiadiazoles and Thiazoles Targeting the Bcr-Abl T315I Mutant: from Docking False Positives to ATP-Noncompetitive Inhibitors
Marco Radi
,
Emmanuele Crespan
,
Federico Falchi
,
Vincenzo Bernardo
,
Samantha Zanoli
,
Fabrizio Manetti
,
Silvia Schenone
,
Giovanni Maga
,
Maurizio Botta
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 408 KB
Your tags:
english, 2010
4
Recent Advances in Endomorphin Engineering
Attila Keresztes
,
Attila Borics
,
Géza Tóth
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 679 KB
Your tags:
english, 2010
5
Bis(7)-tacrine Derivatives as Multitarget-Directed Ligands: Focus on Anticholinesterase and Antiamyloid Activities
Maria Laura Bolognesi
,
Manuela Bartolini
,
Francesca Mancini
,
Gianpaolo Chiriano
,
Luisa Ceccarini
,
Michela Rosini
,
Andrea Milelli
,
Vincenzo Tumiatti
,
Vincenza Andrisano
,
Carlo Melchiorre
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 319 KB
Your tags:
english, 2010
6
A Structure–Activity Relationship Study of the Antimalarial and Antileishmanial Activities of Nonpeptide Macrocyclic Histone Deacetylase Inhibitors
William Guerrant
,
Sandra C. Mwakwari
,
Po C. Chen
,
Shabana I. Khan
,
Babu L. Tekwani
,
Adegboyega K. Oyelere
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 183 KB
Your tags:
english, 2010
7
Synthesis, 3D-QSAR, and Structural Modeling of Benzolactam Derivatives with Binding Affinity for the D2 and D3 Receptors
Laura López
,
Jana Selent
,
Raquel Ortega
,
Christian F. Masaguer
,
Eduardo Domínguez
,
Filipe Areias
,
José Brea
,
María Isabel Loza
,
Ferran Sanz
,
Manuel Pastor
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 1.09 MB
Your tags:
english, 2010
8
Proteins as Possible Targets for Cytotoxic trans-Platinum(II) Complexes with Aliphatic Amine Ligands: Further Exceptions to the DNA Paradigm
Leticia Cubo
,
Michael Groessl
,
Paul J. Dyson
,
Adoración G. Quiroga
,
Carmen Navarro-Ranninger
,
Angela Casini
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 407 KB
Your tags:
english, 2010
9
Discovery of Carboranes as Inducers of 20S Proteasome Activity
Hyun Seung Ban
,
Hidemitsu Minegishi
,
Kazuki Shimizu
,
Minako Maruyama
,
Yuka Yasui
,
Hiroyuki Nakamura
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 287 KB
Your tags:
english, 2010
10
Novel Monocyclam Derivatives as HIV Entry Inhibitors: Design, Synthesis, Anti-HIV Evaluation, and Their Interaction with the CXCR4 Co-receptor
Sofia Pettersson
,
Violeta I. Pérez-Nueno
,
Maria Pau Mena
,
Bonaventura Clotet
,
José A. Esté
,
José I. Borrell
,
Jordi Teixidó
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 1.12 MB
Your tags:
english, 2010
11
Orexin Receptor Antagonists: A New Concept In CNS Disorders?
John Gatfield
,
Catherine Brisbare-Roch
,
Francois Jenck
,
Christoph Boss
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 913 KB
Your tags:
english, 2010
12
Discovery of a Class of Diketopiperazines as Antiprion Compounds
Maria Laura Bolognesi
,
Hoang Ngoc Ai Tran
,
Matteo Staderini
,
Alessandra Monaco
,
Alberto López-Cobeñas
,
Salvatore Bongarzone
,
Xevi Biarnés
,
Pilar López-Alvarado
,
Nieves Cabezas
,
Maria Caramelli
,
Paolo
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 391 KB
Your tags:
english, 2010
13
Off-Target Effects Related to the Phosphorothioate Modification of Nucleic Acids
Johannes Winkler
,
Martina Stessl
,
Jennifer Amartey
,
Christian R. Noe
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 577 KB
Your tags:
english, 2010
14
Inhibition of Eimeria tenella CDK-Related Kinase 2: From Target Identification to Lead Compounds
Kristin Engels
,
Carsten Beyer
,
Maria L. Suárez Fernández
,
Frank Bender
,
Michael Gaßel
,
Gottfried Unden
,
Richard J. Marhöfer
,
Jeremy C. Mottram
,
Paul M. Selzer
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 1.72 MB
Your tags:
english, 2010
15
Structure-Based Virtual Screening and Electrophysiological Evaluation of New Chemotypes of Kv1.5 Channel Blockers
Qian Yang
,
David Fedida
,
Hongjian Xu
,
Binghe Wang
,
Lupei Du
,
Xiaojian Wang
,
Minyong Li
,
Qidong You
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 492 KB
Your tags:
english, 2010
16
Hit Identification and Biological Evaluation of Anticancer Pyrazolopyrimidines Endowed with Anti-inflammatory Activity
