Volume 8; Issue 3

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ChemMedChem
Volume 8; Issue 3

ChemMedChem

Volume 8; Issue 3

1

Modern Subunit Vaccines: Development, Components, and Research Opportunities

Moyle, Peter Michael, Toth, Istvan

Journal:

Year:

2013

Language:

english

File:

PDF, 1.97 MB

english, 2013

2

Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19 F Ligand-and 15 N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series

Goudreau, Nathalie, Coulombe, René, Faucher, Anne-Marie, Grand-Maître, Chantal, Lacoste, Jean-Eric, Lemke, Christopher T., Malenfant, Eric, Bousquet, Yves, Fader, Lee, Simoneau, Bruno, Mercier, Jean-F

Journal:

Year:

2013

Language:

english

File:

PDF, 1.90 MB

english, 2013

3

Synthesis and Biological Evaluation of Purine 2′-Fluoro-2′-deoxyriboside ProTides as Anti-influenza Virus Agents

Meneghesso, Silvia, Vanderlinden, Evelien, Brancale, Andrea, Balzarini, Jan, Naesens, Lieve, McGuigan, Christopher

Journal:

Year:

2013

Language:

english

File:

PDF, 910 KB

english, 2013

4

Novel Type II Fatty Acid Biosynthesis (FAS II) Inhibitors as Multistage Antimalarial Agents

Schrader, Florian C., Glinca, Serghei, Sattler, Julia M., Dahse, Hans-Martin, Afanador, Gustavo A., Prigge, Sean T., Lanzer, Michael, Mueller, Ann-Kristin, Klebe, Gerhard, Schlitzer, Martin

Journal:

Year:

2013

Language:

english

File:

PDF, 2.69 MB

english, 2013

5

Anti-Inflammatory Drug Discovery . Edited by Jeremy I. Levin and Stefan Laufer

Journal:

Year:

2013

Language:

english

File:

PDF, 205 KB

english, 2013

6

Carboxylic Acid (Bio)Isosteres in Drug Design

Ballatore, Carlo, Huryn, Donna M., Smith, Amos B.

Journal:

Year:

2013

Language:

english

File:

PDF, 482 KB

english, 2013

7

Identification of a Small-Molecule Inhibitor of HIV-1 Assembly that Targets the Phosphatidylinositol (4,5)-bisphosphate Binding Site of the HIV-1 Matrix Protein

Zentner, Isaac, Sierra, Luz-Jeannette, Fraser, Ayesha K., Maciunas, Lina, Mankowski, Marie K., Vinnik, Andrei, Fedichev, Peter, Ptak, Roger G., Martín-García, Julio, Cocklin, Simon

Journal:

Year:

2013

Language:

english

File:

PDF, 661 KB

english, 2013

8

Efficient Stacking on Protein Amide Fragments

Harder, Michael, Kuhn, Bernd, Diederich, François

Journal:

Year:

2013

Language:

english

File:

PDF, 995 KB

english, 2013

9

Cover Picture: Efficient Stacking on Protein Amide Fragments (ChemMedChem 3/2013)

Harder, Michael, Kuhn, Bernd, Diederich, François

Journal:

Year:

2013

Language:

english

File:

PDF, 537 KB

english, 2013

10

Structure-Activity Relationships of Glucosamine-Derived Glycerolipids: the Role of the Anomeric Linkage, the Cationic Charge and the Glycero Moiety on the Antitumor Activity

Xu, Yaozu, Ogunsina, Makanjuola, Samadder, Pranati, Arthur, Gilbert, Schweizer, Frank

Journal:

Year:

2013

Language:

english

File:

PDF, 1.24 MB

english, 2013

11

Design, Synthesis, in vitro MAO-B Inhibitory Evaluation, and Computational Studies of Some 6-Nitrobenzothiazole-Derived Semicarbazones

Tripathi, Rati K. P., Goshain, Omprakash, Ayyannan, Senthil Raja

Journal:

Year:

2013

Language:

english

File:

PDF, 1.02 MB

english, 2013

12

Polycyclic Peptide Therapeutics

Baeriswyl, Vanessa, Heinis, Christian

Journal:

Year:

2013

Language:

english

File:

PDF, 1.37 MB

english, 2013

13

Optimization of Marine Triterpene Sipholenols as Inhibitors of Breast Cancer Migration and Invasion

Foudah, Ahmed I., Jain, Sandeep, Busnena, Belnaser A., El Sayed, Khalid A.

