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Volume 100

European Journal of Medicinal Chemistry

Volume 100

1

Design, synthesis and biological evaluation of small molecules as potent glucosidase inhibitors

Hati, Santanu, Madurkar, Sanjay M., Bathula, Chandramohan, Thulluri, Chiranjeevi, Agarwal, Rahul, Siddiqui, Faiza Amber, Dangi, Poonam, Adepally, Uma, Singh, Ashutosh, Singh, Shailja, Sen, Subhabrata

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 4.64 MB

english, 2015

2

Synthesis of 1H-1,2,3-triazole linked aryl(arylamidomethyl) – dihydrofurocoumarin hybrids and analysis of their cytotoxicity

Lipeeva, Alla V., Pokrovsky, Mikhail A., Baev, Dmitry S., Shakirov, Makhmut M., Bagryanskaya, Irina Y., Tolstikova, Tatijana G., Pokrovsky, Andrey G., Shults, Elvira E.

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.04 MB

english, 2015

3

Identification of a potent 5-phenyl-thiazol-2-ylamine-based inhibitor of FLT3 with activity against drug resistance-conferring point mutations

Chen, Chiung-Tong, Hsu, John T.-A., Lin, Wen-Hsing, Lu, Cheng-Tai, Yen, Shih-Chieh, Hsu, Tsu, Huang, Yu-Ling, Song, Jen-Shin, Chen, Chun-Hwa, Chou, Ling-Hui, Yen, Kuei-Jung, Chen, Ching-Ping, Kuo, Po-

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.88 MB

english, 2015

4

Synthesis and antiproliferative activity of imidazo[1,2-a]pyrimidine Mannich bases

Aeluri, Raghunath, Alla, Manjula, Polepalli, Sowjanya, Jain, Nishant

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 2.15 MB

english, 2015

5

Isoquinoline derivatives Zn(II)/Ni(II) complexes: Crystal structures, cytotoxicity, and their action mechanism

Huang, Ke-Bin, Mo, Hui-Yan, Chen, Zhen-Feng, Wei, Jian-Hua, Liu, Yan-Cheng, Liang, Hong

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.32 MB

english, 2015

6

Indoline ureas as potential anti-hepatocellular carcinoma agents targeting VEGFR-2: Synthesis, in vitro biological evaluation and molecular docking

Eldehna, Wagdy M., Fares, Mohamed, Ibrahim, Hany S., Aly, Mohamed H., Zada, Suher, Ali, Mamdouh M., Abou-Seri, Sahar M., Abdel-Aziz, Hatem A., Abou El Ella, Dalal A.

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 4.28 MB

english, 2015

7

Thiosemicarbazones as Aedes aegypti larvicidal

da Silva, João Bosco P., Navarro, Daniela Maria do A.F., da Silva, Aluizio G., Santos, Geanne K.N., Dutra, Kamilla A., Moreira, Diogo Rodrigo, Ramos, Mozart N., Espíndola, José Wanderlan P., de Olivei

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 5.48 MB

english, 2015

8

Styryl-N-phenyl-N′-(2-chloroethyl)ureas and styrylphenylimidazolidin-2-ones as new potent microtubule-disrupting agents using combretastatin A-4 as model

Gagné-Boulet, Mathieu, Fortin, Sébastien, Lacroix, Jacques, Lefebvre, Carole-Anne, Côté, Marie-France, C.-Gaudreault, René

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.33 MB

english, 2015

9

Ferrocene-pyrimidine conjugates: Synthesis, electrochemistry, physicochemical properties and antiplasmodial activities

Chopra, Rakesh, de Kock, Carmen, Smith, Peter, Chibale, Kelly, Singh, Kamaljit

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 4.68 MB

english, 2015

10

Design, synthesis and characterization of dual inhibitors against new targets FabG4 and HtdX of Mycobacterium tuberculosis

Banerjee, Deb Ranjan, Biswas, Rupam, Das, Amit K., Basak, Amit

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 5.80 MB

english, 2015

11

Structure-activity relationship of hybrids of Cinchona alkaloids and bile acids with in vitro antiplasmodial and antitrypanosomal activities

Leverrier, Aurélie, Bero, Joanne, Cabrera, Julián, Frédérich, Michel, Quetin-Leclercq, Joëlle, Palermo, Jorge A.