Stefano Alcaro
,
Anna Artese
,
Maurizio Botta
,
Alessandra T. Zizzari
,
Francisco Orallo
,
Francesco Ortuso
,
Silvia Schenone
,
Chiara Brullo
,
Matilde Yáñez
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 299 KB
Your tags:
english, 2010
17
Synthesis and Biological Characterization of Amidopropenyl Hydroxamates as HDAC Inhibitors
Florian Thaler
,
Mario Varasi
,
Andrea Colombo
,
Roberto Boggio
,
Davide Munari
,
Nickolas Regalia
,
Marco G. Rozio
,
Veronica Reali
,
Anna E. Resconi
,
Antonello Mai
,
Stefania Gagliardi
,
Giulio Dondio
,
Saveri
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 351 KB
Your tags:
english, 2010
18
The Role of Fluorine Atoms in a Fluorinated Prostaglandin Agonist
Ken-ichi Fujimura
,
Yoshimasa Sasabuchi
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 607 KB
Your tags:
english, 2010
19
Synthesis and in vitro Evaluation of 3H-Pyrrolo[3,2-f]quinolin-9-one Derivatives That Show Potent and Selective Anti-leukemic Activity
Maria Grazia Ferlin
,
Roberta Bortolozzi
,
Paola Brun
,
Ignazio Castagliuolo
,
Ernest Hamel
,
Giuseppe Basso
,
Giampietro Viola
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 662 KB
Your tags:
english, 2010
20
HTS and Rational Drug Design to Generate a Class of 5-HT2C-Selective Ligands for Possible Use in Schizophrenia.
Alan P. Kozikowski
,
Sung Jin Cho
,
Niels H. Jensen
,
John A. Allen
,
Andreas M. Svennebring
,
Bryan L. Roth
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 386 KB
Your tags:
english, 2010
21
CycloSal-phosphate Pronucleotides of Cytostatic 6-(Het)aryl-7-deazapurine Ribonucleosides: Synthesis, Cytostatic Activity, and Inhibition of Adenosine Kinases
Pavla Spáčilová
,
Petr Nauš
,
Radek Pohl
,
Ivan Votruba
,
Jan Snášel
,
Helena Zábranská
,
Iva Pichová
,
Ria Ameral
,
Gabriel Birkuš
,
Tomáš Cihlář
,
Michal Hocek
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 378 KB
Your tags:
english, 2010
22
Ligand-Binding Assays: Development, Validation, and Implementation in the Drug Development Arena. Edited by Masood N. Khan and John W. Findlay.
Claudiu Supuran
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 91 KB
Your tags:
english, 2010
23
Facile Oxidation of Leucomethylene Blue and Dihydroflavins by Artemisinins: Relationship with Flavoenzyme Function and Antimalarial Mechanism of Action
Richard K. Haynes
,
Wing-Chi Chan
,
Ho-Ning Wong
,
Ka-Yan Li
,
Wai-Keung Wu
,
Kit-Man Fan
,
Herman H. Y. Sung
,
Ian D. Williams
,
Davide Prosperi
,
Sergio Melato
,
Paolo Coghi
,
Diego Monti
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 913 KB
Your tags:
english, 2010
24
A Practical Guide to Assay Development and High-Throughput Screening in Drug Discovery. Edited by Taosheng Chen.
James Inglese
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 127 KB
Your tags:
english, 2010
25
“Hot Spots” in Medicinal Chemistry
Rainer Metternich
,
Giorgio Tarzia
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 285 KB
Your tags:
english, 2010
26
Cover Picture: Discovery of a Class of Diketopiperazines as Antiprion Compounds (ChemMedChem 8/2010)
Maria Laura Bolognesi
,
Hoang Ngoc Ai Tran
,
Matteo Staderini
,
Alessandra Monaco
,
Alberto López-Cobeñas
,
Salvatore Bongarzone
,
Xevi Biarnés
,
Pilar López-Alvarado
,
Nieves Cabezas
,
Maria Caramelli
,
Paolo
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 996 KB
Your tags:
english, 2010
27
Inside Cover: Inhibition of Eimeria tenella CDK-Related Kinase 2: From Target Identification to Lead Compounds (ChemMedChem 8/2010)
Kristin Engels
,
Carsten Beyer
,
Maria L. Suárez Fernández
,
Frank Bender
,
Michael Gaßel
,
Gottfried Unden
,
Richard J. Marhöfer
,
Jeremy C. Mottram
,
Paul M. Selzer
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 635 KB
Your tags:
english, 2010
28
Graphical Abstract: ChemMedChem 8/2010
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 866 KB
Your tags:
english, 2010
29
Spotlights on our sister journals: ChemMedChem 8/2010
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 774 KB
Your tags:
english, 2010
30
Preview: ChemMedChem 9/2010
Journal:
ChemMedChem
Year:
2010
Language:
english
File:
PDF, 99 KB
Your tags:
english, 2010
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