Volume 6; Issue 7

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ChemMedChem
Volume 6; Issue 7

ChemMedChem

Volume 6; Issue 7

1

Recent Advances in the Development of Dopamine D3 Receptor Antagonists: a Medicinal Chemistry Perspective

Dr. Fabrizio Micheli

Journal:

Year:

2011

Language:

english

File:

PDF, 804 KB

english, 2011

2

Biphenyl Sulfonylamino Methyl Bisphosphonic Acids as Inhibitors of Matrix Metalloproteinases and Bone Resorption

Dr. Maria Teresa Rubino, Dr. Mariangela Agamennone, Dr. Cristina Campestre, Dr. Pietro Campiglia, Dr. Viviana Cremasco, Prof. Roberta Faccio, Dr. Antonio Laghezza, Prof. Fulvio Loiodice, Dr. Dariana M

Journal:

Year:

2011

Language:

english

File:

PDF, 552 KB

english, 2011

3

Carbamate Prodrug Concept for Hydroxamate HDAC Inhibitors

Dr. Sonja Schlimme, Dr. Alexander-Thomas Hauser, Vincenzo Carafa, Ralf Heinke, Dr. Srinivasaraghavan Kannan, Dr. Diana A. Stolfa, Saverio Cellamare, Prof. Angelo Carotti, Prof. Lucia Altucci, Prof. Ma

Journal:

Year:

2011

Language:

english

File:

PDF, 398 KB

english, 2011

4

Early Drug Development: Strategies and Routes to First-in-Human Trials. Edited by Mitchell N. Cayen.

Dr. Klaus Weigand

Journal:

Year:

2011

Language:

english

File:

PDF, 96 KB

english, 2011

5

Synthesis of Triazenoazaindoles: a New Class of Triazenes with Antitumor Activity

Prof. Patrizia Diana, Dr. Antonina Stagno, Prof. Paola Barraja, Dr. Anna Carbone, Dr. Barbara Parrino, Prof. Francesco Dall'Acqua, Prof. Daniela Vedaldi, Dr. Alessia Salvador, Dr. Paola Brun, Prof. Ig

Journal:

Year:

2011

Language:

english

File:

PDF, 435 KB

english, 2011

6

DNA Reactivity Profile of trans-Platinum Planar Amine Derivatives

Dr. Caterina Musetti, Dr. Alexey A. Nazarov, Prof. Nicholas P. Farrell, Prof. Claudia Sissi

Journal:

Year:

2011

Language:

english

File:

PDF, 576 KB

english, 2011

7

The Approach of Conformational Chimeras to Model the Role of Proline-Containing Helices on GPCR Mobility: the Fertile Case of Cys-LTR1

Dr. Ilaria Bettinelli, Dr. Davide Graziani, Dr. Cristina Marconi, Dr. Alessandro Pedretti, Prof. Giulio Vistoli

Journal:

Year:

2011

Language:

english

File:

PDF, 895 KB

english, 2011

8

Neuropeptide S Receptor: Recent Updates on Nonpeptide Antagonist Discovery

Dr. Diego Dal Ben, Prof. Ippolito Antonini, Dr. Michela Buccioni, Dr. Catia Lambertucci, Prof. Gabriella Marucci, Ajiroghene Thomas, Prof. Rosaria Volpini, Prof. Gloria Cristalli

Journal:

Year:

2011

Language:

english

File:

PDF, 407 KB

english, 2011

9

Design, Synthesis, ADME Properties, and Pharmacological Activities of β-Alanyl-D-histidine (D-Carnosine) Prodrugs with Improved Bioavailability

Dr. Marica Orioli, Prof. Giulio Vistoli, Dr. Luca Regazzoni, Dr. Alessandro Pedretti, Prof. Annunziata Lapolla, Dr. Giuseppe Rossoni, Dr. Renato Canevotti, Dr. Luca Gamberoni, Massimo Previtali, Prof.

Journal:

Year:

2011

Language:

english

File:

PDF, 432 KB

english, 2011

10

The Role of the N-Terminal Domain in the Regulation of the “Constitutively Active” Conformation of Protein Kinase CK2α: Insight from a Molecular Dynamics Investigation

Andrea Cristiani, Giorgio Costa, Dr. Giorgio Cozza, Prof. Dr. Flavio Meggio, Prof. Dr. Leonardo Scapozza, Prof. Dr. Stefano Moro

Journal:

Year:

2011

Language:

english

File:

PDF, 971 KB

english, 2011

11

Inhibitors of the Interactions between HIV-1 IN and the Cofactor LEDGF/p75

Dr. Laura De Luca, Dr. Stefania Ferro, Dr. Francesca Morreale, Dr. Sara De Grazia, Prof. Alba Chimirri

Journal:

Year:

2011

Language:

english

File:

PDF, 471 KB

english, 2011

12

Structural Investigation of the Naphthyridone Scaffold: Identification of a 1,6-Naphthyridone Derivative with Potent and Selective Anti-HIV Activity

Prof. Oriana Tabarrini, Dr. Serena Massari, Dr. Luca Sancineto, Dr. Dirk Daelemans, Dr. Stefano Sabatini, Dr. Giuseppe Manfroni, Prof. Violetta Cecchetti, Prof. Christophe Pannecouque