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 460 KB

english, 2015

12

Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design

Pieroni, Marco, Wan, Baojie, Zuliani, Valentina, Franzblau, Scott G., Costantino, Gabriele, Rivara, Mirko

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 647 KB

english, 2015

13

Aryl H-Phosphonates 18. Synthesis, properties, and biological activity of 2′,3′-dideoxynucleoside (N-heteroaryl)phosphoramidates of increased lipophilicity

Kolodziej, Krystian, Romanowska, Joanna, Stawinski, Jacek, Boryski, Jerzy, Dabrowska, Aleksandra, Lipniacki, Andrzej, Piasek, Andrzej, Kraszewski, Adam, Sobkowski, Michal

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 6.80 MB

english, 2015

14

Recent progress in the drug development of coumarin derivatives as potent antituberculosis agents

Keri, Rangappa S., B.S., Sasidhar, Nagaraja, Bhari Mallanna, Santos, M. Amélia

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 730 KB

english, 2015

15

TRPV1 modulators: Synthesis and in vitro evaluation of 1-heteroaryl piperidinecarboxamide and piperazinylurea derivatives

Congiu, Cenzo, Onnis, Valentina, Balboni, Gianfranco, Schiano-Moriello, Aniello, Di Marzo, Vincenzo, De Petrocellis, Luciano

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.58 MB

english, 2015

16

Design, synthesis and antiproliferative activities of novel benzamides derivatives as HDAC inhibitors

Li, Yanyang, Wang, Yongzhen, Xie, Ning, Xu, Ming, Qian, Pengyu, Zhao, Yanjin, Li, Shuxin

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.44 MB

english, 2015

17

11-Keto-boswellic acid derived amides and monodesmosidic saponins induce apoptosis in breast and cervical cancers cells

Csuk, René, Barthel-Niesen, Anja, Barthel, Alexander, Schäfer, Renate, Al-Harrasi, Ahmed

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 949 KB

english, 2015

18

Novel cajaninstilbene acid derivatives as antibacterial agents

Geng, Zhi-Zhong, Zhang, Jian-Jun, Lin, Jing, Huang, Mei-Yan, An, Lin-Kun, Zhang, Hong-Bin, Sun, Ping-Hua, Ye, Wen-Cai, Chen, Wei-Min

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 881 KB

english, 2015

19

1,5-Diarylpyrazole and vanillin hybrids: Synthesis, biological activity and DFT studies

Hernández-Vázquez, Eduardo, Castañeda-Arriaga, Romina, Ramírez-Espinosa, Juan José, Medina-Campos, Omar Noel, Hernández-Luis, Francisco, Chaverri, José Pedraza, Estrada-Soto, Samuel

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.59 MB

english, 2015

20

Development of bis-thiazoles as inhibitors of triosephosphate isomerase from Trypanosoma cruzi. Identification of new non-mutagenic agents that are active in vivo

Álvarez, Guzmán, Martínez, Jennyfer, Varela, Javier, Birriel, Estefania, Cruces, Eugenia, Gabay, Martín, Leal, Sandra M., Escobar, Patricia, Aguirre-López, Beatriz, Cabrera, Nallely, Tuena de Gómez-Pu

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.15 MB

english, 2015

21

Exploring the size adaptability of the B ring binding zone of the colchicine site of tubulin with para-nitrogen substituted isocombretastatins

Jiménez, Carmen, Ellahioui, Younes, Álvarez, Raquel, Aramburu, Laura, Riesco, Alejandra, González, Myriam, Vicente, Alba, Dahdouh, Abdelaziz, Ibn Mansour, Ahmed, Jiménez, Carlos, Martín, Diego, Sarmie

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.68 MB

english, 2015

22

New systematically modified vesamicol analogs and their affinity and selectivity for the vesicular acetylcholine transporter – A critical examination of the lead structure

Barthel, Claudia, Sorger, Dietlind, Deuther-Conrad, Winnie, Scheunemann, Matthias, Schweiger, Stephanie, Jäckel, Petra, Roghani, Ali, Steinbach, Jörg, Schüürmann, Gerrit, Sabri, Osama, Brust, Peter, W

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.40 MB

english, 2015

23

Synthesis and evaluation of thymidine kinase 1-targeting carboranyl pyrimidine nucleoside analogs for boron neutron capture therapy of cancer

Agarwal, Hitesh K., Khalil, Ahmed, Ishita, Keisuke, Yang, Weilian, Nakkula, Robin J., Wu, Lai-Chu, Ali, Tehane, Tiwari, Rohit, Byun, Youngjoo, Barth, Rolf F., Tjarks, Werner

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1019 KB

english, 2015

24

Design, synthesis and in vitro trypanocidal and leishmanicidal activities of novel semicarbazone derivatives

Alves, Marina A., de Queiroz, Aline C., Alexandre-Moreira, Magna Suzana, Varela, Javier, Cerecetto, Hugo, González, Mercedes, Doriguetto, Antonio C., Landre, Iara M., Barreiro, Eliezer J., Lima, Lídia

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 988 KB

english, 2015

25

Synthesis and cancer cell growth inhibitory activity of icaritin derivatives

Wang, Chen, Wu, Ping, Shi, Jing-Fang, Jiang, Zi-Hua, Wei, Xiao-Yi

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 596 KB

english, 2015

26

Living on pyrrolic foundations – Advances in natural and artificial bioactive pyrrole derivatives

Domagala, Anna, Jarosz, Tomasz, Lapkowski, Mieczyslaw

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.04 MB

english, 2015

27

Editorial board

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 56 KB

english, 2015

28

Graphical contents list

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.71 MB

english, 2015