Journal:

Year:

2013

Language:

english

File:

PDF, 1.58 MB

english, 2013

14

Computational Studies Identifying Entry Inhibitor Scaffolds Targeting the Phe 43 Cavity of HIV-1 gp120

Tintori, Cristina, Selvaraj, Manikandan, Badia, Roger, Clotet, Bonaventura, Esté, José A., Botta, Maurizio

Journal:

Year:

2013

Language:

english

File:

PDF, 3.36 MB

english, 2013

15

Back Cover: Computational Studies Identifying Entry Inhibitor Scaffolds Targeting the Phe 43 Cavity of HIV-1 gp120 (ChemMedChem 3/2013)

Tintori, Cristina, Selvaraj, Manikandan, Badia, Roger, Clotet, Bonaventura, Esté, José A., Botta, Maurizio

Journal:

Year:

2013

File:

PDF, 1.15 MB

2013

16

Inside Cover: Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19 F Ligand-and 15 N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series (ChemMedChem 3/2013)

Goudreau, Nathalie, Coulombe, René, Faucher, Anne-Marie, Grand-Maître, Chantal, Lacoste, Jean-Eric, Lemke, Christopher T., Malenfant, Eric, Bousquet, Yves, Fader, Lee, Simoneau, Bruno, Mercier, Jean-F

Journal:

Year:

2013

File:

PDF, 968 KB

2013

17

Novel Schiff-Base-Derived FabH Inhibitors with Dioxygenated Rings as Antibiotic Agents

Zhou, Yang, Du, Qian-Ru, Sun, Jian, Li, Jing-Ran, Fang, Fei, Li, Dong-Dong, Qian, Yong, Gong, Hai-Bin, Zhao, Jing, Zhu, Hai-Liang

Journal:

Year:

2013

Language:

english

File:

PDF, 1010 KB

english, 2013

18

Targets and Emerging Therapies for Schizophrenia . Edited by Jeffrey S. Albert and Michael W. Wood

Journal:

Year:

2013

Language:

english

File:

PDF, 129 KB

english, 2013

19

Graphical Abstract: ChemMedChem 3/2013

Journal:

Year:

2013

Language:

english

File:

PDF, 3.19 MB

english, 2013

20

A “Clickable” MTX Reagent as a Practical Tool for Profiling Small-Molecule-Intracellular Target Interactions via MASPIT

Risseeuw, Martijn D. P., De Clercq, Dries J. H., Lievens, Sam, Hillaert, Ulrik, Sinnaeve, Davy, Van den Broeck, Freya, Martins, José C., Tavernier, Jan, Van Calenbergh, Serge

Journal:

Year:

2013

Language:

english

File:

PDF, 527 KB

english, 2013

21

Applications of Transition Metal Catalysis in Drug Discovery and Development . Edited by Matthew L. Crawley and Barry M. Trost

Farina, Vittorio

Journal:

Year:

2013

Language:

english

File:

PDF, 258 KB

english, 2013

22

A Combination Strategy to Inhibit Pim-1: Synergism between Noncompetitive and ATP-Competitive Inhibitors

Mori, Mattia, Tintori, Cristina, Christopher, Robert Selwyne Arul, Radi, Marco, Schenone, Silvia, Musumeci, Francesca, Brullo, Chiara, Sanità, Patrizia, Delle Monache, Simona, Angelucci, Adriano, Kiss

Journal:

Year:

2013

Language:

english

File:

PDF, 1.18 MB

english, 2013

23

Spotlights on our sister journals: ChemMedChem 3/2013

Journal:

Year:

2013

Language:

english

File:

PDF, 1.38 MB

english, 2013