Volume 8; Issue 6

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ChemMedChem
Volume 8; Issue 6

ChemMedChem

Volume 8; Issue 6

1

MAO Inhibitory Activity of 2-Arylbenzofurans versus 3-Arylcoumarins: Synthesis, in vitro Study, and Docking Calculations

Ferino, Giulio, Cadoni, Enzo, Matos, Maria João, Quezada, Elias, Uriarte, Eugenio, Santana, Lourdes, Vilar, Santiago, Tatonetti, Nicholas P., Yáñez, Matilde, Viña, Dolores, Picciau, Carmen, Serra, Sil

Journal:

Year:

2013

Language:

english

File:

PDF, 2.03 MB

english, 2013

2

Synthesis and Anti-herpetic Activity of Phosphoramidate ProTides

Maiti, Munmun, Persoons, Leentje, Andrei, Graciela, Snoeck, Robert, Balzarini, Jan, Herdewijn, Piet

Journal:

Year:

2013

Language:

english

File:

PDF, 526 KB

english, 2013

3

Synthesis, Antitumor Evaluation and Docking Study of Novel 4-Anilinoquinazoline Derivatives as Potential Epidermal Growth Factor Receptor (EGFR) Inhibitors

Rao, Guo-Wu, Xu, Geng-Jie, Wang, Jian, Jiang, Xu-Liang, Li, Hai-Bo

Journal:

Year:

2013

Language:

english

File:

PDF, 1.33 MB

english, 2013

4

Optimization of Triazine Nitriles as Rhodesain Inhibitors: Structure-Activity Relationships, Bioisosteric Imidazopyridine Nitriles, and X-ray Crystal Structure Analysis with Human Cathepsin L

Ehmke, Veronika, Winkler, Edwin, Banner, David W., Haap, Wolfgang, Schweizer, W. Bernd, Rottmann, Matthias, Kaiser, Marcel, Freymond, Céline, Schirmeister, Tanja, Diederich, François

Journal:

Year:

2013

Language:

english

File:

PDF, 897 KB

english, 2013

5

A Facile Hydroxyindole Carboxylic Acid Based Focused Library Approach for Potent and Selective Inhibitors of Mycobacterium Protein Tyrosine Phosphatase B

Zeng, Li-Fan, Xu, Jie, He, Yantao, He, Rongjun, Wu, Li, Gunawan, Andrea M., Zhang, Zhong-Yin

Journal:

Year:

2013

Language:

english

File:

PDF, 542 KB

english, 2013

6

Design, Synthesis, and Antibacterial Activity of Demethylvancomycin Analogues against Drug-Resistant Bacteria

Chang, Jun, Zhang, Si-Ji, Jiang, Yong-Wei, Xu, Liang, Yu, Jian-Ming, Zhou, Wen-Jiang, Sun, Xun

Journal:

Year:

2013

Language:

english

File:

PDF, 483 KB

english, 2013

7

Graphical Abstract: ChemMedChem 6/2013

Journal:

Year:

2013

Language:

english

File:

PDF, 3.10 MB

english, 2013

8

Bioisosteres in Medicinal Chemistry . Edited by Nathan Brown

Journal:

Year:

2013

Language:

english

File:

PDF, 291 KB

english, 2013

9

Synthesis and Evaluation of Water-Soluble Prodrugs of Ursodeoxycholic Acid (UDCA), an Anti-apoptotic Bile Acid

Dosa, Peter I., Ward, Tim, Castro, Rui E., Rodrigues, Cecília M. P., Steer, Clifford J.

Journal:

Year:

2013

Language:

english

File:

PDF, 467 KB

english, 2013

10

Discovery and Characterization of ACT-335827, an Orally Available, Brain Penetrant Orexin Receptor Type 1 Selective Antagonist

Steiner, Michel A., Gatfield, John, Brisbare-Roch, Catherine, Dietrich, Hendrik, Treiber, Alexander, Jenck, Francois, Boss, Christoph

Journal:

Year:

2013

Language:

english

File:

PDF, 342 KB

english, 2013

11

From a Multipotent Stilbene to Soluble Epoxide Hydrolase Inhibitors with Antiproliferative Properties

Buscató, Estel.la, Büttner, Dominik, Brüggerhoff, Astrid, Klingler, Franca-Maria, Weber, Julia, Scholz, Bastian, Živković, Aleksandra, Marschalek, Rolf, Stark, Holger, Steinhilber, Dieter, Bode, Helge

Journal:

Year:

2013

Language:

english

File:

PDF, 578 KB

english, 2013

12

Structure-Activity Relationships of Quinoxaline-Based 5-HT 3 A and 5-HT 3 AB Receptor-Selective Ligands

Thompson, Andrew J., Verheij, Mark H. P., van Muijlwijk-Koezen, Jacqueline E., Lummis, Sarah C. R., Leurs, Rob, de Esch, Iwan J. P.