Journal:

Year:

2011

Language:

english

File:

PDF, 303 KB

english, 2011

13

Synthesis and Antitumor Activity of 3-(2-Phenyl-1,3-thiazol-4-yl)-1H-indoles and 3-(2-Phenyl-1,3-thiazol-4-yl)-1H-7-azaindoles

Prof. Patrizia Diana, Dr. Anna Carbone, Prof. Paola Barraja, Dr. Alessandra Montalbano, Dr. Barbara Parrino, Dr. Alessia Lopergolo, Dr. Marzia Pennati, Dr. Nadia Zaffaroni, Prof. Girolamo Cirrincione

Journal:

Year:

2011

Language:

english

File:

PDF, 317 KB

english, 2011

14

Pyrrolo[3,2-h]quinazolines as Photochemotherapeutic Agents

Prof. Paola Barraja, Dr. Libero Caracausi, Prof. Patrizia Diana, Dr. Alessandra Montalbano, Dr. Anna Carbone, Dr. Alessia Salvador, Dr. Paola Brun, Prof. Ignazio Castagliuolo, Dr. Silvia Tisi, Prof. F

Journal:

Year:

2011

Language:

english

File:

PDF, 422 KB

english, 2011

15

Development of Novel Peptidomimetics Containing a Vinyl Sulfone Moiety as Proteasome Inhibitors

Dr. Roberta Ettari, Dr. Cinzia Bonaccorso, Dr. Nicola Micale, Cornelia Heindl, Prof. Dr. Tanja Schirmeister, Prof. Maria Luisa Calabrò, Prof. Silvana Grasso, Prof. Maria Zappalà

Journal:

Year:

2011

Language:

english

File:

PDF, 276 KB

english, 2011

16

Selective Inhibition of iNOS by Benzyl- and Dibenzyl Derivatives of N-(3-Aminobenzyl)acetamidine

Dr. Marialuigia Fantacuzzi, Dr. Cristina Maccallini, Dr. Fabio Lannutti, Dr. Antonia Patruno, Dr. Simona Masella, Dr. Mirko Pesce, Dr. Lorenza Speranza, Dr. Alessandra Ammazzalorso, Dr. Barbara De Fil

Journal:

Year:

2011

Language:

english

File:

PDF, 250 KB

english, 2011

17

Chemistry and Biological Activity of Platinum Amidine Complexes

Prof. Rino A. Michelin, Dr. Paolo Sgarbossa, Dr. Silvia Mazzega Sbovata, Dr. Valentina Gandin, Dr. Cristina Marzano, Dr. Roberta Bertani

Journal:

Year:

2011

Language:

english

File:

PDF, 406 KB

english, 2011

18

RNA Interference: Application to Drug Discovery and Challenges to Pharmaceutical Development. Edited by Paul H. Johnson.

Dr. Álvaro Somoza

Journal:

Year:

2011

Language:

english

File:

PDF, 78 KB

english, 2011

19

Gisbert Schneider

Journal:

Year:

2011

Language:

english

File:

PDF, 365 KB

english, 2011

20

Benzisothiazolyliminothiazolidin-4-ones with Chondroprotective Properties: Searching for Potent and Selective Inhibitors of MMP-13

Prof. Paola Vicini, Dr. Lucia Crascì, Dr. Matteo Incerti, Dr. Simone Ronsisvalle, Prof. Venera Cardile, Prof. Anna Maria Panico

Journal:

Year:

2011

Language:

english

File:

PDF, 674 KB

english, 2011

21

Cover Picture: Biphenyl Sulfonylamino Methyl Bisphosphonic Acids as Inhibitors of Matrix Metalloproteinases and Bone Resorption (ChemMedChem 7/2011)

Dr. Maria Teresa Rubino, Dr. Mariangela Agamennone, Dr. Cristina Campestre, Dr. Pietro Campiglia, Dr. Viviana Cremasco, Prof. Roberta Faccio, Dr. Antonio Laghezza, Prof. Fulvio Loiodice, Dr. Dariana M

Journal:

Year:

2011

Language:

english

File:

PDF, 1.33 MB

english, 2011

22

Inside Cover: The Role of the N-Terminal Domain in the Regulation of the “Constitutively Active” Conformation of Protein Kinase CK2α: Insight from a Molecular Dynamics Investigation (ChemMedChem 7/2011)

Andrea Cristiani, Giorgio Costa, Dr. Giorgio Cozza, Prof. Dr. Flavio Meggio, Prof. Dr. Leonardo Scapozza, Prof. Dr. Stefano Moro

Journal:

Year:

2011

File:

PDF, 454 KB

2011

23

Graphical Abstract: ChemMedChem 7/2011

Journal:

Year:

2011

Language:

english

File:

PDF, 1.01 MB

english, 2011

24

Spotlights on our sister journals: ChemMedChem 7/2011

Journal:

Year:

2011

Language:

english

File:

PDF, 580 KB

english, 2011

25

Preview: ChemMedChem 8/2011

Journal:

Year:

2011

Language:

english

File:

PDF, 97 KB

english, 2011

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