Journal:

Year:

2013

Language:

english

File:

PDF, 636 KB

english, 2013

13

Radiolabeled Heterobivalent Peptidic Ligands: an Approach with High Future Potential for in vivo Imaging and Therapy of Malignant Diseases

Fischer, Gabriel, Schirrmacher, Ralf, Wängler, Björn, Wängler, Carmen

Journal:

Year:

2013

Language:

english

File:

PDF, 608 KB

english, 2013

14

Rhenium Complexes with Visible-Light-Induced Anticancer Activity

Kastl, Anja, Dieckmann, Sandra, Wähler, Kathrin, Völker, Timo, Kastl, Lena, Merkel, Anna Lena, Vultur, Adina, Shannan, Batool, Harms, Klaus, Ocker, Matthias, Parak, Wolfgang J., Herlyn, Meenhard, Megg

Journal:

Year:

2013

Language:

english

File:

PDF, 2.18 MB

english, 2013

15

An Efficient Bioorthogonal Strategy Using CuAAC Click Chemistry for Radiofluorinations of SNEW Peptides and the Role of Copper Depletion

Pretze, Marc, Kuchar, Manuela, Bergmann, Ralf, Steinbach, Jörg, Pietzsch, Jens, Mamat, Constantin

Journal:

Year:

2013

Language:

english

File:

PDF, 744 KB

english, 2013

16

Synthesis and in vitro Evaluation of West Nile Virus Protease Inhibitors Based on the 2-{6-[2-(5-Phenyl-4 H -{1,2,4]triazol-3-ylsulfanyl)acetylamino]benzothiazol-2-ylsulfanyl}acetamide Scaffold

Samanta, Sanjay, Lim, Ting Liang, Lam, Yulin

Journal:

Year:

2013

Language:

english

File:

PDF, 797 KB

english, 2013

17

Potent Inhibitors of Phosphatidylinositol 3 (PI3) Kinase that have Antiproliferative Activity Only When Delivered as Prodrug Forms

O'Brien, Nathan J., Amran, Syazwani, Medan, Jelena, Cleary, Ben, Deady, Leslie W., Jennings, Ian G., Thompson, Philip E., Abbott, Belinda M.

Journal:

Year:

2013

Language:

english

File:

PDF, 306 KB

english, 2013

18

Cover Picture: From a Multipotent Stilbene to Soluble Epoxide Hydrolase Inhibitors with Antiproliferative Properties (ChemMedChem 6/2013)

Buscató, Estel.la, Büttner, Dominik, Brüggerhoff, Astrid, Klingler, Franca-Maria, Weber, Julia, Scholz, Bastian, Živković, Aleksandra, Marschalek, Rolf, Stark, Holger, Steinhilber, Dieter, Bode, Helge

Journal:

Year:

2013

Language:

english

File:

PDF, 614 KB

english, 2013

19

Cancer Epigenetics: Biomolecular Therapeutics for Human Cancer . Edited by Antonio Giordano and Marcella Macaluso

Journal:

Year:

2013

Language:

english

File:

PDF, 119 KB

english, 2013

20

Selective Bisubstrate Inhibitors with Sub-nanomolar Affinity for Protein Kinase Pim-1

Ekambaram, Ramesh, Enkvist, Erki, Vaasa, Angela, Kasari, Marje, Raidaru, Gerda, Knapp, Stefan, Uri, Asko

Journal:

Year:

2013

Language:

english

File:

PDF, 388 KB

english, 2013

21

Design, Synthesis and Biological Evaluation of Trimethine Cyanine Dyes as Fluorescent Probes for the Detection of Tau Fibrils in Alzheimer’s Disease Brain and Olfactory Epithelium

Gu, Jiamin, Anumala, Upendra Rao, Heyny-von Haußen, Roland, Hölzer, Jana, Goetschy-Meyer, Valérie, Mall, Gerhard, Hilger, Ingrid, Czech, Christian, Schmidt, Boris

Journal:

Year:

2013

Language:

english

File:

PDF, 683 KB

english, 2013

22

Inside Cover: Design, Synthesis, and Antibacterial Activity of Demethylvancomycin Analogues against Drug-Resistant Bacteria (ChemMedChem 6/2013)

Chang, Jun, Zhang, Si-Ji, Jiang, Yong-Wei, Xu, Liang, Yu, Jian-Ming, Zhou, Wen-Jiang, Sun, Xun

Journal:

Year:

2013

File:

PDF, 974 KB

2013

23

Back Cover: Structure-Activity Relationships of Quinoxaline-Based 5-HT 3 A and 5-HT 3 AB Receptor-Selective Ligands (ChemMedChem 6/2013)

Thompson, Andrew J., Verheij, Mark H. P., van Muijlwijk-Koezen, Jacqueline E., Lummis, Sarah C. R., Leurs, Rob, de Esch, Iwan J. P.

Journal:

Year:

2013

File:

PDF, 1.04 MB

2013

24

Spotlights on our sister journals: ChemMedChem 6/2013

Journal:

Year:

2013

Language:

english

File:

PDF, 1.66 MB

english, 2013

25

Graphical Abstract: ChemMedChem 6/2013

Journal:

Year:

2013

Language:

english

File:

PDF, 3.10 MB

english, 2013

26

Innovations in Biomolecular Modeling and Simulations . Edited by Tamar Schlick

Orozco, Modesto

Journal:

Year:

2013

Language:

english

File:

PDF, 343 KB

english, 2013

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